中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [22]
采集方式
OAI收割 [22]
内容类型
期刊论文 [22]
发表日期
2021 [22]
学科主题
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浏览/检索结果:
共22条,第1-10条
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发表日期:2021
专题:上海药物研究所
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LS-106, a novel EGFR inhibitor targeting C797S, exhibits antitumor activities both in vitro and in vivo
期刊论文
OAI收割
CANCER SCIENCE, 2021, 页码: 12
作者:
Liu, Yingqiang
;
Lai, Mengzhen
;
Li, Shan
;
Wang, Yanan
;
Feng, Fang
  |  
收藏
  |  
浏览/下载:87/0
  |  
提交时间:2022/01/18
C797S
epidermal growth factor receptor
fourth-generation EGFR TKI
non-small cell lung cancer
osimertinib resistance
A camptothecin-based, albumin-binding prodrug enhances efficacy and safety in vivo
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 226, 页码: 11
作者:
Cheng, Zhiyang
;
Huang, Ying
;
Shen, Qianqian
;
Zhao, Yangrong
;
Wang, Lei
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2021/11/04
Cancer
beta-glucuronidase
Bioconjugation
Albumin
Camptothecin
STING inhibitor ameliorates LPS-induced ALI by preventing vascular endothelial cells-mediated immune cells chemotaxis and adhesion
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 12
作者:
Wu, Bing
;
Xu, Meng-meng
;
Fan, Chen
;
Feng, Chun-lan
;
Lu, Qiu-kai
  |  
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2022/01/18
acute lung injury
STING
vascular endothelial cells
inflammatory cytokines
chemokines
chemotaxis
New monoamine antidepressant, hypidone hydrochloride (YL-0919), enhances the excitability of medial prefrontal cortex in mice via a neural disinhibition mechanism
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:
Zhang, Yong-Mei
;
Ye, Lu-Yu
;
Li, Tian-Yu
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2022/01/04
YL-0919
medial prefrontal cortex
GABAergic neurons
5-HT1A receptor
GAD67-GFP transgenic mice
disinhibition
fluoxetine
electrophysiological recording
SN38-based albumin-binding prodrug for efficient targeted cancer chemotherapy
期刊论文
OAI收割
JOURNAL OF CONTROLLED RELEASE, 2021, 卷号: 339, 页码: 297-306
作者:
Huang, Ying
;
Wang, Lei
;
Cheng, Zhiyang
;
Yang, Biyu
;
Yu, Jiahui
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2021/12/01
Antitumour
Chemotherapy
SN38
Drug delivery systems
Albumin
Dezocine as a potent analgesic: overview of its pharmacological characterization
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 12
作者:
Ye, Rong-Rong
;
Jiang, Shuang
;
Xu, Xu
;
Lu, Yan
;
Wang, Yu-Jun
  |  
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2021/12/16
dezocine
opioid receptors
norepinephrine
serotonin transporter
postoperative pain
anesthesia
Identification of phosphodiesterase-4 as the therapeutic target of arctigenin in alleviating psoriatic skin inflammation
期刊论文
OAI收割
JOURNAL OF ADVANCED RESEARCH, 2021, 卷号: 33, 页码: 241-251
作者:
Li, Heng
;
Zhang, Xianglei
;
Xiang, Caigui
;
Feng, Chunlan
;
Fan, Chen
  |  
收藏
  |  
浏览/下载:112/0
  |  
提交时间:2021/11/04
PDE4
Arctigenin
Psoriasis
Inflammation
CsCCD2 Access Tunnel Design for a Broader Substrate Profile in Crocetin Production
期刊论文
OAI收割
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2021, 卷号: 69, 期号: 39, 页码: 11626-11636
作者:
Liang, Nan
;
Yao, Ming-Dong
;
Wang, Ying
;
Liu, Jia
;
Feng, Lu
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2021/12/01
crocetin
CCD2
access tunnel engineering
Saccharomyces cerevisiae
Enhancing the Potential of Miniature-Scale DNA-Compatible Radical Reactions via an Electron Donor-Acceptor Complex and a Reversible Adsorption to Solid Support Strategy
期刊论文
OAI收割
ORGANIC LETTERS, 2021, 卷号: 23, 期号: 19, 页码: 7381-7385
作者:
Lin, Bizhen
;
Lu, Weiwei
;
Chen, Zhen-yu
;
Zhang, Yue
;
Duan, Yin-zhe
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2021/12/01
Quassinoids with Inhibitory Activities against Plant Fungal Pathogens from Picrasma javanica
期刊论文
OAI收割
JOURNAL OF NATURAL PRODUCTS, 2021, 卷号: 84, 期号: 8, 页码: 2111-2120
作者:
Chen, Jian-Jun
;
Bai, Wei
;
Lu, Yu-Bo
;
Feng, Zi-Yun
;
Gao, Kun
  |  
收藏
  |  
浏览/下载:66/0
  |  
提交时间:2021/11/04