中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海硅酸盐研究所 [7]
上海药物研究所 [6]
海洋研究所 [5]
力学研究所 [1]
青岛生物能源与过程研... [1]
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OAI收割 [20]
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期刊论文 [19]
专利 [1]
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2025 [1]
2022 [1]
2021 [1]
2019 [3]
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2017 [1]
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Chemistry,... [1]
Engineerin... [1]
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Discovery of Novel RNA Demethylase FTO Inhibitors Featuring an Acylhydrazone Scaffold with Potent Antileukemia Activity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 22
作者:
Liang, Xuewu
;
Huang, Yue
;
Ren, Hairu
;
Liu, Qi
;
Chen, Liang
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2025/04/01
Design, synthesis, and biological evaluation of novel carbazole derivatives as potent DNMT1 inhibitors with reasonable PK properties
期刊论文
OAI收割
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2022, 卷号: 37, 期号: 1, 页码: 1537-1555
作者:
Li, Ennian
;
Wang, Kai
;
Zhang, Bei
;
Guo, Siqi
;
Xiao, Senhao
  |  
收藏
  |  
浏览/下载:61/0
  |  
提交时间:2022/08/16
DNMT1 inhibitor
A549 cell lines
HCT116 cell lines
antitumor activity
pharmacokinetic
Structure-Guided Development of Small-Molecule PRC2 Inhibitors Targeting EZH2-EED Interaction
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 12, 页码: 8194-8207
作者:
Du, Daohai
;
Xu, Dandan
;
Zhu, Licheng
;
Stazi, Giulia
;
Zwergel, Clemens
  |  
收藏
  |  
浏览/下载:97/0
  |  
提交时间:2021/08/17
Highly Selective Protein Tyrosine Phosphatase Inhibitor, 2,2 ',3,3 '-Tetrabromo-4,4 ',5,5 '-tetrahydroxydiphenylmethane, Ameliorates Type 2 Diabetes Mellitus in BKS db Mice
期刊论文
OAI收割
MOLECULAR PHARMACEUTICS, 2019, 卷号: 16, 期号: 5, 页码: 1839-1850
作者:
Li, Chao
;
Luo, Jiao
;
Guo, Shuju
;
Jia, Xiaoling
;
Guo, Chuanlong
  |  
收藏
  |  
浏览/下载:87/0
  |  
提交时间:2019/08/28
type 2 diabetes mellitus
protein tyrosine phosphatase 1B
insulin resistance
hypoglycemic activity
dyslipidemia
Discovery of Novel Bromophenol Thiosemicarbazone Hybrids as Potent Selective Inhibitors of Poly(ADP-ribose) Polymerase-1 (PARP-1) for Use in Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 6, 页码: 3051-3067
作者:
Guo, Chuanlong
;
Wang, Lijun
;
Li, Xinxue
;
Wang, Shuaiyu
;
Yu, Xuemin
  |  
收藏
  |  
浏览/下载:86/0
  |  
提交时间:2019/08/28
Toward a treatment of diabesity: In vitro and in vivo evaluation of uncharged bromophenol derivatives as a new series of PTP1B inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 166, 页码: 178-185
作者:
Li, Xiangqian
;
Xu, Qi
;
Li, Chao
;
Luo, Jiao
;
Li, Xiuxue
  |  
收藏
  |  
浏览/下载:66/0
  |  
提交时间:2019/05/15
Anti-diabetic
PTP1B inhibitor
Selectivity
BKS db mice
Toxicity
A photo-excited electron transfer hyperchannel constructed in Pt-dispersed pyrimidine-modified carbon nitride for remarkably enhanced water-splitting photocatalytic activity
期刊论文
OAI收割
APPLIED CATALYSIS B-ENVIRONMENTAL, 2018, 卷号: 237, 页码: 888, 894
作者:
Jin, Xixiong
;
Zhang, Lingxia
;
Fan, Xiangqian
;
Tian, Jianjian
;
Wang, Min
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收藏
  |  
浏览/下载:35/0
  |  
提交时间:2018/12/28
Electron transfer
Carbon nitride
Copolymer
Photocatalytic water-splitting
Hydrogen evolution
Core-shell LaPO4/g-C3N4 nanowires for highly active and selective CO2 reduction
期刊论文
OAI收割
APPLIED CATALYSIS B-ENVIRONMENTAL, 2017, 卷号: 201, 页码: 629-635
作者:
Li, Mengli
;
Zhang, Lingxia
;
Fan, Xiangqian
;
Wu, Meiying
;
Wang, Min
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2017/02/24
CO2 photoreduction
Core-shell nanowire
Heterostructure
LaPO4
Graphite carbon nitride
Dual synergetic effects in MoS2/pyridine-modified g-C3N4 composite for highly active and stable photocatalytic hydrogen evolution under visible light
期刊论文
OAI收割
APPLIED CATALYSIS B-ENVIRONMENTAL, 2016, 卷号: 190, 页码: 36-43
作者:
Li, Mengli
;
Zhang, Lingxia
;
Fan, Xiangqian
;
Wu, Meiying
;
Du, Yanyan
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2017/02/27
Hydrogen production
Dual synergetic effects
Photocatalysis
MoS2
Graphite carbon nitride
N-doped graphitic carbon-incorporated g-C3N4 for remarkably enhanced photocatalytic H-2 evolution under visible light
期刊论文
OAI收割
CARBON, 2016, 卷号: 99, 页码: 111-117
作者:
Zhou, Yajun
;
Zhang, Lingxia
;
Huang, Weimin
;
Kong, Qinglu
;
Fan, Xiangqian
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2017/03/01