中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [27]
化学研究所 [5]
金属研究所 [3]
中国科学院大学 [3]
数学与系统科学研究院 [1]
国家天文台 [1]
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OAI收割 [41]
iSwitch采集 [3]
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期刊论文 [44]
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2025 [2]
2024 [3]
2023 [5]
2022 [3]
2021 [2]
2019 [1]
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Energy & F... [1]
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物理化学与绿色催化 [1]
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Diazonium-based derivatization for enhanced detection of phosphorylated metabolites by LC-MS in cells
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2025, 卷号: 255, 页码: 7
作者:
Wang, Yikang
;
Lin, Feifei
;
Zhu, Guozheng
;
Zhou, Xiaoxue
;
Hu, Youhong
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2025/04/01
Phosphorylated metabolite
Derivatization
Chromatographic separation
Quantitative analysis
LC-MS
Discovery of novel biaryl urea derivatives against IL-1/3 release with low toxicity based on NEK7 inhibitor
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 283, 页码: 12
作者:
Wang, Leibo
;
Zhu, Kehan
;
Tian, Ziyang
;
Wang, Haoyu
;
Jia, Yulei
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2025/01/14
NLRP3 inflammasome
NEK7
NLRP3-NEK7
Inhibitors
C(sp
3
)-H Carbonylative Cyclization of Hydrazones with CO
2
: Synthesis of Pyrazolone Derivatives
期刊论文
OAI收割
JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 89, 期号: 24, 页码: 18746-18751
作者:
Wang, Kai
;
Ouyang, Jun
;
Liu, Huan
;
Yin, Lijun
;
Yang, Kuoqi
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/01/14
Single Amine or Guanidine Modification on Norvancomycin and Vancomycin to Overcome Multidrug-Resistance through Augmented Lipid II Binding and Increased Membrane Activity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 22, 页码: 20639-20663
作者:
Bian, Xiaolei
;
Chen, Zhifu
;
Li, Fang
;
Xie, Yuanyuan
;
Li, Yi
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/12/11
A novel phthalazinone derivative as a capsid assembly modulator inhibits hepatitis B virus expression
期刊论文
OAI收割
ANTIVIRAL RESEARCH, 2024, 卷号: 221, 页码: 14
作者:
Yang, Li
;
Gong, Ying
;
Liu, Feifei
;
Chen, Wuhong
;
Wang, Xinran
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2024/02/19
Hepatitis B virus
Capsid assembly
Phthalazinone derivatives
Apoptosis
Crop/Plant Modeling Supports Plant Breeding II. Guidance of Functional Plant Phenotyping for Trait Discovery
期刊论文
OAI收割
PLANT PHENOMICS, 2023, 卷号: 5, 页码: 19
作者:
Zhang, Pengpeng
;
Huang, Jingyao
;
Ma, Yuntao
;
Wang, Xiujuan
;
Kang, Mengzhen
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2024/02/22
A prodrug of the capsid assembly modulator improved druggability and lowing HBsAg and HBeAg for the treatment of chronic hepatitis B
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 257, 页码: 8
作者:
Chen, Wuhong
;
Gong, Ying
;
Long, Guozhang
;
Wang, Xinran
;
Yang, Yurong
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2023/10/17
HBV
Capsid assembly modulators
Prodrug
Hepatitis B surface antigen
Discovery of selective NaV1.8 inhibitors based on 5-chloro-2-(4,4-difluor- oazepan-1-yl)-6-methyl nicotinamide scaffold for the treatment of pain
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 254, 页码: 12
作者:
Qin, Hui
;
Wei, Aihuan
;
Wang, Yunqi
;
Wang, Linlin
;
Xu, Haiyan
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2023/10/17
Pain
Non-addictive analgesics
Na V 1
8-selective inhibitors
Bicyclic aromatic groups
Discovery of (S)-N-(2-Amino-4-fluorophenyl)-4-(1-(3-(4-((dimethylamino)methyl)phenyl)-6-oxopyridazin-1(6H)-yl)ethyl)benzamide as Potent Class I Selective HDAC Inhibitor for Oral Anticancer Drug Candidate
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 10, 页码: 7016-7037
作者:
Li, Daqiang
;
Zhang, Zhuo
;
Li, Yalei
;
Wang, Xinyi
;
Zhong, Hanyue
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/10/17
Experimental Study on the Depressurization of Methane Hydrate in the Clayey Silt Sediments via Hydraulic Fracturing
期刊论文
OAI收割
ENERGY & FUELS, 2023, 卷号: 37, 期号: 6, 页码: 4377
作者:
Wang, Xiaochu
;
Sun, Youhong
;
Chen, Hangkai
;
Peng, Saiyu
;
Jiang, Shuhui
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/08/02