中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共39条,第1-10条 帮助

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Discovery of CZL-046 with an (S)-3-Fluoropyrrolidin-2-one Scaffold as a p300 Bromodomain Inhibitor for the Treatment of Multiple Myeloma 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 20, 页码: 18606-18628
作者:  
Chen, Zonglong;  Yang, Hong;  Zhang, Yan
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/11/05
Development of ketalized unsaturated saccharides as multifunctional cysteine-targeting covalent warheads 期刊论文  OAI收割
COMMUNICATIONS CHEMISTRY, 2024, 卷号: 7, 期号: 1, 页码: 10
作者:  
Dong, Sanfeng;  Huang, Hui;  Li, Jintian;  Li, Xiaomei;  Bunu, Samuel Jacob
  |  收藏  |  浏览/下载:12/0  |  提交时间:2024/10/21
The first record of Lower Cretaceous theropod tracks in Turpan-Hami Basin, Xinjiang, northwestern China 期刊论文  OAI收割
HISTORICAL BIOLOGY, 2023, 页码: 6
作者:  
Li, Yang;  Jiang, Shunxing;  Yan, Feng;  Ma, Yingxia;  Wang, Xiaolin
  |  收藏  |  浏览/下载:32/0  |  提交时间:2023/11/02
Discovery of novel benzimidazole derivatives as potent p300 bromodomain inhibitors with anti-proliferative activity in multiple cancer cells 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2022, 卷号: 66, 页码: 16
作者:  
Chen, Zonglong;  Li, Jiayi;  Yang, Hong;  He, Yulong;  Shi, Qiongyu
  |  收藏  |  浏览/下载:53/0  |  提交时间:2022/08/16
Design, synthesis and biological evaluation of (R)-5-methylpyrrolidin-2-ones as p300 bromodomain inhibitors with Anti-Tumor activities in multiple tumor lines 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 124, 页码: 15
作者:  
Liu, Ruiqi;  Yang, Hong;  Chen, Zonglong;  Zhou, Kaixin;  Shi, Qiongyu
  |  收藏  |  浏览/下载:55/0  |  提交时间:2022/08/16
A novel virtual screening procedure identifies Pralatrexate as inhibitor of SARS-CoV-2 RdRp and it reduces viral replication in vitro 期刊论文  OAI收割
PLOS COMPUTATIONAL BIOLOGY, 2020, 卷号: 16, 期号: 12, 页码: 20
作者:  
Zhang, Haiping;  Yang, Yang;  Li, Junxin;  Wang, Min;  Saravanan, Konda Mani
  |  收藏  |  浏览/下载:39/0  |  提交时间:2021/12/01
Investigation of the remote acyl group participation in glycosylation from conformational perspectives by using trichloroacetimidate as the acetyl surrogate 期刊论文  OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2020, 卷号: 7, 期号: 13, 页码: 1606-1615
作者:  
Xu, Ke;  Man, Qingmin;  Zhang, Yang;  Guo, Jia;  Liu, Yichu
  |  收藏  |  浏览/下载:23/0  |  提交时间:2020/12/24
Design, synthesis, and biological evaluation of a new class of histone acetyltransferase p300 inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 180, 页码: 171-190
作者:  
Liu, Ruiqi;  Zhang, Zhuqing;  Yang, Hong;  Zhou, Kaixin;  Geng, Meiyu
  |  收藏  |  浏览/下载:63/0  |  提交时间:2020/07/01
Scheelite geochemistry in porphyry-skarn W-Mo systems: A case study from the Gaojiabang Deposit, East China 期刊论文  OAI收割
ORE GEOLOGY REVIEWS, 2019, 卷号: 113, 页码: 17
作者:  
Song, Guoxue;  Cook, Nigel J.;  Li, Guangming;  Qin, Kezhang;  Ciobanu, Cristiana L.
  |  收藏  |  浏览/下载:28/0  |  提交时间:2020/05/18
CASCIRE surveillance network and work on avian influenza viruses 期刊论文  OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2017
Bi, Yuhai; Shi, Weifeng; Chen, Jianjun; Chen, Quanjiao; Ma, Zhenghai; Wong, Gary; Tian, Wenxia; Yin, Renfu; Fu, Guanghua; Yang, Yongchun; Liu, William J.; Quan, Chuansong; Wang, Qianli; He, Shenghu; Li, Xiangdong; Xia, Qianfeng; Wang, Lixin; Pan, Zhaohui; Li, Laixing; Li, Hong; Xu, Wen; Luo, Ying; Zeng, Hui; Dai, Lianpan; Xiao, Haixia; Sharshov, Kirill; Shestopalov, Alexander; Shi, Yi; Yan, Jinghua; Li, Xuebing; Liu, Yingxia; Lei, Fumin; Liu, Wenjun; Gao, George F.
  |  收藏  |  浏览/下载:96/0  |  提交时间:2019/06/14