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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [20]
上海应用物理研究所 [1]
上海硅酸盐研究所 [1]
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OAI收割 [22]
内容类型
期刊论文 [22]
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2025 [1]
2024 [2]
2023 [2]
2022 [1]
2021 [3]
2020 [1]
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Design of Selective BRD4 Inhibitors for the Treatment of Autosomal Dominant Polycystic Kidney Disease
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 18
作者:
Yang, Yueyue
;
Liu, Hongli
;
Yuan, Haoxing
;
Lyu, Kaikai
;
Zhong, Haiyang
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2025/04/01
Structure-Based Rational Design and Evaluation of BET-Aurora Kinase Dual-Inhibitors for Treatment of Cancers
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 21
作者:
Lyu, Kaikai
;
Ren, Ying
;
Mou, Jie
;
Yang, Yunfang
;
Pan, Yaoyao
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2025/02/28
Discovery of a brain-permeable bromodomain and extra terminal domain (BET) inhibitor with selectivity for BD1 for the treatment of multiple sclerosis
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 14
作者:
Chen, Xuetao
;
Wu, Tingting
;
Du, Zhiyan
;
Kang, Wenjing
;
Xu, Rujun
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2024/02/27
BET
BD1
Bromodomain
Brain-permeable
Multiple sclerosis
Screening and optimization of phage display cyclic peptides against the WDR5 WBM site
期刊论文
OAI收割
RSC MEDICINAL CHEMISTRY, 2023, 页码: 10
作者:
Song, Lingyu
;
Cao, Jiawen
;
Chen, Lin
;
Du, Zhiyan
;
Zhang, Naixia
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/10/17
Discovery of 1H-Imidazo[4,5-b]pyridine Derivatives as Potent and Selective BET Inhibitors for the Management of Neuropathic Pain
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 13, 页码: 8725-8744
作者:
Chen, Xuetao
;
Cao, Danyan
;
Liu, Chihong
;
Meng, Fanying
;
Zhang, Zijian
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/10/17
Structure-Based of a Series of NSD2-PWWP1 Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 13, 页码: 9459-9477
作者:
Li, Na
;
Yang, Hong
;
Liu, Ke
;
Zhou, Liwei
;
Huang, Yuting
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2024/03/21
Structure-Based Discovery of Potent CARM1 Inhibitors for Solid Tumor and Cancer Immunology Therapy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 22, 页码: 16650-16674
作者:
Zhang, Zhuqing
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2022/06/15
Multi-omics characterization of WNT pathway reactivation to ameliorate BET inhibitor resistance in liver cancer cells
期刊论文
OAI收割
GENOMICS, 2021, 卷号: 113, 期号: 3, 页码: 1057-1069
作者:
Liu, Yuwei
;
Xue, Mengzhu
;
Cao, Danyan
;
Qin, Lihuai
;
Wang, Ying
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2021/08/17
Multi-omics
BET inhibitor responses
WNT pathway
Liver cancer
Precise therapy
Phage-Display Based Discovery and Characterization of Peptide Ligands against WDR5
期刊论文
OAI收割
MOLECULES, 2021, 卷号: 26, 期号: 5, 页码: 12
作者:
Cao, Jiawen
;
Fan, Tiantian
;
Li, Yanlian
;
Du, Zhiyan
;
Chen, Lin
  |  
收藏
  |  
浏览/下载:73/0
  |  
提交时间:2021/05/24
phage display
biopanning
WDR5
cocrystal structure
Rational Design and Evaluation of 6-(Pyrimidin-2-ylamino)-3,4-dihydroquinoxalin-2(1H)-ones as Polypharmacological Inhibitors of BET and Kinases
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 17, 页码: 9787-9802
作者:
Lv, Kaikai
;
Chen, Weicong
;
Chen, Danqi
;
Mou, Jie
;
Zhang, Huijie
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2020/12/21