中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共79条,第1-10条 帮助

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A patent review of KDM4 histone demethylase inhibitors (2014-present) 期刊论文  OAI收割
EXPERT OPINION ON THERAPEUTIC PATENTS, 2026, 页码: 17
作者:  
Yang, Xiaolong;  Han, Yuyan;  Yu, Lei;  Xu, Shilin
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Redox-driven ADAR1 activation promotes Okazaki fragment maturation and DNA replication integrity 期刊论文  OAI收割
NATURE STRUCTURAL & MOLECULAR BIOLOGY, 2026, 页码: 35
作者:  
Chen, Bin;  Sun, Guangchao;  Kloeber, Jake A.;  Xiao, Huaping;  Ouyang, Yaobin
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Furo[2,3-f]quinazolin-7(6H)-one Derivatives as Potent, Selective, and Orally Bioavailable MAT2A Inhibitors for MTAP-Deficient Cancer Therapy 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 22, 页码: 24213-24231
作者:  
Shi, Zihan;  Lin, Kexin;  Lin, Lijie;  Chen, Zhiyi;  Xie, Zhiyin
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Proteome-Wide Ligand and Target Discovery by Using Covalent Probes and Natural Products 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 19, 页码: 20228-20242
作者:  
Liu, Jingqing
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Design, synthesis and structure-activity relationship studies of novel macrocyclic 2,4-diaminopyrimidines as HPK1 inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2025, 卷号: 128, 页码: 12
作者:  
Wu, Feifei;  Sun, Jiaqi;  Xu, Mingyang;  Li, Huiyu;  Wei, Jiarui
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Recent advances in small molecules targeting the METTL3 期刊论文  OAI收割
FUTURE MEDICINAL CHEMISTRY, 2025, 卷号: 17, 期号: 15, 页码: 1933-1944
作者:  
Wu, Feifei;  Yu, Lei;  Xu, Shilin
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Design, Synthesis, and biological evaluation of 7H-Pyrrolo[2,3-d] pyrimidines as potent HPK1 kinase inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2025, 卷号: 119, 页码: 13
作者:  
Wu, Feifei;  Li, Huiyu;  Li, Weiqiang;  Zhang, Laishun;  An, Qi
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Targeting QPCTL: An Emerging Therapeutic Opportunity 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 2, 页码: 929-943
作者:  
Yu, Lei;  Sun, Yaoliang;  Xie, Longyan;  Tan, Xiao;  Wang, Ping
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Discovery of an Efficacious RET PROTAC Degrader with Enhanced Antiproliferative Activity against Resistant Cancer Cells Harboring RET Solvent-Front Mutations 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 68, 期号: 1, 页码: 753-775
作者:  
Zhang, Qian;  He, Yingqi;  Rao, Danni;  He, Rui;  Yu, Lei
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Population genomic analysis reveals a polygenic sex determination system in Apostichopus japonicus 期刊论文  OAI收割
ISCIENCE, 2024, 卷号: 27, 期号: 10, 页码: 16
作者:  
Jiang, Chunxi;  Liu, Shilin;  Yang, Yujia;  Cui, Wei;  Xu, Shuai
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