中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [18]
上海应用物理研究所 [1]
上海硅酸盐研究所 [1]
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OAI收割 [20]
内容类型
期刊论文 [20]
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2024 [1]
2023 [2]
2022 [1]
2021 [3]
2020 [1]
2019 [3]
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Discovery of a brain-permeable bromodomain and extra terminal domain (BET) inhibitor with selectivity for BD1 for the treatment of multiple sclerosis
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 14
作者:
Chen, Xuetao
;
Wu, Tingting
;
Du, Zhiyan
;
Kang, Wenjing
;
Xu, Rujun
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/02/27
BET
BD1
Bromodomain
Brain-permeable
Multiple sclerosis
Screening and optimization of phage display cyclic peptides against the WDR5 WBM site
期刊论文
OAI收割
RSC MEDICINAL CHEMISTRY, 2023, 页码: 10
作者:
Song, Lingyu
;
Cao, Jiawen
;
Chen, Lin
;
Du, Zhiyan
;
Zhang, Naixia
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2023/10/17
Discovery of 1H-Imidazo[4,5-b]pyridine Derivatives as Potent and Selective BET Inhibitors for the Management of Neuropathic Pain
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 13, 页码: 8725-8744
作者:
Chen, Xuetao
;
Cao, Danyan
;
Liu, Chihong
;
Meng, Fanying
;
Zhang, Zijian
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/10/17
Structure-Based of a Series of NSD2-PWWP1 Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 13, 页码: 9459-9477
作者:
Li, Na
;
Yang, Hong
;
Liu, Ke
;
Zhou, Liwei
;
Huang, Yuting
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/03/21
Structure-Based Discovery of Potent CARM1 Inhibitors for Solid Tumor and Cancer Immunology Therapy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 22, 页码: 16650-16674
作者:
Zhang, Zhuqing
;
Guo, Zuhao
;
Xu, Xiaowei
;
Cao, Danyan
;
Yang, Hong
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2022/06/15
Multi-omics characterization of WNT pathway reactivation to ameliorate BET inhibitor resistance in liver cancer cells
期刊论文
OAI收割
GENOMICS, 2021, 卷号: 113, 期号: 3, 页码: 1057-1069
作者:
Liu, Yuwei
;
Xue, Mengzhu
;
Cao, Danyan
;
Qin, Lihuai
;
Wang, Ying
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2021/08/17
Multi-omics
BET inhibitor responses
WNT pathway
Liver cancer
Precise therapy
Phage-Display Based Discovery and Characterization of Peptide Ligands against WDR5
期刊论文
OAI收割
MOLECULES, 2021, 卷号: 26, 期号: 5, 页码: 12
作者:
Cao, Jiawen
;
Fan, Tiantian
;
Li, Yanlian
;
Du, Zhiyan
;
Chen, Lin
  |  
收藏
  |  
浏览/下载:65/0
  |  
提交时间:2021/05/24
phage display
biopanning
WDR5
cocrystal structure
Rational Design and Evaluation of 6-(Pyrimidin-2-ylamino)-3,4-dihydroquinoxalin-2(1H)-ones as Polypharmacological Inhibitors of BET and Kinases
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 17, 页码: 9787-9802
作者:
Lv, Kaikai
;
Chen, Weicong
;
Chen, Danqi
;
Mou, Jie
;
Zhang, Huijie
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2020/12/21
Structure-Based Discovery and Development of a Series of Potent and Selective Bromodomain and Extra-Terminal Protein Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 18, 页码: 8642-8663
作者:
Hu, Jianping
;
Tian, Chang-Qing
;
Damaneh, Mohammadali Soleimani
;
Li, Yanlian
;
Cao, Danyan
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2020/07/01
Design and Synthesis of Potent, Selective Inhibitors of Protein Arginine Methyltransferase 4 against Acute Myeloid Leukemia
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 11, 页码: 5414-5433
作者:
Guo, Zuhao
;
Zhang, Zhuqing
;
Yang, Hong
;
Cao, Danyan
;
Xu, Xiaowei
  |  
收藏
  |  
浏览/下载:61/0
  |  
提交时间:2020/07/01