中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共307条,第1-10条 帮助

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Design, synthesis and pharmacological evaluation of 1,2,3,4-tetrahydrobenzofuro[2,3-c] pyridine derivatives as p21-activated kinase 4 inhibitors for treatment of pancreatic cancer 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 1, 页码: 438-466
作者:  
Li, Yang;  Fang, Yan;  Chen, Xiaoyu;  Tong, Linjiang;  Feng, Fang
  |  收藏  |  浏览/下载:10/0  |  提交时间:2025/04/01
Structure-Based Drug Design of 2-Amino-[1,1′-biphenyl]-3-carboxamide Derivatives as Selective PKMYT1 Inhibitors for the Treatment of CCNE1-Amplified Breast Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 21
作者:  
Wang, Chaofan;  Fang, Yan;  Zhou, Ziqin;  Liu, Zhuoheng;  Feng, Fang
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/09/26
Branched-chain amino acid transaminase 1 confers EGFR-TKI resistance through epigenetic glycolytic activation 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2024, 卷号: 9, 期号: 1, 页码: 17
作者:  
Zhang, Tao;  Pan, Zilu;  Gao, Jing;  Wu, Qingqing;  Bai, Gang
  |  收藏  |  浏览/下载:16/0  |  提交时间:2024/10/21
Discovery of a Covalent Inhibitor That Overcame Resistance to Venetoclax in AML Cells Overexpressing BFL-1 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 36
作者:  
Lou, Jianfeng;  Zhou, Qianqian;  Lyu, Xilin;  Cen, Xinyi;  Liu, Chen
  |  收藏  |  浏览/下载:5/0  |  提交时间:2024/08/22
GFPBW1, a β-glucan from Grifola frondosa as vaccine adjuvant: APCs activation and maturation 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2024, 页码: 11
作者:  
He, Xiang;  Lu, Jiang-ling;  Liao, Wen-feng;  Long, Yi-ru;  Zhang, Xing
  |  收藏  |  浏览/下载:7/0  |  提交时间:2024/08/20
Discovery of a novel BTK inhibitor S-016 and identification of a new strategy for the treatment of lymphomas including BTK inhibitor-resistant lymphomas 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2024, 页码: 11
作者:  
Song, Pei-ran;  Wan, Zhi-peng;  Huang, Ge-ge;  Song, Zi-lan;  Zhang, Tao
  |  收藏  |  浏览/下载:66/0  |  提交时间:2024/07/12
A Novel IRAK4 Inhibitor DW18134 Ameliorates Peritonitis and Inflammatory Bowel Disease 期刊论文  OAI收割
MOLECULES, 2024, 卷号: 29, 期号: 8, 页码: 17
作者:  
Huang, Yuqing;  Ning, Yi;  Chen, Zhiwei;  Song, Peiran;  Tang, Haotian
  |  收藏  |  浏览/下载:14/0  |  提交时间:2024/05/31
Introduction and Safe Use of Gas Cylinders in China 期刊论文  OAI收割
ACS Sustainable Chem. Eng., 2024, 卷号: 2024, 期号: 12, 页码: 5496−5508
作者:  
Ming-Ming Yu;  Zhenghao hang Zhang;  Gui-Ling Guan;  Bhagyesha Patil;  Priya Darshini Srinivasan
  |  收藏  |  浏览/下载:12/0  |  提交时间:2024/12/23
A novel strategy for treating oncogene-mutated tumors by targeting tumor microenvironment and synergistically enhancing anti-PD-1 immunotherapy 期刊论文  OAI收割
CANCER COMMUNICATIONS, 2024, 页码: 5
作者:  
Liu, Yingqiang;  Tong, Linjiang;  Zhang, Mengge;  Zhang, Qi;  Liu, Qiupei
  |  收藏  |  浏览/下载:37/0  |  提交时间:2024/03/13
From bench to bedside: current development and emerging trend of KRAS-targeted therapy 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 18
作者:  
Chen, Yi;  Liu, Qiu-pei;  Xie, Hua;  Ding, Jian
  |  收藏  |  浏览/下载:54/0  |  提交时间:2024/01/16