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Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [7]
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ABPP-CoDEL: Activity-Based Proteome Profiling-Guided Discovery of Tyrosine-Targeting Covalent Inhibitors from DNA-Encoded Libraries 期刊论文  OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2023, 卷号: 145, 期号: 46, 页码: 25283-25292
作者:  
Jiang, Lulu;  Liu, Sixiu;  Jia, Xinglong;  Gong, Qinting;  Wen, Xin
  |  收藏  |  浏览/下载:30/0  |  提交时间:2024/01/16
Sequence-based drug design as a concept in computational drug design 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 21
作者:  
Chen, Lifan;  Fan, Zisheng;  Chang, Jie;  Yang, Ruirui;  Hou, Hui
  |  收藏  |  浏览/下载:18/0  |  提交时间:2023/10/17
Structure-Activity Relationship Study of 1H-Pyrrole-3-carbonitrile Derivatives as STING Receptor Agonists 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2023, 页码: 9
作者:  
Shen, Chang;  Xu, Peijia;  Zhang, Changfa;  Su, Zhaoming;  Shan, Bin
  |  收藏  |  浏览/下载:25/0  |  提交时间:2023/10/17
Triazine-Based Covalent DNA-Encoded Libraries for Discovery of Covalent Inhibitors of Target Proteins 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2022, 页码: 8
作者:  
Li, Linjie;  Su, Mingbo;  Lu, Weiwei;  Song, Hongzhi;  Liu, Jiaxiang
  |  收藏  |  浏览/下载:21/0  |  提交时间:2022/09/30
Discovery of a novel, potent and selective small-molecule inhibitor of PD-1/PD-L1 interaction with robust in vivo anti-tumour efficacy 期刊论文  OAI收割
BRITISH JOURNAL OF PHARMACOLOGY, 2021, 页码: 20
作者:  
Liu, Chenglong;  Zhou, Feilong;  Yan, Ziqin;  Shen, Lian;  Zhang, Xichen
  |  收藏  |  浏览/下载:37/0  |  提交时间:2021/06/11
Palladium-Promoted DNA-Compatible Heck Reaction 期刊论文  OAI收割
ORGANIC LETTERS, 2019, 卷号: 21, 期号: 3, 页码: 719-723
作者:  
Wang, Xuan;  Sun, Hui;  Liu, Jiaxiang;  Zhong, Wenge;  Zhang, Mingqiang
  |  收藏  |  浏览/下载:25/0  |  提交时间:2020/07/01
Ruthenium-Promoted C-H Activation Reactions between DNA-Conjugated Acrylamide and Aromatic Acids 期刊论文  OAI收割
ORGANIC LETTERS, 2018, 卷号: 20, 期号: 16, 页码: 4764-4768
作者:  
Wang, Xuan;  Sun, Hui;  Liu, Jiaxiang;  Dai, Dongcheng;  Zhang, Mingqiang
  |  收藏  |  浏览/下载:30/0  |  提交时间:2019/01/08