中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共20条,第1-10条 帮助

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Discovery of a brain-permeable bromodomain and extra terminal domain (BET) inhibitor with selectivity for BD1 for the treatment of multiple sclerosis 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 14
作者:  
Chen, Xuetao;  Wu, Tingting;  Du, Zhiyan;  Kang, Wenjing;  Xu, Rujun
  |  收藏  |  浏览/下载:20/0  |  提交时间:2024/02/27
Screening and optimization of phage display cyclic peptides against the WDR5 WBM site 期刊论文  OAI收割
RSC MEDICINAL CHEMISTRY, 2023, 页码: 10
作者:  
Song, Lingyu;  Cao, Jiawen;  Chen, Lin;  Du, Zhiyan;  Zhang, Naixia
  |  收藏  |  浏览/下载:6/0  |  提交时间:2023/10/17
Discovery of 1H-Imidazo[4,5-b]pyridine Derivatives as Potent and Selective BET Inhibitors for the Management of Neuropathic Pain 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 13, 页码: 8725-8744
作者:  
Chen, Xuetao;  Cao, Danyan;  Liu, Chihong;  Meng, Fanying;  Zhang, Zijian
  |  收藏  |  浏览/下载:9/0  |  提交时间:2023/10/17
Structure-Based of a Series of NSD2-PWWP1 Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 13, 页码: 9459-9477
作者:  
Li, Na;  Yang, Hong;  Liu, Ke;  Zhou, Liwei;  Huang, Yuting
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/03/21
Structure-Based Discovery of Potent CARM1 Inhibitors for Solid Tumor and Cancer Immunology Therapy 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 22, 页码: 16650-16674
作者:  
Zhang, Zhuqing;  Guo, Zuhao;  Xu, Xiaowei;  Cao, Danyan;  Yang, Hong
  |  收藏  |  浏览/下载:25/0  |  提交时间:2022/06/15
Multi-omics characterization of WNT pathway reactivation to ameliorate BET inhibitor resistance in liver cancer cells 期刊论文  OAI收割
GENOMICS, 2021, 卷号: 113, 期号: 3, 页码: 1057-1069
作者:  
Liu, Yuwei;  Xue, Mengzhu;  Cao, Danyan;  Qin, Lihuai;  Wang, Ying
  |  收藏  |  浏览/下载:25/0  |  提交时间:2021/08/17
Phage-Display Based Discovery and Characterization of Peptide Ligands against WDR5 期刊论文  OAI收割
MOLECULES, 2021, 卷号: 26, 期号: 5, 页码: 12
作者:  
Cao, Jiawen;  Fan, Tiantian;  Li, Yanlian;  Du, Zhiyan;  Chen, Lin
  |  收藏  |  浏览/下载:65/0  |  提交时间:2021/05/24
Rational Design and Evaluation of 6-(Pyrimidin-2-ylamino)-3,4-dihydroquinoxalin-2(1H)-ones as Polypharmacological Inhibitors of BET and Kinases 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 17, 页码: 9787-9802
作者:  
Lv, Kaikai;  Chen, Weicong;  Chen, Danqi;  Mou, Jie;  Zhang, Huijie
  |  收藏  |  浏览/下载:22/0  |  提交时间:2020/12/21
Structure-Based Discovery and Development of a Series of Potent and Selective Bromodomain and Extra-Terminal Protein Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 18, 页码: 8642-8663
作者:  
Hu, Jianping;  Tian, Chang-Qing;  Damaneh, Mohammadali Soleimani;  Li, Yanlian;  Cao, Danyan
  |  收藏  |  浏览/下载:34/0  |  提交时间:2020/07/01
Design and Synthesis of Potent, Selective Inhibitors of Protein Arginine Methyltransferase 4 against Acute Myeloid Leukemia 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 11, 页码: 5414-5433
作者:  
Guo, Zuhao;  Zhang, Zhuqing;  Yang, Hong;  Cao, Danyan;  Xu, Xiaowei
  |  收藏  |  浏览/下载:61/0  |  提交时间:2020/07/01