中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
化学研究所 [10]
上海药物研究所 [9]
西北高原生物研究所 [9]
地质与地球物理研究所 [2]
武汉病毒研究所 [2]
中国科学院大学 [2]
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期刊论文 [39]
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2024 [2]
2023 [1]
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2020 [2]
2019 [2]
2017 [10]
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Marine & F... [1]
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Discovery of CZL-046 with an (
S
)-3-Fluoropyrrolidin-2-one Scaffold as a p300 Bromodomain Inhibitor for the Treatment of Multiple Myeloma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 20, 页码: 18606-18628
作者:
Chen, Zonglong
;
Yang, Hong
;
Zhang, Yan
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/11/05
Development of ketalized unsaturated saccharides as multifunctional cysteine-targeting covalent warheads
期刊论文
OAI收割
COMMUNICATIONS CHEMISTRY, 2024, 卷号: 7, 期号: 1, 页码: 10
作者:
Dong, Sanfeng
;
Huang, Hui
;
Li, Jintian
;
Li, Xiaomei
;
Bunu, Samuel Jacob
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/10/21
The first record of Lower Cretaceous theropod tracks in Turpan-Hami Basin, Xinjiang, northwestern China
期刊论文
OAI收割
HISTORICAL BIOLOGY, 2023, 页码: 6
作者:
Li, Yang
;
Jiang, Shunxing
;
Yan, Feng
;
Ma, Yingxia
;
Wang, Xiaolin
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2023/11/02
Theropod tracks
Lower Cretaceous
Hami pterosaur fauna
Turpan-Hami Basin
Xinjiang
Discovery of novel benzimidazole derivatives as potent p300 bromodomain inhibitors with anti-proliferative activity in multiple cancer cells
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2022, 卷号: 66, 页码: 16
作者:
Chen, Zonglong
;
Li, Jiayi
;
Yang, Hong
;
He, Yulong
;
Shi, Qiongyu
  |  
收藏
  |  
浏览/下载:53/0
  |  
提交时间:2022/08/16
P300
Bromodomain inhibitors
CBP30
SBDD
Design, synthesis and biological evaluation of (R)-5-methylpyrrolidin-2-ones as p300 bromodomain inhibitors with Anti-Tumor activities in multiple tumor lines
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 124, 页码: 15
作者:
Liu, Ruiqi
;
Yang, Hong
;
Chen, Zonglong
;
Zhou, Kaixin
;
Shi, Qiongyu
  |  
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2022/08/16
Epigenetics
p300
CBP
Bromodomain inhibitors
CCS1477
A novel virtual screening procedure identifies Pralatrexate as inhibitor of SARS-CoV-2 RdRp and it reduces viral replication in vitro
期刊论文
OAI收割
PLOS COMPUTATIONAL BIOLOGY, 2020, 卷号: 16, 期号: 12, 页码: 20
作者:
Zhang, Haiping
;
Yang, Yang
;
Li, Junxin
;
Wang, Min
;
Saravanan, Konda Mani
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2021/12/01
Investigation of the remote acyl group participation in glycosylation from conformational perspectives by using trichloroacetimidate as the acetyl surrogate
期刊论文
OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2020, 卷号: 7, 期号: 13, 页码: 1606-1615
作者:
Xu, Ke
;
Man, Qingmin
;
Zhang, Yang
;
Guo, Jia
;
Liu, Yichu
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2020/12/24
Design, synthesis, and biological evaluation of a new class of histone acetyltransferase p300 inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 180, 页码: 171-190
作者:
Liu, Ruiqi
;
Zhang, Zhuqing
;
Yang, Hong
;
Zhou, Kaixin
;
Geng, Meiyu
  |  
收藏
  |  
浏览/下载:63/0
  |  
提交时间:2020/07/01
p300 inhibitors
Epigenetics
Structure-activity relationship
Sensitive tumor cell proliferation
C646
Scheelite geochemistry in porphyry-skarn W-Mo systems: A case study from the Gaojiabang Deposit, East China
期刊论文
OAI收割
ORE GEOLOGY REVIEWS, 2019, 卷号: 113, 页码: 17
作者:
Song, Guoxue
;
Cook, Nigel J.
;
Li, Guangming
;
Qin, Kezhang
;
Ciobanu, Cristiana L.
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2020/05/18
Scheelite
Substitution mechanism
Redox state
Sr-isotopes
Porphyry-skarn system
Gaojiabang deposit
CASCIRE surveillance network and work on avian influenza viruses
期刊论文
OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2017
Bi, Yuhai
;
Shi, Weifeng
;
Chen, Jianjun
;
Chen, Quanjiao
;
Ma, Zhenghai
;
Wong, Gary
;
Tian, Wenxia
;
Yin, Renfu
;
Fu, Guanghua
;
Yang, Yongchun
;
Liu, William J.
;
Quan, Chuansong
;
Wang, Qianli
;
He, Shenghu
;
Li, Xiangdong
;
Xia, Qianfeng
;
Wang, Lixin
;
Pan, Zhaohui
;
Li, Laixing
;
Li, Hong
;
Xu, Wen
;
Luo, Ying
;
Zeng, Hui
;
Dai, Lianpan
;
Xiao, Haixia
;
Sharshov, Kirill
;
Shestopalov, Alexander
;
Shi, Yi
;
Yan, Jinghua
;
Li, Xuebing
;
Liu, Yingxia
;
Lei, Fumin
;
Liu, Wenjun
;
Gao, George F.
  |  
收藏
  |  
浏览/下载:96/0
  |  
提交时间:2019/06/14