中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
  • 上海药物研究所 [14]
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内容类型
发表日期
  • 2018 [14]
学科主题
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浏览/检索结果: 共14条,第1-10条 帮助

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Fragment-based drug discovery of triazole inhibitors to block PDEδ-RAS protein-protein interaction 期刊论文  OAI收割
European journal of medicinal chemistry, 2018, 卷号: 163, 页码: 597-609
作者:  
Chen, Danqi;  Chen, Yuehong;  Lian, Fulin;  Chen, Liu;  Li, Yanlian
  |  收藏  |  浏览/下载:90/0  |  提交时间:2019/01/08
Identification of compound D2923 as a novel anti-tumor agent targeting CSF1R 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 11, 页码: 1768-1776
作者:  
Liu, Ying-Qiang;  Wang, Ya-Nan;  Lu, Xiao-Yun;  Tong, Lin-Jiang;  Li, Yan
  |  收藏  |  浏览/下载:110/0  |  提交时间:2019/01/08
Targeting Epigenetic Crosstalk as a Therapeutic Strategy for EZH2-Aberrant Solid Tumors 期刊论文  OAI收割
CELL, 2018, 卷号: 175, 期号: 1, 页码: 186-+
作者:  
Huang, Xun;  Yan, Juan;  Zhang, Min;  Wang, Yafang;  Chen, Yi
  |  收藏  |  浏览/下载:77/0  |  提交时间:2019/01/08
CUDC-907 displays potent antitumor activity against human pancreatic adenocarcinoma in vitro and in vivo through inhibition of HDAC6 to downregulate c-Myc expression 期刊论文  OAI收割
Acta pharmacologica Sinica, 2018
作者:  
Fu, Xu-Hong;  Zhang, Xiong;  Yang, Hong;  Xu, Xiao-Wei;  Hu, Zong-Long
  |  收藏  |  浏览/下载:27/0  |  提交时间:2019/01/08
CTC clusters induced by heparanase enhance breast cancer metastasis 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 8, 页码: 1326-1337
作者:  
Wei, Rong-rui;  Sun, Dan-ni;  Yang, Hong;  Yan, Juan;  Zhang, Xiong
  |  收藏  |  浏览/下载:89/0  |  提交时间:2019/01/08
Design, synthesis and biological evaluation of a series of novel 2-benzamide-4-(6-oxy-N-methyl-l-naphthamide)-pyridine derivatives as potent fibroblast growth factor receptor (FGFR) inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 154, 页码: 9-28
作者:  
Wei, Manman;  Peng, Xia;  Xing, Li;  Dai, Yang;  Huang, Ruimin
  |  收藏  |  浏览/下载:63/0  |  提交时间:2019/01/08
Design, synthesis and pharmacological evaluation of ALK and Hsp90 dual inhibitors bearing resorcinol and 2,4-diaminopyrimidine motifs 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 76-86
作者:  
Geng, Kaijun;  Liu, Hongchun;  Song, Zilan;  Zhang, Chi;  Zhang, Minmin
  |  收藏  |  浏览/下载:177/0  |  提交时间:2019/01/08
Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrinnido[5,4-b]pyrrolizines as Novel Bruton's Tyrosine Kinase Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 10, 页码: 4608-4627
作者:  
Xue, Yu;  Song, Peiran;  Song, Zilan;  Wang, Aoli;  Tong, Linjiang
  |  收藏  |  浏览/下载:36/0  |  提交时间:2019/01/08
Total synthesis of (+/-)-tanshinol B, tanshinone I, and (+/-)-tanshindiol B, and C 期刊论文  OAI收割
ORGANIC & BIOMOLECULAR CHEMISTRY, 2018, 卷号: 16, 期号: 18, 页码: 3376-3381
作者:  
Wang, Fan;  Yang, Hong;  Yu, Shujuan;  Xue, Yu;  Fan, Zhoulong
  |  收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08
Identification and therapeutic intervention of coactivated anaplastic lymphoma kinase, fibroblast growth factor receptor 2, and ephrin type-A receptor 5 kinases in hepatocellular carcinoma 期刊论文  OAI收割
Hepatology (Baltimore, Md.), 2018
作者:  
Wang, Xin;  Zhang, Minmin;  Ping, Fangfang;  Liu, Hongchun;  Sun, Jingya
  |  收藏  |  浏览/下载:55/0  |  提交时间:2019/01/08