中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共9条,第1-9条 帮助

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Discovery of a brain-permeable bromodomain and extra terminal domain (BET) inhibitor with selectivity for BD1 for the treatment of multiple sclerosis 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 14
作者:  
Chen, Xuetao;  Wu, Tingting;  Du, Zhiyan;  Kang, Wenjing;  Xu, Rujun
  |  收藏  |  浏览/下载:24/0  |  提交时间:2024/02/27
Discovery of 1H-Imidazo[4,5-b]pyridine Derivatives as Potent and Selective BET Inhibitors for the Management of Neuropathic Pain 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 13, 页码: 8725-8744
作者:  
Chen, Xuetao;  Cao, Danyan;  Liu, Chihong;  Meng, Fanying;  Zhang, Zijian
  |  收藏  |  浏览/下载:9/0  |  提交时间:2023/10/17
Insight into Thermodynamic and Kinetic Profiles in Small-Molecule Optimization 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 16, 页码: 10809-10847
作者:  
Liu, Wei;  Jiang, Jingsheng;  Lin, Yating;  You, Qidong;  Wang, Lei
  |  收藏  |  浏览/下载:19/0  |  提交时间:2022/11/11
Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-3 期刊论文  OAI收割
MOLECULES, 2018, 卷号: 23, 期号: 7
作者:  
Mangoni, Arduino A.;  Tuccinardi, Tiziano;  Collina, Simona;  Vanden Eynde, Jean Jacques;  Munoz-Torrero, Diego
  |  收藏  |  浏览/下载:16/0  |  提交时间:2019/01/08
Design, Synthesis and Antitubercular Evaluation of New 2-amino-5-(4-(benzyloxy)benzyl)thiophene-3-carboxylic Acid Derivatives. Part 3 期刊论文  OAI收割
LETTERS IN DRUG DESIGN & DISCOVERY, 2015, 卷号: 12, 期号: 1, 页码: 29-37
作者:  
You, Qidong;  Wan, Baojie;  Lu, Xiaoyun;  Tang, Jian;  Franzblau, Scott G.
  |  收藏  |  浏览/下载:14/0  |  提交时间:2018/12/13
Design, Synthesis and Antitubercular Evaluation of New 2-amino-5-(4-(benzyloxy)benzyl)thiophene-3-carboxylic Acid Derivatives. Part 3 期刊论文  OAI收割
LETTERS IN DRUG DESIGN & DISCOVERY, 2015, 卷号: 12, 期号: 1, 页码: 29-37
Lu, Xiaoyun; Tang, Jian; You, Qidong; Wan, Baojie; Franzblau, Scott G.
收藏  |  浏览/下载:15/0  |  提交时间:2016/12/16
Direct Glycosylation of Bioactive Small Molecules with Glycosyl Iodide and Strained Olefin as Acid Scavenger 期刊论文  OAI收割
JOURNAL OF ORGANIC CHEMISTRY, 2014, 卷号: 79, 期号: 3, 页码: 1100-1110
作者:  
Gu, Xiangying;  Chen, Lin;  Wang, Xin;  Liu, Xiao;  You, Qidong
  |  收藏  |  浏览/下载:13/0  |  提交时间:2019/01/08
Strained olefin enables triflic anhydride mediated direct dehydrative glycosylation 期刊论文  OAI收割
ORGANIC & BIOMOLECULAR CHEMISTRY, 2014, 卷号: 12, 期号: 48, 页码: 9781-9785
作者:  
Chen, Guohua;  Yin, Qiang;  Yin, Jian;  Gu, Xiangying;  Liu, Xiao
  |  收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
BioNMR in Drug Design 期刊论文  OAI收割
Journal of China Pharmaceutical University, 2004, 卷号: 35, 期号: 5, 页码: 387-392
作者:  
Lin Kejiang;  You Qidong;  Lin Donghai;  Wu Wutong;  Ye Boping
  |  收藏  |  浏览/下载:16/0  |  提交时间:2019/01/08