中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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Design, synthesis and pharmacological evaluation of 1,2,3,4-tetrahydrobenzofuro[2,3-c] pyridine derivatives as p21-activated kinase 4 inhibitors for treatment of pancreatic cancer
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 1, 页码: 438-466
作者:
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浏览/下载:10/0
  |  
提交时间:2025/04/01
P21-activated kinase 4
Tetrahydrobenzofuro[2
3-c]pyridine
Structure-activity relationship
Allosteric inhibitor
Pharmacokinetics properties
Kinase selectivity
Pancreatic cancer
Immune infiltration
Design, Synthesis, and Biological Evaluation of Novel Diaminopyrimidine Macrocycles as Fourth Generation Reversible EGFR Inhibitors That Overcome Clinical Resistance to Osimertinib Mediated by C797S Mutation
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 22, 页码: 20531-20558
作者:
Hu, Shiliang
;
Tong, Linjiang
;
Qin, Qiao
;
Wen, Jiaxin
;
Li, Yan
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收藏
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浏览/下载:8/0
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提交时间:2024/12/11
Single-cell mapping of peripheral blood mononuclear cells reveals key transcriptomic changes favoring coronary artery lesion in IVIG-resistant Kawasaki disease
期刊论文
OAI收割
HELIYON, 2024, 卷号: 10, 期号: 18, 页码: 15
作者:
Zheng, Yuanzheng
;
Zhou, Yan
;
Zhu, Di
;
Fu, Xing
;
Xie, Cao
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2024/10/21
Kawasaki disease
IVIG-Resistant
Single cell RNA-Sequencing
Coronary artery lesion
Coupling higher-order probability weighted moments with norming constants method for non-stationary annual maximum flood frequency analysis
期刊论文
OAI收割
JOURNAL OF HYDROLOGY, 2024, 卷号: 641, 页码: 131832
作者:
Chen, Fei
;
Sang, Yan-Fang
;
Xie, Ping
;
Wu, Linqian
;
Huo, Jingqun
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收藏
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浏览/下载:5/0
  |  
提交时间:2024/09/19
Hydrologic frequency analysis
Non-stationary characteristics
Flood
Norming constants method
Higher-order probability weighted moments
The Magnetic Field Effects on The Oxygenation Rate of Recombinant Hemoglobin
期刊论文
OAI收割
PROGRESS IN BIOCHEMISTRY AND BIOPHYSICS, 2024, 卷号: 51
作者:
Liu, Yan
;
Fang, Yan-Wen
;
Zhang, Xin
;
Xie, Can
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收藏
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浏览/下载:5/0
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提交时间:2024/11/20
hemoglobin
magnetic field
human hemoglobin
yak hemoglobin
oxygenation rate
Structure-Based Drug Design of 2-Amino-[1,1′-biphenyl]-3-carboxamide Derivatives as Selective PKMYT1 Inhibitors for the Treatment of
CCNE1
-Amplified Breast Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 21
作者:
Wang, Chaofan
;
Fang, Yan
;
Zhou, Ziqin
;
Liu, Zhuoheng
;
Feng, Fang
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收藏
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浏览/下载:10/0
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提交时间:2024/09/26
LncRNA-
Snhg3
regulates mouse hepatic glycogenesis under normal chow diet
期刊论文
OAI收割
FASEB JOURNAL, 2024, 卷号: 38, 期号: 15, 页码: 15
作者:
Xie, Xianghong
;
Gao, Mingyue
;
Wang, Heping
;
Zhang, Minglong
;
Zhao, Wei
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收藏
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浏览/下载:13/0
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提交时间:2024/09/26
chromatin remodeling
glycogenesis
insulin resistance
lncRNA-Snhg3
Branched-chain amino acid transaminase 1 confers EGFR-TKI resistance through epigenetic glycolytic activation
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2024, 卷号: 9, 期号: 1, 页码: 17
作者:
Zhang, Tao
;
Pan, Zilu
;
Gao, Jing
;
Wu, Qingqing
;
Bai, Gang
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收藏
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浏览/下载:16/0
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提交时间:2024/10/21
Discovery of a novel BTK inhibitor S-016 and identification of a new strategy for the treatment of lymphomas including BTK inhibitor-resistant lymphomas
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2024, 页码: 11
作者:
Song, Pei-ran
;
Wan, Zhi-peng
;
Huang, Ge-ge
;
Song, Zi-lan
;
Zhang, Tao
  |  
收藏
  |  
浏览/下载:66/0
  |  
提交时间:2024/07/12
diffuse large B-cell lymphoma
BTK inhibitors
drug resistance
BTK C481F
BTK A428D
SYHA1813
SRY-Box transcription factor 9 triggers YAP nuclear entry via direct interaction in tumors
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2024, 卷号: 9, 期号: 1, 页码: 13
作者:
Qian, Hui
;
Ding, Chen-Hong
;
Liu, Fang
;
Chen, Shi-Jie
;
Huang, Chen-Kai
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收藏
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浏览/下载:18/0
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提交时间:2024/05/22