中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [55]
广州生物医药与健康研... [2]
昆明植物研究所 [2]
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期刊论文 [63]
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生物化学与分子生物学 [2]
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PROTAC Prodrug-Integrated Nanosensitizer for Potentiating Radiation Therapy of Cancer
期刊论文
OAI收割
ADVANCED MATERIALS, 2024, 页码: 12
作者:
Zhang, Shunan
;
Lai, Yi
;
Pan, Jiaxing
;
Saeed, Madiha
;
Li, Shiqin
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/04/09
active tumor targeting
nanosensitizer
PROTAC prodrug
radiation therapy
tumor microenvironment
Discovery of a brain-permeable bromodomain and extra terminal domain (BET) inhibitor with selectivity for BD1 for the treatment of multiple sclerosis
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 14
作者:
Chen, Xuetao
;
Wu, Tingting
;
Du, Zhiyan
;
Kang, Wenjing
;
Xu, Rujun
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/02/27
BET
BD1
Bromodomain
Brain-permeable
Multiple sclerosis
Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 18
作者:
Zhang, Jingyu
;
Duan, Haiting
;
Gui, Renzhao
;
Wu, Mingfei
;
Shen, Liteng
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/12/19
Acute myeloid leukemia
Bromodomain-containing protein 9
Proteolysis-targeting chimera
Orally bioavailable
Docking
Design, Construction, and Screening of Diversified Pyrimidine-Focused DNA-Encoded Libraries
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 14, 期号: 8, 页码: 1073-1078
作者:
Seydimemet, Mengnisa
;
Yang, Yixuan
;
Lv, Yuhan
;
Liu, Jiaxiang
;
Yan, Ziqin
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/10/17
DNA-encoded library technology
Pyrimidine-focusedDNA-encodedlibrary
BRD4
Affinity screening
Inhibitor
Discovery of 1H-Imidazo[4,5-b]pyridine Derivatives as Potent and Selective BET Inhibitors for the Management of Neuropathic Pain
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 13, 页码: 8725-8744
作者:
Chen, Xuetao
;
Cao, Danyan
;
Liu, Chihong
;
Meng, Fanying
;
Zhang, Zijian
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/10/17
Selective degradation of cellular BRD3 and BRD4-L promoted by PROTAC molecules in six cancer cell lines
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 254, 页码: 17
作者:
Yan, Ziqin
;
Lyu, Xilin
;
Lin, Dongze
;
Wu, Gaoxing
;
Gong, Yang
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2023/10/17
Cyclization strategy leads to highly potent Bromodomain and extra-terminal (BET) Bromodomain inhibitors for the treatment of acute liver injury
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 247, 页码: 13
作者:
Chen, Chao
;
Lu, Tian
;
Chen, Panyu
;
Li, Zizhou
;
Yang, Yaxi
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2023/04/10
BET Bromodomains
Acute liver injury
Anti-inflammatory activity
Inhibitors
Tetracyclic compounds
Design, synthesis, and biological evaluation of BRD4 degraders
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 78, 页码: 12
作者:
Ding, Mengyuan
;
Shao, Yingying
;
Sun, Danwen
;
Meng, Suorina
;
Zang, Yi
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/04/10
PROTAC
BRD4 degradation
Leukemia
Multiple myeloma
Pulmonary fibrosis
In-situ clickable prodrug nanoplatform locally activates T lymphocytes to potentiate cancer immunotherapy
期刊论文
OAI收割
NANO TODAY, 2022, 卷号: 47, 页码: 11
作者:
Hou, Bo
;
Ye, Jiayi
;
Li, Junhao
;
Xu, Zhiai
;
Yu, Haijun
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2023/04/10
Immune-excluded tumor
Extracellular matrix
In-situ click reaction
Prodrug nanoparticles
Immune resistance
Design and development of a novel series of oral bivalent BET inhibitors with potent anticancer activities
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 239, 页码: 13
作者:
Luo, Menglan
;
Wu, Qian
;
Yang, Yueyue
;
Sun, Lin
;
Huan, Xiajuan
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2022/08/30
BET inhibitor
BRD4
Bivalent inhibitor
Anticancer