中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海有机化学研究... [195]
上海药物研究所 [37]
深圳先进技术研究院 [18]
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期刊论文 [322]
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氟化学 [109]
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Discovery of 2(1
H
)-Quinoxalinone Derivatives as Potent and Selective MAT2A Inhibitors for the Treatment of MTAP-Deficient Cancers
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 2, 页码: 1222-1244
作者:
Li, Chunzheng
;
Lan, Xiaojing
;
Li, Xinge
;
Fu, Yixian
;
Gui, Gang
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2025/04/01
Multi-omics landscape and molecular basis of radiation tolerance in a tardigrade
期刊论文
OAI收割
SCIENCE, 2024, 卷号: 386, 期号: 6720, 页码: 13
作者:
Li, Lei
;
Ge, Zhengping
;
Liu, Shihao
;
Zheng, Kun
;
Li, Yaqi
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/12/09
Cross-Model Comparative Loss for Enhancing Neuronal Utility in Language Understanding
期刊论文
OAI收割
ACM TRANSACTIONS ON INFORMATION SYSTEMS, 2024, 卷号: 42, 期号: 5, 页码: 29
作者:
Zhu, Yunchang
;
Pang, Liang
;
Wu, Kangxi
;
Lan, Yanyan
;
Shen, Huawei
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/12/06
Natural language understanding
question answering
pseudo-relevance feedback
loss function
Amlodipine inhibits Synaptotagmin-4's oncogenic activity on gastric cancer proliferation by targeting calcium signaling
期刊论文
OAI收割
FUNCTIONAL & INTEGRATIVE GENOMICS, 2024, 卷号: 24, 期号: 3, 页码: 14
作者:
Huang, Wen
;
Yang, Shuo
;
Deng, Minying
;
Luo, Rongkui
;
Liang, Huaiyu
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/05/22
Gastric cancer
synaptotagmin-4
Calcium ion channel
Mitogen-activated protein kinase signaling pathway
Amlodipine
Discovery, Optimization, and Evaluation of Novel Pyridin-2(1
H
)-one Analogues as Potent TRK Inhibitors for Cancer Treatment
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1168-1183
作者:
Xu, Zichao
;
Peng, Xia
;
Zhang, Renjie
;
Ji, Yinchun
;
You, Mengke
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2024/02/27
Creating a zero amylose barley with high soluble sugar content by genome editing
期刊论文
OAI收割
PLANT MOLECULAR BIOLOGY, 2024, 卷号: 114, 期号: 3
作者:
Li, Yun
;
Jiang, Yanyan
;
Cao, Dong
;
Dang, Bin
;
Yang, Xijuan
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/11/27
Preclinical and early clinical studies of a novel compound SYHA1813 that efficiently crosses the blood-brain barrier and exhibits potent activity against glioblastoma
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 12, 页码: 4748-4764
作者:
Liu, Yingqiang
;
Zhan, Zhengsheng
;
Kang, Zhuang
;
Li, Mengyuan
;
Lv, Yongcong
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2024/01/26
Small molecule inhibitor
Tumor microenvironment
Immune-checkpoint
immune-deficient mouse models
including temozolomide (TMZ) insensitive tumors. Notably
Shifting of the first-order root foraging strategies of Chinese fir (Cunninghamia lanceolata) under varied environmental conditions
期刊论文
OAI收割
TREES-STRUCTURE AND FUNCTION, 2023, 卷号: N/A
作者:
Liao, Yingchun
;
Fan, Houbao
;
Wei, Xiaohua
;
Wang, Huimin
;
Shen, Fangfan
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/01/04
First-order root traits
Root foraging strategies
Environmental gradients
Climatic variables
Soil nutrients
Chinese fir plantations
SYK-mediated epithelial cell state is associated with response to c-Met inhibitors in c-Met-overexpressing lung cancer
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 13
作者:
Zhou, Ji
;
Zhang, Xu-Chao
;
Xue, Shan
;
Dai, Mengdi
;
Wang, Yueliang
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2023/10/17
Intact regulation of G1/S transition renders esophageal squamous cell carcinoma sensitive to PI3Kα inhibitors
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 153
作者:
Zhang, Xu
;
Wang, Yuxiang
;
Zhang, Xi
;
Shen, Yanyan
;
Yang, Kang
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/03/27