中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共40条,第1-10条 帮助

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Discovery of Novel Class of METTL3 Inhibitors with a Pyridin-2(1H)-one Moiety 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 16, 期号: 11, 页码: 2257-2263
作者:  
Zhang, Weihang;  Huang, Yuting;  Yang, Hong;  Wan, Haiyan;  Lei, Xinsheng
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Discovery of CZL-046 with an (S)-3-Fluoropyrrolidin-2-one Scaffold as a p300 Bromodomain Inhibitor for the Treatment of Multiple Myeloma 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 20, 页码: 18606-18628
作者:  
Chen, Zonglong;  Yang, Hong;  Zhang, Yan;  Lyu, Xiaodong;  Shi, Qiongyu
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Development of ketalized unsaturated saccharides as multifunctional cysteine-targeting covalent warheads 期刊论文  OAI收割
COMMUNICATIONS CHEMISTRY, 2024, 卷号: 7, 期号: 1, 页码: 10
作者:  
Dong, Sanfeng;  Huang, Hui;  Li, Jintian;  Li, Xiaomei;  Bunu, Samuel Jacob
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The first record of Lower Cretaceous theropod tracks in Turpan-Hami Basin, Xinjiang, northwestern China 期刊论文  OAI收割
HISTORICAL BIOLOGY, 2023, 页码: 6
作者:  
Li, Yang;  Jiang, Shunxing;  Yan, Feng;  Ma, Yingxia;  Wang, Xiaolin
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Discovery of novel benzimidazole derivatives as potent p300 bromodomain inhibitors with anti-proliferative activity in multiple cancer cells 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2022, 卷号: 66, 页码: 16
作者:  
Chen, Zonglong;  Li, Jiayi;  Yang, Hong;  He, Yulong;  Shi, Qiongyu
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Design, synthesis and biological evaluation of (R)-5-methylpyrrolidin-2-ones as p300 bromodomain inhibitors with Anti-Tumor activities in multiple tumor lines 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 124, 页码: 15
作者:  
Liu, Ruiqi;  Yang, Hong;  Chen, Zonglong;  Zhou, Kaixin;  Shi, Qiongyu
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A novel virtual screening procedure identifies Pralatrexate as inhibitor of SARS-CoV-2 RdRp and it reduces viral replication in vitro 期刊论文  OAI收割
PLOS COMPUTATIONAL BIOLOGY, 2020, 卷号: 16, 期号: 12, 页码: 20
作者:  
Zhang, Haiping;  Yang, Yang;  Li, Junxin;  Wang, Min;  Saravanan, Konda Mani
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Investigation of the remote acyl group participation in glycosylation from conformational perspectives by using trichloroacetimidate as the acetyl surrogate 期刊论文  OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2020, 卷号: 7, 期号: 13, 页码: 1606-1615
作者:  
Xu, Ke;  Man, Qingmin;  Zhang, Yang;  Guo, Jia;  Liu, Yichu
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Design, synthesis, and biological evaluation of a new class of histone acetyltransferase p300 inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 180, 页码: 171-190
作者:  
Liu, Ruiqi;  Zhang, Zhuqing;  Yang, Hong;  Zhou, Kaixin;  Geng, Meiyu
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Scheelite geochemistry in porphyry-skarn W-Mo systems: A case study from the Gaojiabang Deposit, East China 期刊论文  OAI收割
ORE GEOLOGY REVIEWS, 2019, 卷号: 113, 页码: 17
作者:  
Song, Guoxue;  Cook, Nigel J.;  Li, Guangming;  Qin, Kezhang;  Ciobanu, Cristiana L.
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