中国科学院机构知识库网格
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期刊论文 [79]
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A patent review of KDM4 histone demethylase inhibitors (2014-present)
期刊论文
OAI收割
EXPERT OPINION ON THERAPEUTIC PATENTS, 2026, 页码: 17
作者:
Yang, Xiaolong
;
Han, Yuyan
;
Yu, Lei
;
Xu, Shilin
  |  
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Redox-driven ADAR1 activation promotes Okazaki fragment maturation and DNA replication integrity
期刊论文
OAI收割
NATURE STRUCTURAL & MOLECULAR BIOLOGY, 2026, 页码: 35
作者:
Chen, Bin
;
Sun, Guangchao
;
Kloeber, Jake A.
;
Xiao, Huaping
;
Ouyang, Yaobin
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Furo[2,3-
f
]quinazolin-7(6
H
)-one Derivatives as Potent, Selective, and Orally Bioavailable MAT2A Inhibitors for MTAP-Deficient Cancer Therapy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 22, 页码: 24213-24231
作者:
Shi, Zihan
;
Lin, Kexin
;
Lin, Lijie
;
Chen, Zhiyi
;
Xie, Zhiyin
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  |  
Proteome-Wide Ligand and Target Discovery by Using Covalent Probes and Natural Products
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 19, 页码: 20228-20242
作者:
Liu, Jingqing
;
Huang, Chaoming
;
Li, Shengrong
;
Peng, Lijie
;
Sun, Yaoliang
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Design, synthesis and structure-activity relationship studies of novel macrocyclic 2,4-diaminopyrimidines as HPK1 inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2025, 卷号: 128, 页码: 12
作者:
Wu, Feifei
;
Sun, Jiaqi
;
Xu, Mingyang
;
Li, Huiyu
;
Wei, Jiarui
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Recent advances in small molecules targeting the METTL3
期刊论文
OAI收割
FUTURE MEDICINAL CHEMISTRY, 2025, 卷号: 17, 期号: 15, 页码: 1933-1944
作者:
Wu, Feifei
;
Yu, Lei
;
Xu, Shilin
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Design, Synthesis, and biological evaluation of 7H-Pyrrolo[2,3-d] pyrimidines as potent HPK1 kinase inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2025, 卷号: 119, 页码: 13
作者:
Wu, Feifei
;
Li, Huiyu
;
Li, Weiqiang
;
Zhang, Laishun
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Targeting QPCTL: An Emerging Therapeutic Opportunity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 2, 页码: 929-943
作者:
Yu, Lei
;
Sun, Yaoliang
;
Xie, Longyan
;
Tan, Xiao
;
Wang, Ping
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Discovery of an Efficacious RET PROTAC Degrader with Enhanced Antiproliferative Activity against Resistant Cancer Cells Harboring RET Solvent-Front Mutations
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 68, 期号: 1, 页码: 753-775
作者:
Zhang, Qian
;
He, Yingqi
;
Rao, Danni
;
He, Rui
;
Yu, Lei
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Population genomic analysis reveals a polygenic sex determination system in
Apostichopus japonicus
期刊论文
OAI收割
ISCIENCE, 2024, 卷号: 27, 期号: 10, 页码: 16
作者:
Jiang, Chunxi
;
Liu, Shilin
;
Yang, Yujia
;
Cui, Wei
;
Xu, Shuai
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