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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [32]
广州地球化学研究所 [4]
新疆理化技术研究所 [4]
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期刊论文 [59]
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Design and Development of a Novel Oral 4′-Fluorouridine Double Prodrug VV261 against SFTSV
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 9, 页码: 9811-9826
作者:
Cheng, Yong
;
Zheng, Wei
;
Dong, Xinru
;
Sun, Tengxiao
;
Xu, Mengwei
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/06/23
F-CPI: A Multimodal Deep Learning Approach for Predicting Compound Bioactivity Changes Induced by Fluorine Substitution
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 13
作者:
Zhang, Qian
;
Yin, Wenhai
;
Chen, Xinyao
;
Zhou, Aimin
;
Zhang, Guixu
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2025/02/28
Hygroscopic Properties of Plateau Surface Salts: Insights from Chemical Composition and Isotope Signatures
期刊论文
OAI收割
ACS EARTH AND SPACE CHEMISTRY, 2024, 卷号: 8, 期号: 5, 页码: 1111-1121
作者:
Hao, Yuxin
;
Qiu, Yuhe
;
Li, Jun
;
Liu, Wanyu
;
Chen, Lanxiadi
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/09/13
hygroscopicity
salt evaporites
geochemicalisotopes
sulfur
chlorine
atmosphere
Identification of Dihydrobenzofuran Neolignans as Novel PDE4 Inhibitors and Evaluation of Antiatopic Dermatitis Efficacy in DNCB-Induced Mice Model
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 6, 页码: 4855-4869
作者:
Gu, Chenming
;
Liu, Jiayuan
;
Qian, Fei
;
Yu, Wenchao
;
Huang, Doudou
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/05/07
Glimepiride, a novel soluble epoxide hydrolase inhibitor, protects against heart failure via increasing epoxyeicosatrienoic acids
期刊论文
OAI收割
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY, 2023, 卷号: 185, 页码: 13-25
作者:
Zhao, Chengcheng
;
Jiang, Xiangrui
;
Peng, Liyuan
;
Zhang, Yan
;
Li, Huihui
  |  
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2024/01/16
Heart failure
Hypertrophy
Epoxyeicosatrienoic acids
Soluble epoxide hydrolase
TPN10475 alleviates concanavalin A-induced autoimmune hepatitis by limiting T cell development and function through inhibition of PI3K-AKT pathway
期刊论文
OAI收割
INTERNATIONAL IMMUNOPHARMACOLOGY, 2023, 卷号: 125, 页码: 13
作者:
Wang, Chun
;
Han, Mengyao
;
Li, Xinhang
;
Lv, Jie
;
Zhuang, Wei
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2024/01/16
AIH
T cell
Pro-inflammatory
IFN-gamma
PI3K-AKT
Structure-based development and preclinical evaluation of the SARS-CoV-2 3C-like protease inhibitor simnotrelvir
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 15
作者:
Jiang, Xiangrui
;
Su, Haixia
;
Shang, Weijuan
;
Zhou, Feng
;
Zhang, Yan
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2024/03/25
A new Einstein coefficient method for mesopause–lower thermosphere atmosphere temperature retrieval under a non-local thermal equilibrium situation
期刊论文
OAI收割
Optics Express, 2023, 卷号: 31, 期号: 19, 页码: 30413-30434
作者:
Li, Haotian
;
Feng, Yutao
;
Li, Faquan
;
Wang, Houmao
;
Hu, Xiangrui
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2023/10/26
Synthesis, cytotoxicity, and pharmacokinetic evaluations of niclosamide analogs for anti-SARS-CoV-2
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 253, 页码: 11
作者:
Li, Rui
;
Zhang, Zherui
;
Huang, Shuhong
;
Peng, Ke
;
Jiang, Hualiang
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2023/10/17
SARS-CoV-2
Niclosamide analogs
Cytotoxicity
Pharmacokinetic
SKP2 inhibition
Preventive and therapeutic benefits of nelfinavir in rhesus macaques and human beings infected with SARS-CoV-2
期刊论文
OAI收割
Signal Transduction and Targeted Therapy, 2023, 卷号: 8, 期号: 5, 页码: 2384-2391
作者:
Xu, Zhijian
;
Shi, Danrong
;
Han, Jianbao
;
Ling, Yun
;
Jiang, Xiangrui
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2024/03/27