中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [8]
金属研究所 [2]
化学研究所 [1]
上海有机化学研究所 [1]
采集方式
OAI收割 [12]
内容类型
期刊论文 [12]
发表日期
2023 [1]
2022 [2]
2016 [2]
2009 [3]
2007 [2]
2005 [1]
更多
学科主题
天然产物有机化学 [1]
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Enhancing the mechanical property of laser powder bed fusion CoCrMo alloy by tailoring the microstructure and phase constituent
期刊论文
OAI收割
MATERIALS SCIENCE AND ENGINEERING A-STRUCTURAL MATERIALS PROPERTIES MICROSTRUCTURE AND PROCESSING, 2023, 卷号: 862, 页码: 14
作者:
Zhang, Yu
;
Lin, Wenhu
;
Zhai, Zirong
;
Wu, Yingna
;
Yang, Rui
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2023/05/09
CoCrMo alloy
Laser powder bed fusion
Cellular structure
Mechanical property
Phase constituent
Discovery of 10H-Benzo[b]pyrido[2,3-e][1,4]oxazine AXL Inhibitors via Structure-Based Drug Design Targeting c-Met Kinase
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 15
作者:
Zhan, Zhengsheng
;
Ji, Yinchun
;
Su, Haixia
;
Fang, Chen
;
Peng, Xia
  |  
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2023/04/10
On the orientation dependent microstructure and mechanical behavior of Hastelloy X superalloy fabricated by laser powder bed fusion
期刊论文
OAI收割
MATERIALS SCIENCE AND ENGINEERING A-STRUCTURAL MATERIALS PROPERTIES MICROSTRUCTURE AND PROCESSING, 2022, 卷号: 844, 页码: 14
作者:
Huang, Ziliang
;
Zhai, Zirong
;
Lin, Wenhu
;
Chang, Hai
;
Wu, Yingna
  |  
收藏
  |  
浏览/下载:46/0
  |  
提交时间:2022/07/14
Laser powder bed fusion
Hastelloy X
Anisotropy
Mechanical properties
Orientation dependent
Discovery of 6-(difluoro(6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b] [1,2,4]triazin-3-yl)methyl)quinoline as a highly potent and selective c-Met inhibitor
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 239-251
作者:
Zhan, Zhengsheng
;
Peng, Xia
;
Liu, Qiufeng
;
Chen, Fang
;
Ji, Yinchun
  |  
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2019/01/08
Antitumor
c-Met
Kinase inhibitor
Triazolotriazines
Discovery of 1,3-Diaryl-pyridones as Potent VEGFR-2 Inhibitors: Design, Synthesis, and Biological Evaluation
期刊论文
OAI收割
CHEMICAL BIOLOGY & DRUG DESIGN, 2016, 卷号: 87, 期号: 5, 页码: 694-703
作者:
Yan, Wei
;
Huang, Zhaoru
;
Wang, Zhengyu
;
Cao, Sufen
;
Tong, Linjiang
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2019/01/08
1
3-Diaryl-pyridone
angiogenesis
anticancer agent
Chan-Lam coupling
VEGFR-2 inhibitors
Synthesis and biological activity of novel shikonin analogues
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 卷号: 19, 期号: 3, 页码: 735-737
作者:
Wang, Wenjing
;
Dai, Mei
;
Zhu, Caihua
;
Zhang, Jiangang
;
Lin, Liping
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
Shikonin analogue
Synthesis
Cytotoxicity
Hypoxia-inducible factor 1 alpha
Antitumor activity of a novel EGFR tyrosine kinase inhibitor against human lung carcinoma in vitro and in vivo
期刊论文
OAI收割
INVESTIGATIONAL NEW DRUGS, 2009, 卷号: 27, 期号: 1, 页码: 1-11
作者:
Xiong, Xishan
;
Fu, Lili
;
Wang, Li
;
Cai, Houan
;
Li, Lin
  |  
收藏
  |  
浏览/下载:46/0
  |  
提交时间:2019/01/08
EGFR
SPC-A1
tyrosine kinase inhibitor
quinazoline
non-small cell lung cancer
ga3anewgambogicacidderivativeexhibitspotentantitumoractivitiesinvitroviaapoptosisinvolvedmechanisms
期刊论文
OAI收割
actapharmacologicasinica, 2009, 卷号: 30, 期号: 3, 页码: 346
作者:
Hua XIE
;
Yuxin QIN
;
Yunlong ZHOU
;
Linjiang TONG
;
Liping LIN
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2020/07/01
DRUG DISCOVERY
CELLS
BAX
PROTEIN
TRANSLOCATION
CYTOTOXICITY
PATHWAY
BINDING
DOMAIN
DEATH
gambogic acid
GA3
antitumor
apoptosis
caspase
Bcl-2
cytochrome c
Gambogic acid inhibits the catalytic activity of human topoisomerase II alpha by binding to its ATPase domain
期刊论文
OAI收割
MOLECULAR CANCER THERAPEUTICS, 2007, 卷号: 6, 期号: 9, 页码: 2429-2440
作者:
Qin, Yuxin
;
Meng, Linghua
;
Hu, Chaoxin
;
Duan, Wenhu
;
Zuo, Zhili
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/01/08
Caspase-8 preferentially senses the apoptosis-inducing action of NG-18, a gambogic acid derivative, in human leukemia HL-60 cells
期刊论文
OAI收割
CANCER BIOLOGY & THERAPY, 2007, 卷号: 6, 期号: 5, 页码: 691-696
作者:
Tao, Zhijian
;
Zhou, Yunlong
;
Lu, Jinjian
;
Duan, Wenhu
;
Qin, Yuxin
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2019/01/08
gambogic acid
NG-18
HL-60
apoptosis
caspase-8
Bcl-2
anti-tumor