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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [91]
计算技术研究所 [7]
西北高原生物研究所 [6]
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期刊论文 [146]
会议论文 [2]
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生命有机化学 [2]
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Discovery of a Potent, selective and orally bioavailable CDK9 degrader for targeting transcription regulation in Triple-Negative breast cancer
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 153, 页码: 16
作者:
Nie, Hui-Jun
;
Li, Ben-Fu
;
Sun, Jingya
;
Yuan, Yali
;
Zhang, Zhi-Gao
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/11/26
Triple-negative breast cancer
Targeting transcription regulation
Orally bioavailable degrader
PROTAC
Cyclin-dependent Kinase 9
Discovery of Alkyl Conjugated Diene Diacids as Novel ACLY Inhibitors
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 44, 期号: 11, 页码: 3476-3489
作者:
Cheng, Tingting
;
Song, Gaolei
;
Cheng, Long
;
Wang, Fan
;
Sun, Xinyu
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2025/02/28
metabolic diseases
ATP-citrate lyase (ACLY)
lipogenesis
ACLY inhibitors
dienyldicarboxylic acid
DPU-Direct: Unleashing Remote Accelerators via Enhanced RDMA for Disaggregated Datacenters
期刊论文
OAI收割
IEEE TRANSACTIONS ON COMPUTERS, 2024, 卷号: 73, 期号: 8, 页码: 2081-2095
作者:
Liao, Yunkun
;
Wu, Jingya
;
Lu, Wenyan
;
Li, Xiaowei
;
Yan, Guihai
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2024/12/06
Central Processing Unit
Engines
Jitter
Computers
Pipelines
Programming
Encryption
Disaggregated datacenter
SmartNIC
RDMA
hardware accelerator
Discovery of Orally Bioavailable and Potent CDK9 Inhibitors for Targeting Transcription Regulation in Triple-Negative Breast Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 12, 页码: 10035-10056
作者:
Wang, Wen-Jing
;
Gao, Lixin
;
Wang, Simei
;
Huang, Wensi
;
Meng, Xin-Yu
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/08/20
Simultaneous determination of BGT-002 and its acyl glucuronide metabolite ZM326E-M2 in human plasma by liquid chromatography-tandem mass spectrometry and its application to a pharmacokinetic study
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2024, 卷号: 243, 页码: 8
作者:
Zhu, Xueran
;
Cui, Shumin
;
Liu, Xinjing
;
Zhang, Mei
;
Xie, Zhifu
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/05/31
ATP-Citrate Lyase
BGT-002
Acyl glucuronide metabolite
Pseudo-MRM
LC-MS/MS
Pharmacokinetics
Polyphenol Compound 18a Modulates UCP1-Dependent Thermogenesis to Counteract Obesity
期刊论文
OAI收割
BIOMOLECULES, 2024, 卷号: 14, 期号: 6, 页码: 21
作者:
Wen, Xueping
;
Song, Yufei
;
Zhang, Mei
;
Kang, Yiping
;
Chen, Dandan
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/08/22
18a
adipocytes
polyphenols
thermogenesis
UCP1
Exploring the Structural Plasticity Mechanism of Corticospinal Tract during Stroke Rehabilitation Based Automated Fiber Quantification Tractography
期刊论文
OAI收割
NEUROREHABILITATION AND NEURAL REPAIR, 2024, 页码: 12
作者:
Zhang, Haojie
;
Zhao, Jun
;
Fan, Lingzhong
;
Wu, Xia
;
Li, Fang
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/05/30
automated fiber quantification
corticospinal tract
MRI
rehabilitation
stroke
structural plasticity
DRAK2 suppresses autophagy by phosphorylating ULK1 at Ser
56
to diminish pancreatic β cell function upon overnutrition
期刊论文
OAI收割
SCIENCE TRANSLATIONAL MEDICINE, 2024, 卷号: 16, 期号: 733, 页码: 16
作者:
Lu, Yuting
;
Xu, Junyu
;
Li, Yufeng
;
Wang, Ruoran
;
Dai, Chengqiu
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2024/03/13
AMPK phosphorylation of FNIP1 (S220) controls mitochondrial function and muscle fuel utilization during exercise
期刊论文
OAI收割
SCIENCE ADVANCES, 2024, 卷号: 10, 期号: 6, 页码: 15
作者:
Xiao, Liwei
;
Yin, Yujing
;
Sun, Zongchao
;
Liu, Jing
;
Jia, Yuhuan
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/05/31
Increased frequency of extreme climatic events weakens the community stability of natural grassland under directional climate changes by reducing resilience
期刊论文
OAI收割
GLOBAL ECOLOGY AND BIOGEOGRAPHY, 2024, 卷号: 33, 期号: 6
作者:
Liu, Peipei
;
Lv, Wangwang
;
Sun, Jianping
;
Piao, Shilong
;
Wang, Yanfen
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/11/27