中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
  • 上海药物研究所 [15]
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发表日期
  • 2019 [15]
学科主题
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浏览/检索结果: 共15条,第1-10条 帮助

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Discovery and biological evaluation of vinylsulfonamide derivatives as highly potent, covalent TEAD autopalmitoylation inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 184, 页码: 15
作者:  
Lu, Wenchao;  Wang, Jun;  Li, Yong;  Tao, Hongru;  Xiong, Huan
  |  收藏  |  浏览/下载:83/0  |  提交时间:2020/07/01
A complex structure of arrestin-2 bound to a G protein-coupled receptor 期刊论文  OAI收割
CELL RESEARCH, 2019, 卷号: 29, 期号: 12, 页码: 971-983
作者:  
Yin, Wanchao;  Li, Zhihai;  Jin, Mingliang;  Yin, Yu-Ling;  de Waal, Parker W.
  |  收藏  |  浏览/下载:59/0  |  提交时间:2020/07/01
Synthesis of Aryl Propionamide Scaffold Containing a Pentafluorosulfanyl Moiety as SARMs 期刊论文  OAI收割
MOLECULES, 2019, 卷号: 24, 期号: 23, 页码: 13
作者:  
Shao, Pingxuan;  Zhou, Yan;  Yang, Dehua;  Wang, Ming-Wei;  Lu, Wei
  |  收藏  |  浏览/下载:25/0  |  提交时间:2020/07/01
YTHDF1 links hypoxia adaptation and non-small cell lung cancer progression 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2019, 卷号: 10, 页码: 14
作者:  
Shi, Yulin;  Fan, Songqing;  Wu, Mengge;  Zuo, Zhixiang;  Li, Xingyang
  |  收藏  |  浏览/下载:30/0  |  提交时间:2020/07/01
Integrating yeast chemical genomics and mammalian cell pathway analysis 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 9, 页码: 1245-1255
作者:  
Zhou, Fu-lai;  Li, Sheena C.;  Zhu, Yue;  Guo, Wan-jing;  Shao, Li-jun
  |  收藏  |  浏览/下载:22/0  |  提交时间:2020/07/01
Small molecule IVQ, as a prodrug of gluconeogenesis inhibitor QVO, efficiently ameliorates glucose homeostasis in type 2 diabetic mice 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 9, 页码: 1193-1204
作者:  
Zhou, Ting-ting;  Zhao, Tong;  Ma, Fei;  Zhang, Yi-nan;  Jiang, Jing
  |  收藏  |  浏览/下载:20/0  |  提交时间:2020/07/01
Discovery and Development of a Series of Pyrazolo[3,4-d]pyridazinone Compounds as the Novel Covalent Fibroblast Growth Factor Receptor Inhibitors by the Rational Drug Design 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 16, 页码: 7473-7488
作者:  
Wang, Yulan;  Dai, Yang;  Wu, Xiaowei;  Li, Fei;  Liu, Bo
  |  收藏  |  浏览/下载:40/0  |  提交时间:2020/07/01
Identification of new NIK inhibitors by discriminatory analysis-based molecular docking and biological evaluation 期刊论文  OAI收割
ARCHIV DER PHARMAZIE, 2019, 卷号: 352, 期号: 7, 页码: 9
作者:  
Cheng, Gang;  Mei, Xiao-Bing;  Yan, You-You;  Chen, Jing;  Zhang, Bo
  |  收藏  |  浏览/下载:21/0  |  提交时间:2020/07/01
Identification of a USP9X Substrate NFX1-123 by SILAC-Based Quantitative Proteomics 期刊论文  OAI收割
JOURNAL OF PROTEOME RESEARCH, 2019, 卷号: 18, 期号: 6, 页码: 2654-2665
作者:  
Chen, Xiangling;  Lu, Dayun;  Gao, Jing;  Zhu, Hongwen;  Zhou, Yanting
  |  收藏  |  浏览/下载:35/0  |  提交时间:2020/07/01
Identification of Glutaminyl Cyclase isoenzyme isoQC as a regulator of SIRP alpha-CD47 axis 期刊论文  OAI收割
CELL RESEARCH, 2019, 卷号: 29, 期号: 6, 页码: 502-505
作者:  
Wu, Zhiqiang;  Weng, Linjun;  Zhang, Tengbo;  Tian, Hongling;  Fang, Lan
  |  收藏  |  浏览/下载:29/0  |  提交时间:2020/07/01