中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [45]
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期刊论文 [62]
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Residue-Selective Inhibitors Discovery via Covalent DNA-Encoded Chemical Libraries with Diverse Warheads
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2025, 卷号: 147, 期号: 18, 页码: 15469-15481
作者:
Wu, Xinyuan
;
Pan, Jiayi
;
Fan, Rufeng
;
Zhang, Yiwei
;
Wang, Chao
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/06/23
Proteome-Wide Data Guides the Discovery of Lysine-Targeting Covalent Inhibitors Using DNA-Encoded Chemical Libraries
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 14
作者:
Wu, Xinyuan
;
Li, Shunyao
;
Liang, Ting
;
Yu, Qing
;
Zhang, Yiwei
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/06/23
Activity-based protein profiling data
Covalent DNA-encoded chemical library
Covalent ligand selection
Lysine-targeting covalent inhibitors
Age-related decline in CD8
+
tissue resident memory T cells compromises antitumor immunity
期刊论文
OAI收割
NATURE AGING, 2024, 卷号: 4, 期号: 12, 页码: 1828-+
作者:
Pei, Siyu
;
Deng, Xiuyu
;
Yang, Ruirui
;
Wang, Hui
;
Shi, Jian-Hong
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2025/02/28
Covalent DNA-Encoded Library Workflow Drives Discovery of SARS-CoV-2 Nonstructural Protein Inhibitors
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2024, 页码: 14
作者:
Wang, Xudong
;
Xiong, Liwei
;
Zhu, Ying
;
Liu, Sixiu
;
Zhao, Wenfeng
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2024/12/25
Enhancing the Predictive Power of Machine Learning Models through a Chemical Space Complementary DEL Screening Strategy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 12
作者:
Suo, Yanrui
;
Qian, Xu
;
Xiong, Zhaoping
;
Liu, Xiaohong
;
Wang, Chao
  |  
收藏
  |  
浏览/下载:98/0
  |  
提交时间:2024/11/26
Amelioration of nonalcoholic fatty liver disease by inhibiting the deubiquitylating enzyme RPN11
期刊论文
OAI收割
CELL METABOLISM, 2024, 卷号: 36, 期号: 10, 页码: 25
作者:
Zhou, Bing
;
Luo, Yunchen
;
Bi, Hanqi
;
Zhang, Ni
;
Ma, Mingyue
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2024/11/26
Study of high-precision time transfer method enhanced by PPP-AR/PPP-RTK
期刊论文
OAI收割
MEASUREMENT SCIENCE AND TECHNOLOGY, 2024, 卷号: 35, 期号: 9, 页码: 15
作者:
Liu, Mingyue
;
Tu, Rui
;
Chen, Qiushi
;
Li, Qi
;
Chen, Junmei
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2025/04/03
time transfer
integer ambiguity fixing
PPP-AR
PPP-RTK
Generic protein-ligand interaction scoring by integrating physical prior knowledge and data augmentation modelling
期刊论文
OAI收割
NATURE MACHINE INTELLIGENCE, 2024, 页码: 21
作者:
Cao, Duanhua
;
Chen, Geng
;
Jiang, Jiaxin
;
Yu, Jie
;
Zhang, Runze
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2024/07/12
Study of Fast and Reliable Time Transfer Methods Using Low Earth Orbit Enhancement
期刊论文
OAI收割
REMOTE SENSING, 2024, 卷号: 16, 期号: 11, 页码: 20
作者:
Liu, Mingyue
;
Tu, Rui
;
Chen, Qiushi
;
Li, Qi
;
Chen, Junmei
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2025/04/03
low Earth orbit satellite
precise point positioning
global navigation satellite system
time transfer
Structure-based design of pan-coronavirus inhibitors targeting host cathepsin L and calpain-1
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2024, 卷号: 9, 期号: 1, 页码: 14
作者:
Xie, Xiong
;
Lan, Qiaoshuai
;
Zhao, Jinyi
;
Zhang, Sulin
;
Liu, Lu
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2024/05/07