中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [24]
上海神经科学研究所 [5]
大连化学物理研究所 [5]
水生生物研究所 [5]
生态环境研究中心 [5]
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期刊论文 [63]
会议论文 [4]
学位论文 [3]
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2022 [1]
2021 [1]
2020 [1]
2019 [2]
2018 [7]
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Cell Biolo... [3]
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A proteomic landscape of pharmacologic perturbations for functional relevance
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL ANALYSIS, 2024, 卷号: 14, 期号: 1, 页码: 128-139
作者:
Liu, Zhiwei
;
Jiang, Shangwen
;
Hao, Bingbing
;
Xie, Shuyu
;
Liu, Yingluo
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/04/09
Proteomics
Drug
Perturbation
Drug target
Drug combination
Discovery of Thieno[2,3-e]indazole Derivatives as Novel Oral Selective Estrogen Receptor Degraders with Highly Improved Antitumor Effect and Favorable Druggability br
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 7, 页码: 5724-5750
作者:
Lu, Zhengyu
;
Cao, Yangzhi
;
Zhang, Dan
;
Meng, Xin
;
Guo, Bin
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2022/08/16
Ionizing radiation downregulates estradiol synthesis via endoplasmic reticulum stress and inhibits the proliferation of estrogen receptor-positive breast cancer cells
期刊论文
OAI收割
CELL DEATH & DISEASE, 2021, 卷号: 12, 期号: 11, 页码: 10
作者:
Yang, Pengfei
;
Feng, Xiu
;
Li, Jin
;
Zhang, Tianyi
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2021/12/13
Research Progress on Long Non-coding RNAs and Drug Resistance of Breast Cancer
期刊论文
OAI收割
CLINICAL BREAST CANCER, 2020, 卷号: 20
作者:
Zhang, Xiping
;
Yang, Hongjian
  |  
收藏
  |  
浏览/下载:60/0
  |  
提交时间:2020/10/26
Breast cancer
Drug resistance
Epithelial to mesenchymal transitions (EMT)
Long non-coding ribonucleic acids (LncRNAs)
Molecular mechanisms
A selenium- containing selective histone deacetylase 6 inhibitor for targeted in vivo breast tumor imaging and therapy
期刊论文
OAI收割
JOURNAL OF MATERIALS CHEMISTRY B, 2019, 卷号: 7, 期号: 22, 页码: 3528-3536
作者:
Tang, Chu
;
Du, Yang
;
Liang, Qian
;
Cheng, Zhen
;
Tian, Jie
  |  
收藏
  |  
浏览/下载:56/0
  |  
提交时间:2019/09/30
Preclinical characterization of SHR6390, a novel CDK 4/6 inhibitor, invitro and in human tumor xenograft models
期刊论文
OAI收割
CANCER SCIENCE, 2019, 卷号: 110, 期号: 4, 页码: 1420-1430
作者:
Long, Fei
;
He, Ye
;
Fu, Haoyu
;
Li, Yun
;
Bao, Xubin
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2020/07/01
breast cancer
CDK 4/6
drug resistance
palbociclib
SHR6390
The mTOR inhibitor AZD8055 overcomes tamoxifen resistance in breast cancer cells by down-regulating HSPB8
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 8, 页码: 1338-1346
作者:
Shi, Jia-jie
;
Chen, Si-meng
;
Guo, Chen-Liang
;
Li, Yi-xue
;
Ding, Jian
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
tamoxifen resistance
HSPB8
AZD8055
estrogen receptor
mTOR inhibitor
Development of a Novel Ferrocenyl Histone Deacetylase Inhibitor for Triple-Negative Breast Cancer Therapy
期刊论文
OAI收割
ORGANOMETALLICS, 2018, 卷号: 37, 期号: 14, 页码: 2368-2375
作者:
Tang, Chu
;
Du, Yang
;
Liang, Qian
;
Cheng, Zhen
;
Tian, Jie
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2018/10/10
Evaluating estrogenic and anti-estrogenic effect of endocrine disrupting chemicals (EDCs) by zebrafish (Danio rerio) embryo-based vitellogenin 1 (vtgl) mRNA expression
期刊论文
OAI收割
COMPARATIVE BIOCHEMISTRY AND PHYSIOLOGY C-TOXICOLOGY & PHARMACOLOGY, 2018, 卷号: 204, 页码: 45-50
作者:
Chen, Minjie
;
Liang, Yong
;
Song, Maoyong
;
Sun, Yonghua
;
Wang, Ling
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/06/20
Zebrafish embryo
Vitellogenin 1
Estrogenic effect
Endocrine disrupting chemicals
Evaluating estrogenic and anti-estrogenic effect of endocrine disrupting chemicals (EDCs) by zebrafish (Danio rerio) embryo-based vitellogenin 1 (vtgl) mRNA expression
期刊论文
OAI收割
COMPARATIVE BIOCHEMISTRY AND PHYSIOLOGY C-TOXICOLOGY & PHARMACOLOGY, 2018, 卷号: 204, 期号: 1, 页码: 45-50
作者:
Chen, Minjie
;
Zhang, Jie
;
Pang, Shaochen
;
Wang, Chang
;
Wang, Ling
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2019/07/03
Zebrafish embryo
Vitellogenin 1
Estrogenic effect
Endocrine disrupting chemicals