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Chinese Academy of Sciences Institutional Repositories Grid
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Pharmacokinetics, mass balance, and metabolism of [
14
C]FCN-437c, a selective and potent CDK4/6 inhibitor in humans
期刊论文
OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2025, 卷号: 95, 期号: 1, 页码: 12
作者:
Gao, Lei
;
Ma, Sheng
;
Yan, Shu
;
Zhang, Hua
;
Tian, Ling
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2025/07/25
FCN-437c
CDK4/6 inhibitor
Mass balance
Radiopharmacokinetics
Drug metabolism
UBE4B modulates BET inhibitor sensitivity via KLHL22-JAK2-PIM1 axis in hepatocellular carcinoma
期刊论文
OAI收割
BIOCHEMICAL PHARMACOLOGY, 2025, 卷号: 237, 页码: 19
作者:
Wang, Li
;
Huan, Xia-Juan
;
Song, Shan-Shan
;
Bao, Xu-Bin
;
Tian, Chang-Qing
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2025/06/23
UBE4B
BET inhibitors
Resistance
KLHL22
JAK2
Cbl-b inhibitor NX-1607 activates MAPK/ERK signaling pathway and enhances T-cell activation
期刊论文
OAI收割
JOURNAL FOR IMMUNOTHERAPY OF CANCER, 2025, 卷号: 13, 期号: 5, 页码: 18
作者:
Zhu, Wenting
;
Lu, Shan
;
Jia, Li
;
Liu, Benjin
;
Song, Shanshan
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/08/20
Tumor microenvironment - TME
T cell
Immunotherapy
Immune modulatory
Immune Checkpoint Inhibitor
Discovery and Extensive Follow-up of SN 2024ggi, a Nearby Type IIP Supernova in NGC 3621
期刊论文
OAI收割
ASTROPHYSICAL JOURNAL, 2025, 卷号: 983, 期号: 1
作者:
Chen, Ting-Wan
;
Yang, Sheng
;
Srivastav, Shubham
;
Moriya, Takashi J.
;
Smartt, Stephen J.
  |  
收藏
  |  
浏览/下载:89/0
  |  
提交时间:2025/04/21
Assessing and predicting Bojiang lake area and LULC changes from 2000 to 2045
期刊论文
OAI收割
JOURNAL OF HYDROLOGY-REGIONAL STUDIES, 2025, 卷号: 58, 页码: 102216
作者:
Naeem, Muhammad
;
Zhang, Yongqiang
;
Tian, Xiaoqiang
;
Miao, Ping
;
Li, Congcong
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2025/03/18
Machine Learning
CA-ANN Model
Lake changes
Land Use and Land Cover (LULC) Changes
Climate Change
Water management
Mantle metasomatism by subducted Indian continental crust: Evidence from post-collisional basaltic ultrapotassic rocks in southern Tibetan plateau
期刊论文
OAI收割
LITHOS, 2025, 卷号: 498, 页码: 11
作者:
Zhang, Miao-Yan
;
Hao, Lu-Lu
;
Qi, Yue
;
Wang, Qiang
;
Kerr, Andrew C.
  |  
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2025/04/03
Mo - B isotopes
Post-collisional ultrapotassic rocks
Continental crust recycling
Crust-mantle interaction
Tibetan Plateau
New Phenolic Compounds from
Eucalyptus tereticornis
with Antioxidant Activity
期刊论文
OAI收割
CHEMISTRY & BIODIVERSITY, 2025, 页码: 8
作者:
Zhang, Yu
;
Miao, Lei
;
Li, Guo-Li
;
Zhang, Chuan-Rui
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2025/05/27
antioxidant activity
configuration determination
Eucalyptus tereticornis
glycosides
sesquilignans
Unveiling the Emission Properties of Three Long-period Pulsars Using FAST
期刊论文
OAI收割
ASTROPHYSICAL JOURNAL SUPPLEMENT SERIES, 2025, 卷号: 277, 期号: 2, 页码: 39
作者:
Tedila, H. M.
;
Li, D.
;
Wang, P.
;
Yuen, R.
;
Yuan, J. P.
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2025/05/21
Structure-Based Discovery of a Series of Novel MAT2a Inhibitors
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2025, 页码: 5
作者:
Zhou, Yushan
;
Wang, Li
;
Ren, Ruyue
;
Zhang, Junjie
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2025/05/27
MAT2a
MTAP
Synthetic lethality
Allosteric inhibitor
Structure-activity relationship
USP7 V517F mutation as a mechanism of inhibitor resistance
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2025, 卷号: 16, 期号: 1, 页码: 14
作者:
Miao, Yu-Ling
;
Fan, Fengying
;
Cheng, Yong-Jun
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2025/05/27