中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共103条,第1-10条 帮助

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Identification of [1,2,4]Triazolo[4,3-a]pyrazine PARP1 inhibitors with overcome acquired resistance activities 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 259, 页码: 19
作者:  
Wang, Pingyuan;  Zhu, Wen-Ting;  Wang, Yajing;  Song, Shan-Shan;  Xi, Yong
  |  收藏  |  浏览/下载:59/0  |  提交时间:2023/10/17
Proteasome inhibitors reduce CD73 expression partly via decreasing p-ERK in NSCLC cells 期刊论文  OAI收割
LIFE SCIENCES, 2023, 卷号: 332, 页码: 10
作者:  
Su, Ai-Ling;  Tian, Chang-Qing;  Ou, Ying-Jie;  Bao, Xu-Bin;  Huan, Xia-Juan
  |  收藏  |  浏览/下载:10/0  |  提交时间:2023/12/08
Thioparib inhibits homologous recombination repair, activates the type I IFN response, and overcomes olaparib resistance 期刊论文  OAI收割
EMBO MOLECULAR MEDICINE, 2023, 页码: 24
作者:  
Wang, Li-Min;  Wang, Pingyuan;  Chen, Xiao-Min;  Yang, Hui;  Song, Shan-Shan
  |  收藏  |  浏览/下载:21/0  |  提交时间:2023/04/10
Loss of VOPP1 Contributes to BET Inhibitor Acquired Resistance in Non-Small Cell Lung Cancer Cells 期刊论文  OAI收割
MOLECULAR CANCER RESEARCH, 2022, 卷号: 20, 期号: 12, 页码: 1785-1798
作者:  
Sun, Lin;  Wu, Qian;  Huan, Xia-Juan;  Tian, Chang-Qing;  Wang, Ying-Qing
  |  收藏  |  浏览/下载:14/0  |  提交时间:2024/03/21
Design, synthesis and pharmacological evaluation of new PARP1 inhibitors by merging pharmacophores of olaparib and the natural product alantolactone 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 240, 页码: 114574
作者:  
Kayumov, Muzaffar;  Jia, Li;  Pardaev, Azizbek;  Song, Shan-Shan;  Mirzaakhmedov, Sharafitdin
  |  收藏  |  浏览/下载:19/0  |  提交时间:2024/03/21
SOMCL-19-133, a novel, selective, and orally available inhibitor of NEDD8-activating enzyme (NAE) for cancer therapy 期刊论文  OAI收割
NEOPLASIA, 2022, 卷号: 32, 页码: 12
作者:  
Zhou, Li-Na;  Xiong, Chaodong;  Cheng, Yong-Jun;  Song, Shan-Shan;  Bao, Xu-Bin
  |  收藏  |  浏览/下载:14/0  |  提交时间:2023/04/10

Identification of 2-substituted pyrrolo[1,2-b]pyridazine derivatives as new PARP-1 inhibitors (vol 31, 127710, 2021)

期刊论文  OAI收割

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2022, 卷号: 56, 页码: 1
作者:  
Xiang, Hao-Yue;  Chen, Jian-Yang;  Huan, Xia-Juan;  Chen, Yi;  Gao, Zhao-bing
  |  收藏  |  浏览/下载:22/0  |  提交时间:2022/06/15
Repeated treatments of Capan-1 cells with PARP1 and Chk1 inhibitors promote drug resistance, migration and invasion 期刊论文  OAI收割
CANCER BIOLOGY & THERAPY, 2022, 页码: 14
作者:  
Guo, Ne;  Li, Meng-Zhu;  Wang, Li-Min;  Chen, Hua-Dong;  Song, Shan-Shan
  |  收藏  |  浏览/下载:27/0  |  提交时间:2022/06/15
TNKS inhibitors potentiate proliferative inhibition of BET inhibitors via reducing beta-Catenin in colorectal cancer cells 期刊论文  OAI收割
AMERICAN JOURNAL OF CANCER RESEARCH, 2022, 卷号: 12, 期号: 3, 页码: 1069-+
作者:  
Wu, Qian;  Xuan, Yi-Fei;  Su, Ai-Ling;  Bao, Xu-Bin;  Miao, Ze-Hong
  |  收藏  |  浏览/下载:27/0  |  提交时间:2022/06/15
The cell-impermeable Ru(II) polypyridyl complex as a potent intracellular photosensitizer under visible light irradiation via ion-pairing with suitable lipophilic counter-anions 期刊论文  OAI收割
FREE RADICAL BIOLOGY AND MEDICINE, 2021, 卷号: 171, 页码: 69-79
作者:  
Yan, Zhu-Ying;  Chen, Jing;  Shao, Jie;  Jiao, Ze-Qing;  Tang, Tian-Shu
  |  收藏  |  浏览/下载:12/0  |  提交时间:2021/12/22