中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [61]
南京土壤研究所 [27]
工程热物理研究所 [14]
长春光学精密机械与物... [4]
寒区旱区环境与工程研... [3]
生态环境研究中心 [3]
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OAI收割 [133]
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期刊论文 [118]
会议论文 [12]
专利 [2]
译著 [1]
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2024 [5]
2023 [8]
2022 [2]
2021 [3]
2020 [9]
2019 [3]
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Covalent DNA-Encoded Library Workflow Drives Discovery of SARS-CoV-2 Nonstructural Protein Inhibitors
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2024, 页码: 14
作者:
Wang, Xudong
;
Xiong, Liwei
;
Zhu, Ying
;
Liu, Sixiu
;
Zhao, Wenfeng
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/12/25
Discovery of Novel Nonpeptidic and Noncovalent Small Molecule 3CL
pro
Inhibitors as anti-SARS-CoV-2 Drug Candidate
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 15, 页码: 12760-12783
作者:
Jiang, Zhidong
;
Feng, Bo
;
Chen, Lu
;
Nie, Tianqing
;
Chen, Shizhao
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2024/09/26
PPIA dictates NRF2 stability to promote lung cancer progression
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2024, 卷号: 15, 期号: 1, 页码: 20
作者:
Lu, Weiqiang
;
Cui, Jiayan
;
Wang, Wanyan
;
Hu, Qian
;
Xue, Yun
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2024/07/12
Chemical Space Profiling of SARS-CoV-2 PL
pro
Using DNA-Encoded Focused Libraries
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2024, 页码: 10
作者:
Wang, Xudong
;
Zhu, Ying
;
Zhao, Qingyi
;
Lu, Weiwei
;
Xu, Yechun
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/05/07
DNA-Encoded Focused Libraries (DEFLs)
SARS-CoV-2
Papain-like Protease
Library Design
ProteinInhibitors
Oral Simnotrelvir for Adult Patients with Mild-to-Moderate Covid-19
期刊论文
OAI收割
NEW ENGLAND JOURNAL OF MEDICINE, 2024, 卷号: 390, 期号: 3, 页码: 230-241
作者:
Cao, Bin
;
Wang, Yeming
;
Lu, Hongzhou
;
Huang, Chaolin
;
Yang, Yumei
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2024/05/07
Efficacy and safety of SIM0417 (SSD8432) plus ritonavir for COVID-19 treatment: a randomised, double-blind, placebo- controlled, phase 1b trial
期刊论文
OAI收割
LANCET REGIONAL HEALTH-WESTERN PACIFIC, 2023, 卷号: 38, 页码: 13
作者:
Wang, Fuxiang
;
Xiao, Wen
;
Tang, Yimin
;
Cao, Mengli
;
Shu, Dan
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2023/10/17
Covid-19
3CL protease inhibitor
SARS-CoV-2 viral load
Alleviation of COVID-19 symptoms
Multi-omics for COVID-19: driving development of therapeutics and vaccines
期刊论文
OAI收割
NATIONAL SCIENCE REVIEW, 2023, 卷号: 10, 期号: 9, 页码: 30
作者:
Guo, Mengyu
;
Xiong, Muya
;
Peng, Jinying
;
Guan, Tong
;
Su, Haixia
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/12/19
COVID-19
SARS-CoV-2
multi-omics
antibodies
small-molecule drugs
vaccines
Novel thieno[2,3-b]quinoline-procaine hybrid molecules: A new class of allosteric SHP-1 activators evolved from PTP1B inhibitors
期刊论文
OAI收割
CHINESE CHEMICAL LETTERS, 2023, 卷号: 34, 期号: 8, 页码: 6
作者:
Xu, Lei
;
Xuyan, Xuyang
;
Minmi, Minmin
;
Wang, Zhiji
;
Shee, Chao
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2023/10/17
Activator
PTPs
Inhibitor
Thieno[2
b ]quinoline derivatives
Diffuse large B-cell lymphoma
Structural insights into dimerization and activation of the mGlu2-mGlu3 and mGlu2-mGlu4 heterodimers
期刊论文
OAI收割
CELL RESEARCH, 2023, 页码: 13
作者:
Wang, Xinwei
;
Wang, Mu
;
Xu, Tuo
;
Feng, Ye
;
Shao, Qiang
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2023/10/17
Structure-Based Design of Potent Peptidomimetic Inhibitors Covalently Targeting SARS-CoV-2 Papain-like Protease
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2023, 卷号: 24, 期号: 10, 页码: 15
作者:
Wang, Qian
;
Chen, Guofeng
;
He, Jian
;
Li, Jiameng
;
Xiong, Muya
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2023/10/17
SARS-CoV-2
papain-like protease
covalent inhibitor
co-crystal structure
in vitro assay