中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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大连化学物理研究所 [80]
上海药物研究所 [53]
上海营养与健康研究... [13]
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期刊论文 [164]
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Discovery of pyrrolo[2,3-d]pyrimidine derivatives as novel FLT3/ IRAK4 inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 296, 页码: 23
作者:
Yuan, Haibin
;
Gao, Yue
;
Wang, Peipei
;
Dong, Xiaowu
;
Li, Jia
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/08/20
AML
FLT3/IRAK4 inhibitor
Pyrrolo [2,3-d] pyrimidine
Acquired resistance
Adaptive resistance
Targeted characterisation of bioactive prenylated flavonoids from
Ficus
carica
L. fruits
期刊论文
OAI收割
FOOD CHEMISTRY, 2025, 卷号: 483, 页码: 11
作者:
Yuan, Yue
;
Li, Zuopeng
;
Aisa, Haji Akber
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2025/06/23
Figs
Targeted isolation
Prenylated flavonoids
Antioxidant
Anti-inflammatory
Antitubercular
Concise synthesis of NDP-activated uronic acid by an oxidation reaction insertion strategy
期刊论文
OAI收割
CHINESE CHEMICAL LETTERS, 2025, 卷号: 36, 期号: 8, 页码: 7
作者:
Yang, Nana
;
Yuan, Rui
;
Fu, Xinyue
;
Tian, Xiao
;
Yu, Jin
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/08/20
NDP-uronic acids
Biocatalysis
Enzyme-mediated biomimetic synthesis
Oxidation reaction insertion strategy
Integrative Proteomics and Histone PTMomics Study on Anti-TNBC Effect of JIB-04
期刊论文
OAI收割
JOURNAL OF THE AMERICAN SOCIETY FOR MASS SPECTROMETRY, 2025, 页码: 12
作者:
Tao, Shengna
;
Guo, Jingli
;
Zhang, Jingdan
;
Zhang, Mingya
;
Wang, Zhe
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2025/08/20
Proteomics
histone PTMomics
epigenetic inhibitor
JIB-04
TNBC
Covalent sortase A inhibitor, α, β-unsaturated aldehydes, prevents Staphylococcus aureus infection
期刊论文
OAI收割
MICROBIAL PATHOGENESIS, 2025, 卷号: 204, 页码: 12
作者:
Wang, Jianchao
;
He, Yuan
;
Chu, Chenliang
;
Wu, Ziqi
;
Zhang, Ting
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2025/06/23
Sortase A
Covalent inhibitor
alpha
beta-unsaturated aldehydes
Anti-virulence therapy
Staphylococcus aureus
Ginsenoside (20)S-APPT induces ferroptosis in hepatocellular carcinoma and cholangiocarcinoma by targeting FSP1
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 18
作者:
Liu, Fan-yu
;
Yang, Yuan-jie
;
Wang, Xue-long
;
Hong, Yan
;
Ou-Yang, Xiao-peng
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/08/20
A long-term paddy rice distribution dataset in Asia at a 30 m spatial resolution
期刊论文
OAI收割
SCIENTIFIC DATA, 2025, 卷号: 12, 期号: 1, 页码: 1052
作者:
Li, Shaoping
;
Shen, Ruoque
;
Jiang, Jiale
;
Peng, Qiongyan
;
Chen, Xuebing
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2025/07/18
Discovery of novel GluN1/GluN3A NMDA receptor inhibitors using a deep learning-based method
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 8
作者:
Wang, Shi-hang
;
Zeng, Yue
;
Yang, Hao
;
Tian, Si-yuan
;
Zhou, Yong-qi
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2025/07/25
N
-methyl-
D
-aspartate receptors
GluN1/GluN3A
ligand-based virtual screening
scaffold hopping
deep learning
GeminiMol
Molecular mechanism of the arrestin-biased agonism of neurotensin receptor 1 by an intracellular allosteric modulator
期刊论文
OAI收割
CELL RESEARCH, 2025, 卷号: 35, 期号: 4, 页码: 284-295
作者:
Sun, Demeng
;
Li, Xiang
;
Yuan, Qingning
;
Wang, Yuanxia
;
Shi, Pan
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2025/05/27
A holistic strategy for the in-depth discrimination and authentication of 16 citrus herbs and associated commercial products based on machine learning techniques and non-targeted metabolomics
期刊论文
OAI收割
JOURNAL OF CHROMATOGRAPHY A, 2025, 卷号: 1745, 页码: 12
作者:
Huang, Yu-shi
;
An, Ya-ling
;
Zheng, Yue-yuan
;
Zhao, Wen-jie
;
Song, Chun-qian
  |  
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2025/04/01
Citrus herbs
Discrimination
LC-MS
Machine learning
Differential markers