中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [57]
地理科学与资源研究所 [1]
遥感与数字地球研究所 [1]
昆明植物研究所 [1]
合肥物质科学研究院 [1]
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OAI收割 [61]
内容类型
期刊论文 [61]
发表日期
2024 [3]
2023 [7]
2022 [3]
2021 [5]
2020 [7]
2019 [3]
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The Association Between Environmental Factors and Longevity in Hezhou, China Based on the Drinking Water Quality
期刊论文
OAI收割
EXPOSURE AND HEALTH, 2024, 卷号: N/A
作者:
Deng, Qucheng
;
Liu, Yaqing
;
Zhu, Kaixian
;
Han, Xuerong
;
Erpeng, Yang
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2025/01/17
Healthy aging
Centenarian
Drinking water
Trace elements indicators
Longevity city
Chemoproteomics of Marine Natural Product Naamidine J Unveils CSE1L as a Therapeutic Target in Acute Lung Injury
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2024, 页码: 14
作者:
Gao, Cheng-Long
;
Song, Jin-Qian
;
Yang, Ze-Nan
;
Wang, Haojie
;
Wu, Xin-Yuan
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/11/05
Dual-site molecular glues for enhancing protein-protein interactions of the CDK12-DDB1 complex
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2024, 卷号: 15, 期号: 1, 页码: 13
作者:
Zhang, Zemin
;
Li, Yuanqing
;
Yang, Jie
;
Li, Jiacheng
;
Lin, Xiongqiang
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2024/09/26
Naringenin improves muscle endurance via activation of the Sp1-ERRg transcriptional axis
期刊论文
OAI收割
CELL REPORTS, 2023, 卷号: 42, 期号: 11, 页码: 25
作者:
Lv, Zhenyu
;
Meng, Jiao
;
Yao, Sheng
;
Xiao, Fu
;
Li, Shilong
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/12/11
OTTM: an automated classification tool for translational drug discovery from omics data
期刊论文
OAI收割
BRIEFINGS IN BIOINFORMATICS, 2023, 页码: 12
作者:
Yang, Xiaobo
;
Zhang, Bei
;
Wang, Siqi
;
Lu, Ye
;
Chen, Kaixian
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2023/10/17
OTTM
omics data
translational drug discovery
literature mining
hepatocellular carcinoma
Design, synthesis and biological evaluation of salicylanilides as novel allosteric inhibitors of human pancreatic lipase
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 91, 页码: 11
作者:
Zhao, Yitian
;
Zhang, Min
;
Hou, Xudong
;
Han, Jiaxin
;
Qin, Xiaoya
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2023/10/17
Salicylanilide
hPL inhibitor
Structure -activity relationship
Anti -obesity
Discovery of a Novel Bifunctional Steroid Analog, YXG-158, as an Androgen Receptor Degrader and CYP17A1 Inhibitor for the Treatment of Enzalutamide-Resistant Prostate Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 14, 页码: 9972-9991
作者:
Wang, Ao
;
Luo, Xianggang
;
Meng, Xin
;
Lu, Zhengyu
;
Chen, Kaixian
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/10/17
Structural Mass Spectrometry Probes the Inhibitor-Induced Allosteric Activation of CDK12/CDK13-Cyclin K Dissociation
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2023, 卷号: 145, 期号: 21, 页码: 11477-11481
作者:
Bai, Yu
;
Liu, Zheyi
;
Li, Yuanqing
;
Zhao, Heng
;
Lai, Can
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2023/10/17
Design, Synthesis, and Biological Evaluation of Bipyridazine Derivatives as Stimulator of Interferon Genes (STING) Receptor Agonists
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 5, 页码: 3327-3347
作者:
Shan, Bin
;
Hou, Hui
;
Zhang, Keke
;
Li, Rui
;
Shen, Chang
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2024/03/27
Cyclization strategy leads to highly potent Bromodomain and extra-terminal (BET) Bromodomain inhibitors for the treatment of acute liver injury
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 247, 页码: 13
作者:
Chen, Chao
;
Lu, Tian
;
Chen, Panyu
;
Li, Zizhou
;
Yang, Yaxi
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2023/04/10
BET Bromodomains
Acute liver injury
Anti-inflammatory activity
Inhibitors
Tetracyclic compounds