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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [153]
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期刊论文 [206]
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Dynamic-GLEP: a dynamics-informed deep learning framework for ligand efficacy prediction in representative Class A GPCRs
期刊论文
OAI收割
BRIEFINGS IN BIOINFORMATICS, 2026, 卷号: 27, 期号: 1, 页码: 15
作者:
Chen, Zhiyi
;
Hao, Yongxin
;
Su, Yuhong
;
Agren, Hans
;
Chen, Mingan
  |  
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Discovery of novel selective PRMT5-MTA inhibitors through structure-based virtual screening
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2026, 卷号: 168, 页码: 17
作者:
Ma, Ning
;
Chen, Yang
;
Liang, Yiru
;
Chen, Xiaoxu
;
Song, Fengnan
  |  
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  |  
Mechanistic Insights into the Allosteric Regulation of P53 Y220C by Small-Molecule Stabilizers
期刊论文
OAI收割
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2025, 卷号: 65, 期号: 23, 页码: 12945-12958
作者:
Wen, Yiming
;
Niu, Buying
;
Meng, Jingyi
;
Chen, Danye
;
Li, Xutong
  |  
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  |  
Furo[2,3-
f
]quinazolin-7(6
H
)-one Derivatives as Potent, Selective, and Orally Bioavailable MAT2A Inhibitors for MTAP-Deficient Cancer Therapy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 22, 页码: 24213-24231
作者:
Shi, Zihan
;
Lin, Kexin
;
Lin, Lijie
;
Chen, Zhiyi
;
Xie, Zhiyin
  |  
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  |  
Unveiling conformation-selective regulation of the norepinephrine transporter
期刊论文
OAI收割
CELL, 2025, 卷号: 188, 期号: 24, 页码: 27
作者:
Zhang, Heng
;
Zhang, Tianwei
;
Wang, Dingyan
;
Dai, Antao
;
Mao, Jianhang
  |  
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  |  
Deep Learning-Driven Co-Assembly of Naturally Sourced Compound Nanoparticles for Potentiated Cancer Immunotherapy
期刊论文
OAI收割
ADVANCED FUNCTIONAL MATERIALS, 2025, 页码: 14
作者:
Shan, Yiming
;
Zhang, Zimei
;
Zhou, Huiling
;
Hou, Bo
;
Chen, Fangmin
  |  
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  |  
A nitrogen-containing diphyllin derivative C156-P1 exhibited broad-spectrum antiviral activity against
Flaviviridae
viruses by preventing endosomal acidification
期刊论文
OAI收割
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2025, 页码: 23
作者:
Chen, Guoquan
;
Li, Wanfei
;
Lam, Ka Hei
;
Hu, Mingyue
;
Wu, Qian
  |  
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Engineering STING Nanoadjuvants for spatiotemporally-tailored innate immunity stimulation and cancer vaccination therapy
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2025, 卷号: 16, 期号: 1, 页码: 21
作者:
Chen, Fangmin
;
Zhang, Huijuan
;
Li, Shiqin
;
Ren, Siyuan
;
Huang, Lujia
  |  
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  |  
NMRExtractor: leveraging large language models to construct an experimental NMR database from open-source scientific publications
期刊论文
OAI收割
CHEMICAL SCIENCE, 2025, 卷号: 16, 期号: 25, 页码: 11548-11558
作者:
Wang, Qinggong
;
Zhang, Wei
;
Chen, Mingan
;
Li, Xutong
;
Xiong, Zhaoping
  |  
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A Unified Strategy for Transition-Metal-Free Synthesis of Benzothienopyridines, Benzoselenopyridines, and Benzotelluropyridines and Related Analogues
期刊论文
OAI收割
ORGANIC LETTERS, 2025, 卷号: 27, 期号: 23, 页码: 6047-6053
作者:
Wen, Zhaoyue
;
Wu, Jianlian
;
Wang, Chun
;
Shen, Bingjie
;
Fu, Mingyue
  |  
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