中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [13]
生物物理研究所 [2]
力学研究所 [1]
长春应用化学研究所 [1]
采集方式
OAI收割 [17]
内容类型
期刊论文 [17]
发表日期
2023 [2]
2022 [6]
2021 [4]
2018 [1]
2016 [1]
2012 [1]
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学科主题
Infectious... [1]
Multidisci... [1]
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共17条,第1-10条
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Structure-based development and preclinical evaluation of the SARS-CoV-2 3C-like protease inhibitor simnotrelvir
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 15
作者:
Jiang, Xiangrui
;
Su, Haixia
;
Shang, Weijuan
;
Zhou, Feng
;
Zhang, Yan
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2024/03/25
A viral RNA-dependent RNA polymerase inhibitor VV116 broadly inhibits human coronaviruses and has synergistic potency with 3CLpro inhibitor nirmatrelvir
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 10
作者:
Zhang, Yumin
;
Sun, Yuan
;
Xie, Yuanchao
;
Shang, Weijuan
;
Wang, Zhen
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/12/08
In vitro and in vivo evaluation of the main protease inhibitor FB2001 against SARS-CoV-2
期刊论文
OAI收割
ANTIVIRAL RESEARCH, 2022, 卷号: 208, 页码: 10
作者:
Shang, Weijuan
;
Dai, Wenhao
;
Yao, Cheng
;
Xu, Ling
;
Tao, Xiangming
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2023/04/10
SARS-CoV-2
SARS-CoV-2 variants
FB2001
Main protease
PBPK
Anti-SARS-CoV-2 in vivo
Disturbed Flow-Facilitated Margination and Targeting of Nanodisks Protect against Atherosclerosis
期刊论文
OAI收割
SMALL, 2022, 页码: 15
作者:
Zhao, ChuanRong
;
Li, Jingyi
;
Jiang, ZhiTong
;
Zhu, JuanJuan
;
Zhao, JiaNan
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2022/12/20
atherosclerosis
decitabine
endothelial inflammation
hemodynamics
nanoparticles
Disturbed Flow-Facilitated Margination and Targeting of Nanodisks Protect against Atherosclerosis
期刊论文
OAI收割
SMALL, 2022, 页码: 15
作者:
Zhao, Chuan-Rong
;
Li, Jingyi
;
Jiang, Zhi-Tong
;
Zhu, Juan-Juan
;
Zhao, Jia-Nan
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2023/04/10
atherosclerosis
decitabine
endothelial inflammation
hemodynamics
nanoparticles
Discovery of Novel N-(5-(Pyridin-3-yl)-1H-indazol-3-yl)benzamide Derivatives as Potent Cyclin-Dependent Kinase 7 Inhibitors for the Treatment of Autosomal Dominant Polycystic Kidney Disease
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 19
作者:
Yang, Bowen
;
Zhang, Haoran
;
Li, Na
;
Gao, Lixin
;
Jiang, Hong
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2023/04/10
Oral remdesivir derivative VV116 is a potent inhibitor of respiratory syncytial virus with efficacy in mouse model
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2022, 卷号: 7, 期号: 1, 页码: 3
作者:
Zhang, Ruxue
;
Zhang, Yumin
;
Zheng, Wei
;
Shang, Weijuan
;
Wu, Yan
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2022/06/15
Structure-Activity Relationship Study of Indolin-5-yl-cyclopropanamine Derivatives as Selective Lysine Specific Demethylase 1 (LSD1) Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 5, 页码: 4335-4349
作者:
Li, Chunpu
;
Su, Mingbo
;
Zhu, Wei
;
Kan, Weijuan
;
Ge, Tianpeng
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2022/06/15
Rational Design and Development of Novel CDK9 Inhibitors for the Treatment of Acute Myeloid Leukemia
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14647-14663
作者:
Han, Xu
;
Song, Ning
;
Saidahmatov, Abdusaid
;
Wang, Peipei
;
Wang, Yong
  |  
收藏
  |  
浏览/下载:78/0
  |  
提交时间:2021/12/16
Design and development of an oral remdesivir derivative VV116 against SARS-CoV-2
期刊论文
OAI收割
CELL RESEARCH, 2021, 页码: 3
作者:
Xie, Yuanchao
;
Yin, Wanchao
;
Zhang, Yumin
;
Shang, Weijuan
;
Wang, Zhen
  |  
收藏
  |  
浏览/下载:82/0
  |  
提交时间:2021/11/04