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上海药物研究所 [50]
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期刊论文 [207]
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Galaxy morphology classification based on Convolutional vision Transformer (CvT)
期刊论文
OAI收割
ASTRONOMY & ASTROPHYSICS, 2024, 卷号: 683
作者:
Cao, Jie
;
Xu, Tingting
;
Deng, Yuhe
;
Deng, Linhua
;
Yang, Mingcun
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/04/08
methods: data analysis
techniques: image processing
Galaxy: general
Structure-Based Ligand Discovery Targeting the Transmembrane Domain of Frizzled Receptor FZD7
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 14
作者:
Li, Cuixia
;
Wu, Yiran
;
Wang, Wenli
;
Xu, Lu
;
Zhou, Yan
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/10/17
D3CARP: a comprehensive platform with multiple-conformation based docking, ligand similarity search and deep learning approaches for target prediction and virtual screening
期刊论文
OAI收割
COMPUTERS IN BIOLOGY AND MEDICINE, 2023, 卷号: 164, 页码: 8
作者:
Shi, Yulong
;
Zhang, Xinben
;
Yang, Yanqing
;
Cai, Tingting
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2023/10/17
Target prediction
Virtual screening
Molecular docking
Ligand similarity search
Deep learning
Discovery of 2-Aminopyrimidine Derivatives as Potent Dual FLT3/CHK1 Inhibitors with Significantly Reduced hERG Inhibitory Activities
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 23
作者:
Li, Xuemei
;
Wang, Peipei
;
Wang, Chang
;
Jin, Tingting
;
Xu, Ran
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/10/17
Galaxy morphology classification using multiscale convolution capsule network
期刊论文
OAI收割
MONTHLY NOTICES OF THE ROYAL ASTRONOMICAL SOCIETY, 2023, 卷号: 523, 期号: 1, 页码: 488-497
作者:
Li, Guangping
;
Xu, Tingting
;
Li, Liping
;
Gao, Xianjun
;
Liu, Zhijing
  |  
收藏
  |  
浏览/下载:59/0
  |  
提交时间:2023/07/03
methods: data analysis
techniques: image processing
galaxies: general
Effect of cold rolling on microstructure, texture, and tensile properties of a Ni-Fe-based superalloy
期刊论文
OAI收割
JOURNAL OF ALLOYS AND COMPOUNDS, 2023, 卷号: 937, 页码: 14
作者:
Wang, Jiaqi
;
Cheng, Sihan
;
Wu, Yunsheng
;
Wang, Tingting
;
Qin, Xuezhi
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/05/09
Ni-Fe-based superalloy
Cold rolling
Microstructure
Texture
Strength
Deformation twinning
Dual inhibition of CHK1/FLT3 enhances cytotoxicity and overcomes adaptive and acquired resistance in FLT3-ITD acute myeloid leukemia
期刊论文
OAI收割
LEUKEMIA, 2022, 页码: 11
作者:
Jiang, Kailong
;
Li, Xuemei
;
Wang, Chang
;
Hu, Xiaobei
;
Wang, Peipei
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/04/10
A potent PGK1 antagonist reveals PGK1 regulates the production of IL-1 beta and IL-6
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2022, 卷号: 12, 期号: 11, 页码: 4180-4192
作者:
Liao, Liping
;
Dang, Wenzhen
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/04/10
Glycolysis
Phosphoglycerate kinase 1
Macrophages
NRF2
Inflammation
Exploring the Binding Affinity and Mechanism between ACE2 and the Trimers of Delta and Omicron Spike Proteins by Molecular Dynamics Simulation and Bioassay
期刊论文
OAI收割
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2022, 页码: 11
作者:
Zhou, Liping
;
Liu, Tingting
;
Mo, Mengxia
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2022/11/11
Artemisinin analog SM934 alleviates epithelial barrier dysfunction via inhibiting apoptosis and caspase-1-mediated pyroptosis in experimental colitis
期刊论文
OAI收割
FRONTIERS IN PHARMACOLOGY, 2022, 卷号: 13, 页码: 18
作者:
Shao, Meijuan
;
Yan, Yuxi
;
Zhu, Fenghua
;
Yang, Xiaoqian
;
Qi, Qing
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2022/11/11
SM934
colitis
intestinal epithelial barrier
apoptosis
pyroptosis
NLRP3/caspase-1/GSDMD
MAPK/NF-kB