机构

• 上海药物研究所 [11]
• 中国科学院大学 [9]
• 上海营养与健康研究所 [2]
• 生物物理研究所 [1]
• 金属研究所 [1]
• 深圳先进技术研究院 [1]
• 更多

采集方式

• OAI收割 [25]
• iSwitch采集 [9]

内容类型

• 期刊论文 [32]
• 会议论文 [2]

发表日期

• 2025 [1]
• 2024 [3]
• 2023 [1]
• 2022 [3]
• 2021 [2]
• 2020 [1]
• 更多

学科主题

• Pharmacolo... [1]
• 生物资源::功能基因... [1]

筛选

浏览/检索结果: 共34条，第1-10条 帮助 条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择题名升序题名降序提交时间升序提交时间降序作者升序作者降序发表日期升序发表日期降序 Development of novel epoxyketone macrocyclic peptidyl proteasome inhibitors through OPA-mediated one-step cyclization of unprotected peptides 期刊论文  OAI收割 BIOORGANIC CHEMISTRY, 2025, 卷号: 156, 页码: 16 作者:  Zeng, Gongruixue;  Xu, Gaoya;  Gao, Lixin;  Zheng, Xiaoli;  Chi, Xinglong   |  收藏  |  浏览/下载：9/0  |  提交时间：2025/04/01 Proteasome inhibitors  Macrocycle  Stability  Anti-cancer activities   Exploration of novel 20S proteasome activators featuring anthraquinone structures and their application in hypoxic cardiomyocyte protection 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2024, 卷号: 115, 页码: 10 作者:  Yu, Qian;  Gao, Lixin;  Xu, Linhao;  Han, Yubing;  Cao, Yu   |  收藏  |  浏览/下载：11/0  |  提交时间：2024/12/11 Discovery of the First BRD4 Second Bromodomain (BD2)-Selective Inhibitors 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 23, 页码: 21577-21616 作者:  Li, Junhua;  Hu, Qingqing;  Zhu, Run;  Dong, Ruibo;  Shen, Hui   |  收藏  |  浏览/下载：3/0  |  提交时间：2025/01/10 Proteasome activation: A novel strategy for targeting undruggable intrinsically disordered proteins 期刊论文  OAI收割 BIOORGANIC CHEMISTRY, 2024, 卷号: 145, 页码: 17 作者:  Yu, Qian;  Wang, Zheng;  Tu, Yutong;  Cao, Yu;  Zhu, Huajian   |  收藏  |  浏览/下载：15/0  |  提交时间：2024/05/07 20S proteasome  Proteasome activation  IDPs  Undruggable  Protein homeostasis   Exploration of novel four-membered-heterocycle constructed peptidyl proteasome inhibitors with improved metabolic stability for cancer treatment 期刊论文  OAI收割 BIOORGANIC CHEMISTRY, 2023, 卷号: 138, 页码: 22 作者:  Wang, Hanlin;  Wu, Zhaoxiao;  Cao, Yu;  Gao, Lixin;  Shao, Jiaan   |  收藏  |  浏览/下载：25/0  |  提交时间：2023/10/17 Metabolic stability  Four-membered heterocycles  Proteasome inhibitors  Multiple myeloma   Discovery and prospecting potential of volcanic beryllium mineralization in Kulongshan, northern Hebei Province. 期刊论文  OAI收割 ACTA PETROLOGICA SINICA, 2022, 卷号: 38, 期号: 7, 页码: 1901-1914 作者:  Chen ZhenYu;  Li ShengLi;  Li XiaoFeng;  Pan Shuo;  Zhang XingKang   |  收藏  |  浏览/下载：20/0  |  提交时间：2023/03/31 Konglongshan  Alterated rocks  Volcanic Be -U deposit  Helvite  Prospecting potential   Metabolism guided optimization of peptidomimetics as non-covalent proteasome inhibitors for cancer treatment 期刊论文  OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 233, 页码: 18 作者:  Cao, Yu;  Tu, Yutong;  Fu, Liping;  Yu, Qian;  Gao, Lixin   |  收藏  |  浏览/下载：45/0  |  提交时间：2022/06/15 Metabolism  Design  Proteasome inhibitors  Non-covalent  Multiple myeloma   Origin of pegmatitic melts from granitic magmas in the formation of the Jiajika lithium deposit in the eastern Tibetan Plateau 期刊论文  OAI收割 Journal of Asian Earth Sciences, 2022, 卷号: 222, 期号: 2022, 页码: 105147 作者:  Jingyi Deng;  Jiankang Li;  Dehui Zhang;  I-Ming Chou;  Qinggao Yan   |  收藏  |  浏览/下载：14/0  |  提交时间：2022/12/09 Encrustation patterns on brachiopods from the Middle-Upper Devonian and their paleo-environmental implications 期刊论文  OAI收割 PALAEOGEOGRAPHY PALAEOCLIMATOLOGY PALAEOECOLOGY, 2021, 卷号: 584, 页码: 16 作者:  Chang, Xiaolin;  Hou, Mingcai;  Shi, He;  Wang, Hu;  Lai, Jiankang   |  收藏  |  浏览/下载：63/0  |  提交时间：2021/12/13 Epibiont  Host brachiopods  Encruster  Paleoecology  Frasnian-Famennian event   Optimization of piperidine constructed peptidyl derivatives as proteasome inhibitors 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 29, 页码: 14 作者:  Zhao, Yanmei;  Xu, Lei;  Zhang, Jiankang;  Zhang, Mengmeng;  Lu, Jingyi   |  收藏  |  浏览/下载：39/0  |  提交时间：2021/05/24 Proteasome inhibitor  Piperidine  Peptidyl  Anti-cancer  SAR