中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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金属研究所 [18]
上海药物研究所 [10]
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期刊论文 [57]
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Development of Orally Bioavailable Octahydroindole-Based Peptidomimetic Derivative as a Broad-Spectrum Inhibitor against HCoV-OC43 and SARS-CoV-2
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 11, 页码: 10823-10844
作者:
Hu, Shulei
;
Zhang, Yumin
;
Wang, Chenchen
;
Li, Jian
;
Su, Haixia
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收藏
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浏览/下载:19/0
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提交时间:2025/07/25
Substrate recognition and cleavage mechanism of the monkeypox virus core protease
期刊论文
OAI收割
NATURE, 2025, 页码: 29
作者:
Gao, Yan
;
Xie, Xiong
;
Zhang, Xiaoyu
;
Cao, Junyuan
;
Lan, Weiqi
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收藏
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浏览/下载:5/0
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提交时间:2025/08/20
Design, Synthesis, and Biological Evaluation of Peptidomimetic Tetrahydropyrrole Spirodihydroindolones as SARS-CoV-2 3CL Protease Inhibitors
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 16, 期号: 5, 页码: 790-796
作者:
Hu, Liuyan
;
Zhao, Zhi
;
Zhang, Shujing
;
Yang, Lei
;
Cui, Wenjie
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2025/06/23
COVID-19
SARS-CoV-2
3CL protease
Peptidomimetic inhibitors
Tetrahydropyrrole spirodihydroindolone
Discovery of Novel Nonpeptidic and Noncovalent Small Molecule 3CL
pro
Inhibitors as anti-SARS-CoV-2 Drug Candidate
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 15, 页码: 12760-12783
作者:
Jiang, Zhidong
;
Feng, Bo
;
Chen, Lu
;
Nie, Tianqing
;
Chen, Shizhao
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收藏
  |  
浏览/下载:43/0
  |  
提交时间:2024/09/26
Discovery and characterization of novel potent non-covalent small molecule inhibitors targeting papain-like protease from SARS-CoV-2
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2024, 卷号: 14, 期号: 7, 页码: 3286-3290
作者:
Zheng, Miao
;
Feng, Bo
;
Zhang, Yumin
;
Liu, Xin
;
Zhao, Na
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收藏
  |  
浏览/下载:30/0
  |  
提交时间:2024/08/22
Non-covalent PLpro inhibitors
Antiviral activity
Structural-based drug design
Imidazo[4,5-b]pyridine scaffold
New measurements reveal a large contribution of nitrogenous molecules to ambient organic aerosol
期刊论文
OAI收割
NPJ CLIMATE AND ATMOSPHERIC SCIENCE, 2024, 卷号: 7, 期号: 1, 页码: 9
作者:
Yu, Xu
;
Li, Qianfeng
;
Liao, Kezheng
;
Li, Yumin
;
Wang, Xinming
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收藏
  |  
浏览/下载:33/0
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提交时间:2024/09/12
eIF2α-mediated integrated stress response links multiple intracellular signaling pathways to reprogram vascular smooth muscle cell fate in carotid artery plaque
期刊论文
OAI收割
HELIYON, 2024, 卷号: 10, 期号: 5, 页码: 14
作者:
Luo, Jichang
;
Zhang, Xiao
;
Li, Wenjing
;
Wang, Tao
;
Cui, Shengyan
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收藏
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浏览/下载:50/0
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提交时间:2024/07/03
Carotid artery atherosclerosis
Primary vascular smooth muscle cells
Organelles
Plaque vulnerability
Translation initiation factor 2 alpha
Structure-based design of pan-coronavirus inhibitors targeting host cathepsin L and calpain-1
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2024, 卷号: 9, 期号: 1, 页码: 14
作者:
Xie, Xiong
;
Lan, Qiaoshuai
;
Zhao, Jinyi
;
Zhang, Sulin
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收藏
  |  
浏览/下载:39/0
  |  
提交时间:2024/05/07
Design, synthesis and biological evaluation of peptidomimetic benzothiazolyl ketones as 3CLpro inhibitors against SARS-CoV-2
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 257, 页码: 13
作者:
Yang, Hanxi
;
You, Mengyuan
;
Shu, Xiaoyang
;
Zhen, Jingyao
;
Zhu, Mengwei
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2023/10/17
Peptidomimetics
Benzothiazolyl ketone
3CLpro inhibitor
Pharmacokinetic properties
SARS-CoV-2
Estimation of China Fusion Engineering Test Reactor performance and burning fraction in different pellet fueling scenarios by a multi-species radial transport model
期刊论文
OAI收割
Plasma Science and Technology, 2022, 卷号: 24
作者:
LIN,Weisheng
;
WANG,Xiaogang
;
XU,Xueqiao
;
KONG,Defeng
;
WANG,Yumin
  |  
收藏
  |  
浏览/下载:57/0
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提交时间:2022/12/22
CFETR
tritium burning fraction
fueling scenarios