中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [13]
自动化研究所 [10]
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OAI收割 [54]
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期刊论文 [44]
会议论文 [8]
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学位论文 [1]
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2025 [3]
2024 [10]
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Targeting the histone reader ZMYND8 inhibits antiandrogen-induced neuroendocrine tumor transdifferentiation of prostate cancer
期刊论文
OAI收割
NATURE CANCER, 2025, 页码: 37
作者:
Wang, Hanling
;
Zhang, Sulin
;
Pan, Qiang
;
Guo, Jiacheng
;
Li, Ni
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/05/27
Discovery of novel covalent stabilizers for p53 Y220C using structure-based drug discovery methods
期刊论文
OAI收割
MOLECULAR DIVERSITY, 2025, 页码: 14
作者:
Wen, Yiming
;
Xu, Peijia
;
Chen, Yijie
;
Meng, Jingyi
;
Zheng, Mingyue
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2025/04/01
p53 Y220C
Covalent stabilizer
Virtual screening
Molecular dynamics
DNA binding
Structure-activity relationship
Cancer therapy
Design, synthesis, and structure-activity relationship studies of triazolo-pyrimidine derivatives as WRN inhibitors for the treatment of MSI tumors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 282, 页码: 21
作者:
Sui, Qibang
;
Zhou, Yuanyang
;
Li, Manjia
;
Wang, Dan
;
Cui, Rongrong
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/12/25
Synthetic lethal
MSI tumors
WRN inhibitors
Triazolo-pyrimidine derivatives
Ginkgetin Alleviates Inflammation and Senescence by Targeting STING
期刊论文
OAI收割
ADVANCED SCIENCE, 2024, 页码: 15
作者:
Liu, Yadan
;
Ye, Jialin
;
Fan, Zisheng
;
Wu, Xiaolong
;
Zhang, Yinghui
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/12/16
cGAS-STING signaling
Ginkgetin
senescence
STING inhibitor
target identification
Ecological restoration enhances dryland carbon stock by reducing surface soil carbon loss due to wind erosion
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2024, 卷号: 121, 期号: 46, 页码: 10
作者:
Song, Jian
;
Wan, Shiqiang
;
Zhang, Kesheng
;
Hong, Songbai
;
Xia, Jianyang
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2025/02/06
carbon neutrality
climate solutions
plant productivity
soil carbon
soil erosion
Research on the viscoelastic scCO 2 foam systems synergistically stabilized by nonionic/zwitterionic mixed surfactants
期刊论文
OAI收割
COLLOIDS AND SURFACES A-PHYSICOCHEMICAL AND ENGINEERING ASPECTS, 2024, 卷号: 697, 页码: 14
作者:
Zheng, Nanxin
;
Zhu, Jingyi
;
Yang, Zhaozhong
;
Li, Xiaogang
;
Li, Qi
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/06/27
ScCO2 foam fluid
Synergistic effect
Wormlike micelles
Foam stabilization mechanism
Microstructure
Stillbirths Associated with Particle Pollution are Disproportionally Contributed by Sand Dust: Findings from 52 Low- and Middle-Income Countries
期刊论文
OAI收割
ENVIRONMENTAL SCIENCE & TECHNOLOGY, 2024, 卷号: 58, 期号: 36, 页码: 15971-15983
作者:
Li, Pengfei
;
Wu, Jingyi
;
Tong, Mingkun
;
Wang, Ruohan
;
Tang, Mingjin
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2024/10/10
particulate matter
sand dust
stillbirth
joint exposure-response function
maternal health
health inequality
Targeting STING oligomerization with licochalcone D ameliorates STING-driven inflammatory diseases
期刊论文
OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2024, 页码: 14
作者:
Zhang, Yinghui
;
Liu, Yadan
;
Jiang, Bing
;
Chen, Lifan
;
Hu, Jie
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2024/10/21
cGAS-STING signaling
STING inhibitor
TransformerCPI model
Licochalcone D
inflammatory diseases
Deep representation learning of chemical-induced transcriptional profile for phenotype-based drug discovery
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2024, 卷号: 15, 期号: 1, 页码: 14
作者:
Tong, Xiaochu
;
Qu, Ning
;
Kong, Xiangtai
;
Ni, Shengkun
;
Zhou, Jingyi
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2024/08/22
KinomeMETA: a web platform for kinome-wide polypharmacology profiling with meta-learning
期刊论文
OAI收割
NUCLEIC ACIDS RESEARCH, 2024, 页码: 9
作者:
Li, Zhaojun
;
Qu, Ning
;
Zhou, Jingyi
;
Sun, Jingjing
;
Ren, Qun
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2024/06/27