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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [9]
采集方式
OAI收割 [9]
内容类型
期刊论文 [9]
发表日期
2018 [9]
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发表日期:2018
内容类型:期刊论文
专题:上海药物研究所
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Rational design of 5-((1H-imidazol-1-yl)methyl)quinolin-8-ol derivatives as novel bromodomain-containing protein 4 inhibitors
期刊论文
OAI收割
European journal of medicinal chemistry, 2018, 卷号: 163, 页码: 281-294
作者:
Xing, Jing
;
Zhang, Rukang
;
Jiang, Xiangrui
;
Hu, Tianwen
;
Wang, Xinjun
  |  
收藏
  |  
浏览/下载:86/0
  |  
提交时间:2019/01/08
Development and evaluation of a novel series of Nitroxoline-derived BET inhibitors with antitumor activity in renal cell carcinoma
期刊论文
OAI收割
ONCOGENESIS, 2018, 卷号: 7
作者:
Chen, Wei
;
Zhang, Hao
;
Chen, Zhifeng
;
Jiang, Hao
;
Liao, Liping
  |  
收藏
  |  
浏览/下载:108/0
  |  
提交时间:2019/01/08
Immune modulation of a lipid-soluble extract of Pinellia pedatisecta Schott in the tumor microenvironment of an HPV+ tumor-burdened mouse model
期刊论文
OAI收割
JOURNAL OF ETHNOPHARMACOLOGY, 2018, 卷号: 225, 页码: 103-115
作者:
Huang, Haixia
;
Zhang, Mingxing
;
Yao, Sheng
;
Zhang, Meng
;
Peng, Jing
  |  
收藏
  |  
浏览/下载:69/0
  |  
提交时间:2019/01/08
Pinellia pedatisecta extract (PE)
Cervical cancer
HPV+ tumor
TC-1 cell line
Helper T (Th) cellular immunity
CUDC-907 displays potent antitumor activity against human pancreatic adenocarcinoma in vitro and in vivo through inhibition of HDAC6 to downregulate c-Myc expression
期刊论文
OAI收割
Acta pharmacologica Sinica, 2018
作者:
Fu, Xu-Hong
;
Zhang, Xiong
;
Yang, Hong
;
Xu, Xiao-Wei
;
Hu, Zong-Long
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2019/01/08
Pharmacological inhibition of dihydroorotate dehydrogenase induces apoptosis and differentiation in acute myeloid leukemia cells
期刊论文
OAI收割
HAEMATOLOGICA, 2018, 卷号: 103, 期号: 9, 页码: 1472-1483
作者:
Wu, Dang
;
Wang, Wanyan
;
Chen, Wuyan
;
Lian, Fulin
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2019/01/08
Design, synthesis and biological evaluation of benzo[cd]indo1-2(1H)-ones derivatives as BRD4 inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 264-273
作者:
Feng, Yuxin
;
Xiao, Senhao
;
Chen, Yantao
;
Jiang, Hao
;
Liu, Na
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2019/01/08
Benzo[cd]indol-2(1H)-one
Sulfonamide
BRD4 inhibitor
Bromodomain and extra-terminal domain
Acetyl-lysine binding pocket
Structure-based optimization of a series of selective BET inhibitors containing aniline or indoline groups
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 页码: 156-175
作者:
Hu, Jianping
;
Wang, Yingqing
;
Li, Yanlian
;
Cao, Danyan
;
Xu, Lin
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2019/01/08
BRD4
BI2536
Indoline
WPF binders
c-Myc
PD-L1
Targeting death receptors for drug-resistant cancer therapy: Codelivery of pTRAIL and monensin using dual-targeting and stimuli-responsive self-assembling nanocomposites
期刊论文
OAI收割
BIOMATERIALS, 2018, 卷号: 158, 页码: 56-73
作者:
Xu, Fan
;
Zhong, Huihai
;
Chang, Ya
;
Li, Dongdong
;
Jin, Hongyue
  |  
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2019/01/08
TRAIL
Gene delivery
Monensin
Poly-gamma-glutamic acid
Death receptor
Drug resistance
A regulatory circuit HP1 gamma/miR-451a/c-Myc promotes prostate cancer progression
期刊论文
OAI收割
ONCOGENE, 2018, 卷号: 37, 期号: 4, 页码: 415-426
作者:
Chang, C.
;
Liu, J.
;
He, W.
;
Qu, M.
;
Huang, X.
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/01/08