中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共19条,第1-10条 帮助

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Discovery of aldolase A inhibitors via high-throughput screening assay based on an enzymatic coupling reaction 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 128, 页码: 7
作者:  
Xiong, Qingwen;  Qian, Rongyu;  Huang, Qingcheng;  Liu, Jingqiu;  Zhou, Chen
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Purification, structural characterization, and anti-ulcerative colitis activity of a novel pectin-like polysaccharide AH-H4-1 from Alhagi honey 期刊论文  OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2025, 卷号: 319, 页码: 16
作者:  
Wang, Zhe;  Chi, Yaping;  Wang, Menghua;  Zhou, Qianqian;  Yan, Zexiang
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Structure-Based Design and Discovery of a Potent and Cell-Active LC3A/B Covalent Inhibitor 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 14, 页码: 12184-12204
作者:  
Zhou, Zhenfei;  Huang, Siqi;  Fan, Shijie;  Li, Xueyuan;  Wang, Chengyu
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Uncovering PROTAC Sensitivity and Efficacy by Multidimensional Proteome Profiling: A Case for STAT3 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 6, 页码: 4804-4818
作者:  
Suo, Yuying;  Du, Daohai;  Chen, Chao;  Zhu, Hongwen;  Wang, Xiongjun
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A RhoA structure with switch II flipped outward revealed the conformational dynamics of switch II region 期刊论文  OAI收割
JOURNAL OF STRUCTURAL BIOLOGY, 2023, 卷号: 215, 期号: 2, 页码: 107942
作者:  
Jiang, Hao;  Zu, Shijia;  Lu, Yu;  Sun, Zhongya;  Adeerjiang, Akejiang
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Thimerosal, a competitive thioredoxin reductase 1 (TrxR1) inhibitor discovered via high-throughput screening 期刊论文  OAI收割
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2023, 卷号: 650, 页码: 117-122
作者:  
Ni, Yicheng;  Luo, Zhongyuan;  Lv, Yixin;  Ma, Shuyuan;  Luo, Cheng
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(-)-Epigallocatechin Gallate is a Noncompetitive Inhibitor of NAD Kinase 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2022, 页码: 8
作者:  
Liu, Tonghai;  Shi, Wenjia
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The discovery of a non-competitive GOT1 inhibitor, hydralazine hydrochloride, via a coupling reaction-based high-throughput screening assay 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2022, 卷号: 73, 页码: 6
作者:  
Wu, Qiqi;  Sun, Zhongya;  Chen, Zhifeng;  Liu, Jingqiu;  Ding, Hong
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Computational and Structure-Based Development of High Potent Cell-Active Covalent Inhibitor Targeting the Peptidyl-Prolyl Isomerase NIMA-Interacting-1 (Pin1) 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 3, 页码: 2174-2190
作者:  
Liu, Liping;  Zhu, Rui;  Li, Jiacheng;  Pei, Yuan;  Wang, Shuangshuang
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Structural basis of ketamine action on human NMDA receptors 期刊论文  OAI收割
NATURE, 2021, 卷号: 596, 期号: 7871, 页码: 301-+
作者:  
Zhang, Youyi;  Ye, Fei;  Zhang, Tongtong;  Lv, Shiyun;  Zhou, Liping
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