中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
化学研究所 [10]
上海药物研究所 [10]
西北高原生物研究所 [9]
地质与地球物理研究所 [2]
武汉病毒研究所 [2]
中国科学院大学 [2]
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期刊论文 [40]
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2025 [1]
2024 [2]
2023 [1]
2022 [2]
2020 [2]
2019 [2]
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Marine & F... [1]
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Discovery of Novel Class of METTL3 Inhibitors with a Pyridin-2(1
H
)-one Moiety
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 16, 期号: 11, 页码: 2257-2263
作者:
Zhang, Weihang
;
Huang, Yuting
;
Yang, Hong
;
Wan, Haiyan
;
Lei, Xinsheng
  |  
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  |  
Discovery of CZL-046 with an (
S
)-3-Fluoropyrrolidin-2-one Scaffold as a p300 Bromodomain Inhibitor for the Treatment of Multiple Myeloma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 20, 页码: 18606-18628
作者:
Chen, Zonglong
;
Yang, Hong
;
Zhang, Yan
;
Lyu, Xiaodong
;
Shi, Qiongyu
  |  
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  |  
Development of ketalized unsaturated saccharides as multifunctional cysteine-targeting covalent warheads
期刊论文
OAI收割
COMMUNICATIONS CHEMISTRY, 2024, 卷号: 7, 期号: 1, 页码: 10
作者:
Dong, Sanfeng
;
Huang, Hui
;
Li, Jintian
;
Li, Xiaomei
;
Bunu, Samuel Jacob
  |  
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  |  
The first record of Lower Cretaceous theropod tracks in Turpan-Hami Basin, Xinjiang, northwestern China
期刊论文
OAI收割
HISTORICAL BIOLOGY, 2023, 页码: 6
作者:
Li, Yang
;
Jiang, Shunxing
;
Yan, Feng
;
Ma, Yingxia
;
Wang, Xiaolin
  |  
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  |  
Discovery of novel benzimidazole derivatives as potent p300 bromodomain inhibitors with anti-proliferative activity in multiple cancer cells
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2022, 卷号: 66, 页码: 16
作者:
Chen, Zonglong
;
Li, Jiayi
;
Yang, Hong
;
He, Yulong
;
Shi, Qiongyu
  |  
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  |  
Design, synthesis and biological evaluation of (R)-5-methylpyrrolidin-2-ones as p300 bromodomain inhibitors with Anti-Tumor activities in multiple tumor lines
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 124, 页码: 15
作者:
Liu, Ruiqi
;
Yang, Hong
;
Chen, Zonglong
;
Zhou, Kaixin
;
Shi, Qiongyu
  |  
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  |  
A novel virtual screening procedure identifies Pralatrexate as inhibitor of SARS-CoV-2 RdRp and it reduces viral replication in vitro
期刊论文
OAI收割
PLOS COMPUTATIONAL BIOLOGY, 2020, 卷号: 16, 期号: 12, 页码: 20
作者:
Zhang, Haiping
;
Yang, Yang
;
Li, Junxin
;
Wang, Min
;
Saravanan, Konda Mani
  |  
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  |  
Investigation of the remote acyl group participation in glycosylation from conformational perspectives by using trichloroacetimidate as the acetyl surrogate
期刊论文
OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2020, 卷号: 7, 期号: 13, 页码: 1606-1615
作者:
Xu, Ke
;
Man, Qingmin
;
Zhang, Yang
;
Guo, Jia
;
Liu, Yichu
  |  
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  |  
Design, synthesis, and biological evaluation of a new class of histone acetyltransferase p300 inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 180, 页码: 171-190
作者:
Liu, Ruiqi
;
Zhang, Zhuqing
;
Yang, Hong
;
Zhou, Kaixin
;
Geng, Meiyu
  |  
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  |  
Scheelite geochemistry in porphyry-skarn W-Mo systems: A case study from the Gaojiabang Deposit, East China
期刊论文
OAI收割
ORE GEOLOGY REVIEWS, 2019, 卷号: 113, 页码: 17
作者:
Song, Guoxue
;
Cook, Nigel J.
;
Li, Guangming
;
Qin, Kezhang
;
Ciobanu, Cristiana L.
  |  
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