中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共27条,第1-10条 帮助

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Construction of PROTAC Library via Liquid-Phase Synthesis Enabled by a Hydrophobic Tag 期刊论文  OAI收割
ORGANIC LETTERS, 2026, 卷号: 28, 期号: 8, 页码: 2747-2752
作者:  
Zhou, Yifeng;  He, Wei;  Zhou, Zehui;  Wu, Min;  Wu, Qianping
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Targeting Cbl-b by a small molecular inhibitor potentiates T cell receptor signaling and suggests rational combination strategies 期刊论文  OAI收割
INTERNATIONAL IMMUNOPHARMACOLOGY, 2026, 卷号: 169, 页码: 15
作者:  
Li, Yuantong;  Tang, Haotian;  Shi, Wenhao;  Zhou, Yu;  Wen, Jiaxin
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An overview of PROTACs targeting KRAS and SOS1 as antitumor agents 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 125, 页码: 13
作者:  
Han, Zhiqiu;  Wu, Qianping;  Rao, Hongxin;  Xu, Tianfeng;  Zhou, Chuan
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An updated patent review of SOS1 inhibitors (2022-present) 期刊论文  OAI收割
EXPERT OPINION ON THERAPEUTIC PATENTS, 2024, 页码: 15
作者:  
Zhou, Guizhen;  Zhou, Chuan;  Ma, Xinyi;  Xu, Jiahang;  Zhou, Zehui
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Design, Synthesis, and Biological Evaluation of 2,4-Diaminopyrimidine Derivatives as Potent CDK7 Inhibitors 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2024, 页码: 8
作者:  
Zhang, Hualin;  Tu, Yutong;  Tao, Zhaofan;  Gao, Lixin;  Huang, Shengjie
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Design, synthesis, and bioevaluation of SOS1 PROTACs derived from pyrido [2,3- d ]pyrimidin-7-one-based SOS1 inhibitor 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 107, 页码: 9
作者:  
Wang, Kun;  Zhou, Zehui;  Ma, Xinyi;  Xu, Jiahang
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Design, Synthesis, and Bioevaluation of Transcriptional Enhanced Assocciated Domain (TEAD) PROTAC Degraders 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 15, 期号: 5, 页码: 631-639
作者:  
Li, Huajie;  Ge, Zhiming;  Lin, Kexin;  He, Wei;  Chu, Qinyu
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Design, Synthesis, and Biological Evaluation of Potent and Selective PROTAC Degraders of Oncogenic KRASG12D 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1147-1167
作者:  
Zhou, Chuan;  Fan, Zisheng;  Gu, Yuejiao;  Ge, Zhiming;  Tao, Zhaofan
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Discovery of ARD-1676 as a Highly Potent and Orally Efficacious AR PROTAC Degrader with a Broad Activity against AR Mutants for the Treatment of AR plus Human Prostate Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 18, 页码: 13280-13303
作者:  
Xiang, Weiguo;  Zhao, Lijie;  Han, Xin;  Xu, Tianfeng;  Kregel, Steven
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Stimuli-activatable PROTACs for precise protein degradation and cancer therapy 期刊论文  OAI收割
SCIENCE BULLETIN, 2023, 卷号: 68, 期号: 10, 页码: 1069-1085
作者:  
Gao, Jing;  Yang, Lei;  Lei, Shumin;  Zhou, Feng;  Nie, Huijun
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