中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共195条,第1-10条 帮助

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NMRExtractor: leveraging large language models to construct an experimental NMR database from open-source scientific publications 期刊论文  OAI收割
CHEMICAL SCIENCE, 2025, 卷号: 16, 期号: 25, 页码: 11548-11558
作者:  
Wang, Qinggong;  Zhang, Wei;  Chen, Mingan;  Li, Xutong;  Xiong, Zhaoping
  |  收藏  |  浏览/下载:1/0  |  提交时间:2025/08/20
A Unified Strategy for Transition-Metal-Free Synthesis of Benzothienopyridines, Benzoselenopyridines, and Benzotelluropyridines and Related Analogues 期刊论文  OAI收割
ORGANIC LETTERS, 2025, 卷号: 27, 期号: 23, 页码: 6047-6053
作者:  
Wen, Zhaoyue;  Wu, Jianlian;  Wang, Chun;  Shen, Bingjie;  Fu, Mingyue
  |  收藏  |  浏览/下载:1/0  |  提交时间:2025/08/20
Structural Optimization of Next-Generation TRK Inhibitors against Acquired Drug Resistance Mutations for the Treatment of Solid Tumors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 11, 页码: 11484-11501
作者:  
Xu, Zichao;  Liu, Yueling;  Wang, Peng;  Peng, Xia;  Cheng, Jiawei
  |  收藏  |  浏览/下载:1/0  |  提交时间:2025/08/20
Discovery of 3-(Fluoro-imidazolyl)pyridazine Derivatives as Potent STING Agonists with Antitumor Activity 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 10, 页码: 9864-9885
作者:  
Hou, Hui;  Zhou, Jingyi;  Sui, Qibang;  Zhang, Changfa;  Su, Zhaoming
  |  收藏  |  浏览/下载:11/0  |  提交时间:2025/07/25
Proteome-Wide Data Guides the Discovery of Lysine-Targeting Covalent Inhibitors Using DNA-Encoded Chemical Libraries 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 14
作者:  
Wu, Xinyuan;  Li, Shunyao;  Liang, Ting;  Yu, Qing;  Zhang, Yiwei
  |  收藏  |  浏览/下载:22/0  |  提交时间:2025/06/23
Targeting the histone reader ZMYND8 inhibits antiandrogen-induced neuroendocrine tumor transdifferentiation of prostate cancer 期刊论文  OAI收割
NATURE CANCER, 2025, 页码: 37
作者:  
Wang, Hanling;  Zhang, Sulin;  Pan, Qiang;  Guo, Jiacheng;  Li, Ni
  |  收藏  |  浏览/下载:14/0  |  提交时间:2025/05/27
IHCH9033, a novel class I HDAC inhibitor, synergizes with FLT3 inhibitor and rescues quizartinib resistance in FLT3-ITD AML via enhancing DNA damage response 期刊论文  OAI收割
EXPERIMENTAL HEMATOLOGY & ONCOLOGY, 2025, 卷号: 14, 期号: 1, 页码: 19
作者:  
Yao, Mingyue;  Yan, Wenzhong;  Wang, Yafang;  Zhao, Yu;  Xu, Xiaowei
  |  收藏  |  浏览/下载:25/0  |  提交时间:2025/04/01
Discovery of novel covalent stabilizers for p53 Y220C using structure-based drug discovery methods 期刊论文  OAI收割
MOLECULAR DIVERSITY, 2025, 页码: 14
作者:  
Wen, Yiming;  Xu, Peijia;  Chen, Yijie;  Meng, Jingyi;  Zheng, Mingyue
  |  收藏  |  浏览/下载:36/0  |  提交时间:2025/04/01
Harnessing the Magic Methyl Effect: Discovery of CLPP-2068 as a Novel HsClpP Activator for the Treatment of Diffuse Large B-Cell Lymphoma 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 4, 页码: 4287-4307
作者:  
Sun, Mingyang;  Chen, Beijing;  Teng, Dan;  Zhao, Hongshen;  Liao, Yilie
  |  收藏  |  浏览/下载:34/0  |  提交时间:2025/04/01
2-(1-Phenylvinyl)benzoic acid as a highly active leaving group for metal-free glycosylation 期刊论文  OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2025, 页码: 7
作者:  
  |  收藏  |  浏览/下载:26/0  |  提交时间:2025/04/01