中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共205条,第1-10条 帮助

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Development of 3-arylaminothiophenic-2-carboxylic acid derivatives as new FTO inhibitors showing potent antileukemia activities 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 289, 页码: 17
作者:  
Zhang, Deyan;  Liu, Lu;  Li, Ming;  Hu, Xinyi;  Zhang, Xi
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/04/24
Modular Synthesis of the Potent Antibiotic Amycolamicin and Diastereomeric Analogues Thereof 期刊论文  OAI收割
ORGANIC LETTERS, 2025, 卷号: 27, 期号: 14, 页码: 3631-3636
作者:  
Yin, Xuejian;  Zhang, Zhengxuan;  Yuan, Ziqi;  Zhu, Qiuyu;  Xu, Peng
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/05/27
A patenting perspective of fat mass and obesity associated protein (FTO) inhibitors: 2017-present 期刊论文  OAI收割
EXPERT OPINION ON THERAPEUTIC PATENTS, 2025, 页码: 10
作者:  
Dong, Ze;  Huang, Yue;  Xia, Wenyang;  Liao, Yonggang;  Yang, Cai-Guang
  |  收藏  |  浏览/下载:1/0  |  提交时间:2025/05/27
Discovery of Covalent and Cell-Active ALKBH5 Inhibitors with Potent Antileukemia Effects In Vivo 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 9
作者:  
Wu, Hengbo;  Lai, Gan-Qiang;  Cheng, Ruixiang;  Huang, Hui;  Wang, Ju
  |  收藏  |  浏览/下载:1/0  |  提交时间:2025/04/24
Terrestrial ecosystem response to Early Cretaceous global environmental change: A calibrated, high-resolution Aptian record from Northeast China 期刊论文  OAI收割
EARTH AND PLANETARY SCIENCE LETTERS, 2025, 卷号: 653, 页码: 13
作者:  
Sun, Ming-Dao;  Lin, Qin;  Ramezani, Jahandar;  Liu, Jiang-Si;  Lu, Zheng-An
  |  收藏  |  浏览/下载:22/0  |  提交时间:2025/04/03
Discovery of Novel RNA Demethylase FTO Inhibitors Featuring an Acylhydrazone Scaffold with Potent Antileukemia Activity 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 22
作者:  
Liang, Xuewu;  Huang, Yue;  Ren, Hairu;  Liu, Qi;  Chen, Liang
  |  收藏  |  浏览/下载:12/0  |  提交时间:2025/04/01
Structure-Guided Development of ClpP Agonists with Potent Therapeutic Activities against Staphylococcus aureus Infection 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 2, 页码: 1810-1823
作者:  
Zhang, Tao;  Wu, Wei;  Zhao, Yanling;  Ding, Ziang;  Wei, Bingyan
  |  收藏  |  浏览/下载:11/0  |  提交时间:2025/04/01
Structure-guided development of selective caseinolytic protease P agonists as antistaphylococcal agents 期刊论文  OAI收割
CELL REPORTS MEDICINE, 2024, 卷号: 5, 期号: 12, 页码: 20
作者:  
Zhang, Tao;  Wang, Pengyu;  Zhou, Hailing;  Wei, Bingyan;  Zhao, Yanling
  |  收藏  |  浏览/下载:18/0  |  提交时间:2025/04/01
Integrative study of lung cancer adeno-to-squamous transition in EGFR TKI resistance identifies RAPGEF3 as a therapeutic target 期刊论文  OAI收割
NATIONAL SCIENCE REVIEW, 2024, 卷号: 11, 期号: 12, 页码: 20
作者:  
Wang, Hua;  Tang, Shijie;  Wu, Qibiao;  He, Yayi;  Zhu, Weikang
  |  收藏  |  浏览/下载:19/0  |  提交时间:2025/02/28
Discovery of a potent PROTAC degrader for RNA demethylase FTO as antileukemic therapy 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2024, 卷号: 14, 期号: 12, 页码: 5382-5392
作者:  
Liu, Lu;  Qiu, Yuanlai;  Suo, Yuying;  Tong, Siyao;  Wang, Yiqing
  |  收藏  |  浏览/下载:12/0  |  提交时间:2025/04/01