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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [14]
过程工程研究所 [6]
地球环境研究所 [5]
地理科学与资源研究所 [3]
地质与地球物理研究所 [1]
新疆理化技术研究所 [1]
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OAI收割 [36]
内容类型
期刊论文 [36]
发表日期
2023 [4]
2022 [3]
2021 [6]
2020 [5]
2019 [6]
2018 [4]
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学科主题
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浏览/检索结果:
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Drug repurposing and structure-based discovery of new PDE4 and PDE5 inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 14
作者:
Liu, Jiayuan
;
Zhang, Xianglei
;
Chen, Guofeng
;
Shao, Qiang
;
Zou, Yi
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/01/16
Phosphodiesterase-4 (PDE4)
PDE5
Inhibitor
Drug repurposing
Crystal structure
Structure -guided optimization
Discovery, structural optimization, and anti-tumor bioactivity evaluations of betulinic acid derivatives as a new type of ROR & gamma; antagonists
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 257, 页码: 15
作者:
Mei, Lianghe
;
Xu, Lansong
;
Wu, Sanan
;
Wang, Yafang
;
Xu, Chao
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2023/10/17
Betulinic acid
ROR & gamma
Target identification
Rationale structure optimization
Anti-tumor effects
antagonists
Discovery and Mechanism Study of SARS-CoV-2 3C-like Protease Inhibitors with a New Reactive Group
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 18
作者:
Ren, Pengxuan
;
Li, Hui
;
Nie, Tianqing
;
Jian, Xiaoqin
;
Yu, Changyue
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/10/17
Discovery, synthesis and mechanism study of 2,3,5-substituted [1,2,4]-thiadiazoles as covalent inhibitors targeting 3C-Like protease of SARS-CoV-2
期刊论文
OAI收割
European journal of medicinal chemistry, 2023, 卷号: 249, 页码: 115129
作者:
Ren, Pengxuan
;
Yu, Changyue
;
Zhang, Ruxue
;
Nie, Tianqing
;
Hu, Qiaoyu
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/03/26
Synthesis of maleimide-braced peptide macrocycles and their potential anti-SARS-CoV-2 mechanisms
期刊论文
OAI收割
CHEMICAL COMMUNICATIONS, 2022, 页码: 4
作者:
Li, Jian
;
Sun, Jina
;
Zhang, Xianglei
;
Zhang, Ruxue
;
Wang, Qian
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2023/04/10
Formation of robust CEI film on high voltage LiNi0.6Co0.2Mn0.2O2 cathode enabled by functional [PIVM][TFSA] ionic liquid additive
期刊论文
OAI收割
ELECTROCHIMICA ACTA, 2022, 卷号: 424, 页码: 8
作者:
Cai, Yingjun
;
Xu, Tinghua
;
Meng, Xianglei
;
von Solms, Nicolas
;
Zhang, Haitao
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/02/24
Lithium ion batteries
Electrolyte
Ionic liquid
High-voltage
Additive
Interaction-Aware Cut-In Trajectory Prediction and Risk Assessment in Mixed Traffic
期刊论文
OAI收割
IEEE/CAA Journal of Automatica Sinica, 2022, 卷号: 9, 期号: 10, 页码: 1752-1762
作者:
Xianglei Zhu
;
Wen Hu
;
Zejian Deng
;
Jinwei Zhang
;
Fengqing Hu
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2022/09/08
Cut-in behavior
interaction-aware
mixed traffic
risk assessment
trajectory prediction
Penultimate deglaciation Asian monsoon response to North Atlantic circulation collapse
期刊论文
OAI收割
NATURE GEOSCIENCE, 2021, 页码: 15
作者:
Wassenburg, Jasper A.
;
Vonhof, Hubert B.
;
Cheng, Hai
;
Martinez-Garcia, Alfredo
;
Ebner, Pia-Rebecca
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2022/08/18
Efficient transformation of CO2 to cyclic carbonates using bifunctional protic ionic liquids under mild conditions (vol 21, pg 3456, 2019)
期刊论文
OAI收割
GREEN CHEMISTRY, 2021, 卷号: 23, 期号: 22, 页码: 9179-9179
作者:
Meng, Xianglei
;
Ju, Zhaoyang
;
Zhang, Suojiang
;
Liang, Xiaodong
;
von Solms, Nicolas
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2022/06/15
Identification of phosphodiesterase-4 as the therapeutic target of arctigenin in alleviating psoriatic skin inflammation
期刊论文
OAI收割
JOURNAL OF ADVANCED RESEARCH, 2021, 卷号: 33, 页码: 241-251
作者:
Li, Heng
;
Zhang, Xianglei
;
Xiang, Caigui
;
Feng, Chunlan
;
Fan, Chen
  |  
收藏
  |  
浏览/下载:112/0
  |  
提交时间:2021/11/04
PDE4
Arctigenin
Psoriasis
Inflammation