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From Hit to Lead: Discovery of Novel Selective RIPK1 Inhibitor with Pyridoimidazole Scaffold for the Treatment of Autoimmune Diseases through Phenotypic Screening and Structural Optimization
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2026, 卷号: 69, 期号: 3, 页码: 3252-3288
作者:
Wan, Jihong
;
Xiong, Xiao-Yu
;
Geng, Zixiang
;
Yuan, Benjun
;
Ma, Youzhen
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Targeting intrinsic and CAF-mediated signaling by PI3Kα inhibitor CYH33 attenuated metastasis in lung squamous cell carcinoma
期刊论文
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ACTA PHARMACOLOGICA SINICA, 2026, 页码: 14
作者:
Ma, Xiao-yu
;
Deng, Jie-ting
;
Cao, Zhe-rui
;
Xu, Lan
;
Ding, Jian
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BMAL1/PGC1a4-FNDC5/irisin axis impacts distinct outcomes of time-of-day resistance exercise
期刊论文
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JOURNAL OF SPORT AND HEALTH SCIENCE, 2025, 卷号: 14, 页码: 23
作者:
Guo, Mingwei
;
Shen, Fei
;
Guo, Xiaozhen
;
Zhang, Jun
;
Ma, Ying
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A pan-KRAS inhibitor and its derived degrader elicit multifaceted anti-tumor efficacy in
KRAS
-driven cancers
期刊论文
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CANCER CELL, 2025, 卷号: 43, 期号: 10, 页码: 32
作者:
Feng, Juanjuan
;
Xiao, Xuanzheng
;
Xia, Xinting
;
Min, Jian
;
Tang, Weiying
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Spectral Hardening Reveals Afterglow Emergence in Long-duration Fast X-Ray Transients: A Case Study of GRB 250404A/EP250404a
期刊论文
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ASTROPHYSICAL JOURNAL LETTERS, 2025, 卷号: 989, 期号: 2, 页码: L39
作者:
Yin, Yi-Han Iris
;
Fang, Yuan
;
Zhang, Bin-Bin
;
Deng, Chen
;
Yang, Jun
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Benzothiazole amide analogues as antagonists of TRPC 6 channels: A therapeutic approach for kidney fibrosis
期刊论文
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EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 291, 页码: 16
作者:
Ren, Chunlin
;
Xu, Qiding
;
Luo, Qiusi
;
Qiao, Xue
;
Ding, Taotao
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Extensive Early Cretaceous arc-like magmatic rocks in central Tibet manifest subduction rollback of the Neo-Tethyan ocean
期刊论文
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GEOLOGICAL SOCIETY OF AMERICA BULLETIN, 2025, 页码: 16
作者:
Wen, Ding-Jun
;
Hu, Xiumian
;
Klemd, Reiner
;
Wang, Xiao-Lei
;
Ge, Rongfeng
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REG3A secreted by peritumoral acinar cells enhances pancreatic ductal adenocarcinoma progression via activation of EGFR signaling
期刊论文
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CELL COMMUNICATION AND SIGNALING, 2025, 卷号: 23, 期号: 1, 页码: 19
作者:
Ren, Xiaojing
;
Teng, Yunfei
;
Xie, Kunxin
;
He, Xiao
;
Chen, Gang
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Acoustic emission and microfracture analysis of strain rockbursts in deep granite under varying intermediate principal stresses
期刊论文
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MEASUREMENT, 2025, 卷号: 242, 页码: 16
作者:
Guo, Guang-tao
;
Xu, Ding-Ping
;
Wu, Xiao-gang
;
Zhu, Jun-xing
;
Xu, Huai-sheng
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GRB 240529A: A Tale of Two Shocks
期刊论文
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ASTROPHYSICAL JOURNAL LETTERS, 2024, 卷号: 976, 期号: 2
作者:
Sun, Tian-Rui
;
Geng, Jin-Jun
;
Yan, Jing-Zhi
;
Hu, You-Dong
;
Wu, Xue-Feng
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