中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [22]
上海光学精密机械研究... [4]
生物物理研究所 [3]
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OAI收割 [50]
内容类型
期刊论文 [50]
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2025 [3]
2024 [4]
2023 [4]
2022 [4]
2021 [8]
2020 [1]
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Biochemica... [1]
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Design, synthesis, and evaluation of Menin-targeting compounds for the treatment of acute Myelocytic leukemia (AML)
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 296, 页码: 17
作者:
Mo, Jun
;
Wang, Yuxian
;
Pan, Youlu
;
Xiao, Qitao
;
Zhao, Jinyi
  |  
收藏
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浏览/下载:5/0
  |  
提交时间:2025/08/20
Menin
High binding affinity
Anti-proliferation activity
AML
Substrate recognition and cleavage mechanism of the monkeypox virus core protease
期刊论文
OAI收割
NATURE, 2025, 页码: 29
作者:
Gao, Yan
;
Xie, Xiong
;
Zhang, Xiaoyu
;
Cao, Junyuan
;
Lan, Weiqi
  |  
收藏
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浏览/下载:6/0
  |  
提交时间:2025/08/20
Exploratory research on the effective chemical basis of tanreqing injection for treating acute lung injury: In vivo, in vitro and in silico
期刊论文
OAI收割
JOURNAL OF ETHNOPHARMACOLOGY, 2025, 卷号: 337, 页码: 11
作者:
Tang, Bixi
;
Xie, Like
;
Wang, Yangyang
;
Shi, Yulong
;
Kan, Weijuan
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2024/11/26
Lung first-pass effect
Tanreqing injection
Pharmacokinetics
Sepsis-associated acute lung injury
Acute respiratory distress syndrome
Design and development of a series of 4-(piperazin-1-yl)pyrimidines as irreversible menin inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 280, 页码: 20
作者:
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2024/11/26
Menin
Covalent inhibitor
Antitumor
Degradation
Discovery of Novel 2-Aminopyridine-Based and 2-Aminopyrimidine-Based Derivatives as Potent CDK/HDAC Dual Inhibitors for the Treatment of Refractory Solid Tumors and Hematological Malignancies
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 17, 页码: 15220-15245
作者:
Saidahmatov, Abdusaid
;
Li, Jianan
;
Xu, Shihao
;
Hu, Xiaobei
;
Gao, Xiangqian
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2024/10/21
Discovery of a Highly Potent, Selective and Efficacious USP7 Degrader for the Treatment of Acute Lymphoblastic Leukemia
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 20
作者:
Xu, Miaomiao
;
Fu, Jingfeng
;
Pei, Yuan
;
Li, Mengna
;
Kan, Weijuan
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2024/08/22
Research progress of biochar modification technology and its application in environmental remediation
期刊论文
OAI收割
BIOMASS & BIOENERGY, 2024, 卷号: 184, 页码: 13
作者:
Lan, Weijuan
;
Zhao, Xinxin
;
Wang, Yingxian
;
Jin, Xin
;
Ji, Jiangtao
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2025/11/17
Biomass
Biochar
Preparation methods
Modification technology
Environmental remediation
A viral RNA-dependent RNA polymerase inhibitor VV116 broadly inhibits human coronaviruses and has synergistic potency with 3CLpro inhibitor nirmatrelvir
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 10
作者:
Zhang, Yumin
;
Sun, Yuan
;
Xie, Yuanchao
;
Shang, Weijuan
;
Wang, Zhen
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2023/12/08
DNA methyltransferase 1 deficiency improves macrophage motility and wound healing by ameliorating cholesterol accumulation
期刊论文
OAI收割
NPJ REGENERATIVE MEDICINE, 2023, 卷号: 8, 期号: 1, 页码: 29
作者:
Zhao, Chuanrong
;
Yang, Qianru
;
Tang, Runze
;
Li, Wang
;
Wang, Jin
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2023/07/17
Targeting C/EBP alpha overcomes primary resistance and improves the efficacy of FLT3 inhibitors in acute myeloid leukaemia
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 18
作者:
Wang, Hanlin
;
Luo, Guanghao
;
Hu, Xiaobei
;
Xu, Gaoya
;
Wang, Tao
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2023/10/17