中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [6]
采集方式
OAI收割 [6]
内容类型
期刊论文 [6]
发表日期
2024 [2]
2022 [1]
2021 [3]
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Discovery of Novel 2-Aminopyridine-Based and 2-Aminopyrimidine-Based Derivatives as Potent CDK/HDAC Dual Inhibitors for the Treatment of Refractory Solid Tumors and Hematological Malignancies
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 17, 页码: 15220-15245
作者:
Saidahmatov, Abdusaid
;
Li, Jianan
;
Xu, Shihao
;
Hu, Xiaobei
;
Gao, Xiangqian
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/10/21
Development of Potent MALT1 Inhibitors Featuring a Novel "2-Thioxo-2,3-dihydrothiazolo[4,5-
d
]pyrimidin-7(6
H
)-one" Scaffold for the Treatment of B Cell Lymphoma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 4, 页码: 2884-2906
作者:
Liang, Xuewu
;
Yu, Haolan
;
Liang, Renwen
;
Feng, Zhuanghui
;
Saidahmatov, Abdusaid
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2024/04/09
Discovery of Novel Pyrrolo[2,3-d]pyrimidine-based Derivatives as Potent JAK/HDAC Dual Inhibitors for the Treatment of Refractory Solid Tumors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 2, 页码: 1243-1264
作者:
Liang, Xuewu
;
Tang, Shuai
;
Liu, Xuyi
;
Liu, Yingluo
;
Xu, Qifu
  |  
收藏
  |  
浏览/下载:52/0
  |  
提交时间:2022/06/15
Rational Design and Development of Novel CDK9 Inhibitors for the Treatment of Acute Myeloid Leukemia
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14647-14663
作者:
Han, Xu
;
Song, Ning
;
Saidahmatov, Abdusaid
;
Wang, Peipei
;
Wang, Yong
  |  
收藏
  |  
浏览/下载:75/0
  |  
提交时间:2021/12/16
Efficient Synthesis and Docking Analysis of Selective CDK9 Inhibitor NVP-2
期刊论文
OAI收割
Pharmaceutical Fronts, 2021, 期号: 3, 页码: E50-E55
作者:
Saidahmatov, Abdusaid
;
Liang, Xue-Wu
;
Shi, Yuqiang
;
Han, Xu
;
Liu, Hong
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2024/03/14
NVP-2
CDK9 inhitor
efficient synthesis
docking analysis
Synthesis of Pyrazolo[1,2-a]cinnolines via Rhodium(III)-Catalyzed [4+2] Annulation Reactions of Pyrazolidinones with Sulfoxonium Ylides
期刊论文
OAI收割
ADVANCED SYNTHESIS & CATALYSIS, 2021, 页码: 8
作者:
Hu, Shulei
;
Han, Xu
;
Xie, Xiong
;
Fang, Feifei
;
Wang, Yong
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2021/08/17
annulation reactions
C-H activation
pyrazolidinone
Rhodium (III)-catalyzed
sulfoxonium ylide