中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [18]
昆明植物研究所 [7]
昆明动物研究所 [1]
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OAI收割 [26]
内容类型
期刊论文 [26]
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2022 [1]
2017 [3]
2016 [1]
2014 [1]
2013 [3]
2012 [5]
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Chemistry,... [3]
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Development and structure-activity relationships of tanshinones as selective 11beta-hydroxysteroid dehydrogenase 1 inhibitors
期刊论文
OAI收割
Natural products and bioprospecting, 2022, 卷号: 12, 期号: 1, 页码: 36
作者:
Deng, Xu
;
Huang, Su-Ling
;
Ren, Jian
;
Pan, Zheng-Hong
;
Shen, Yu
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2024/03/15
Metabolic syndrome
Selective 11beta-HSD1 inhibitors
Structure-activity relationships
Tanshinones
Synthesis of selective 11 beta-HSD1 inhibitors based on dammarane scaffold
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 135, 页码: 324-338
作者:
Shao, Li-Dong
;
Bao, Ying
;
Shen, Yu
;
Su, Jia
;
Leng, Ying
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2017/07/31
11 beta-HSD1 inhibitor
Hupehenols
Dammarane
SAR
Synthesis of selective 11 beta-HSD1 inhibitors based on dammarane scaffold
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 135, 页码: 324-338
作者:
Shao, Li-Dong
;
Bao, Ying
;
Shen, Yu
;
Su, Jia
;
Leng, Ying
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
11 beta-HSD1 inhibitor
Hupehenols
Dammarane
SAR
Deheiculatins A-L, 20-oxygenated cembranoids from Macaranga deheiculata
期刊论文
OAI收割
PHYTOCHEMISTRY, 2017, 卷号: 136, 页码: 101-107
作者:
Qi, Wei-Yan
;
Shen, Yu
;
Wu, Yan
;
Leng, Ying
;
Gao, Kun
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/01/08
Macaranga deheiculata
Cembrane diterpenoids
Dehiculatins
11 beta-HSD1
Two new sesquiterpenoids from cultures of the basidiomycete Tremella foliacea
期刊论文
OAI收割
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2016, 卷号: 18, 期号: 1, 页码: 46-50
作者:
Ding, Jian-Hai
;
Li, Zheng-Hui
;
Wei, Kun
;
Dong, Ze-Jun
;
Ding, Zhi-Hui
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2016/06/27
cytotoxicities
trefoliols B and C
11 beta-HSD
Tremella foliacea
Lithocarpic acids O-S, five homo-cycloartane derivatives from the cupules of Lithocarpus polystachyus
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 23, 页码: 5395-5398
作者:
Ning, Ruo-nan
;
Wang, Hong-min
;
Shen, Yu
;
Chen, Zhen-hua
;
Zhang, Ru-jun
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
24-Homo-cycloartane derivative
3,4-seco-Homo-cycloartane derivative
Lithocarpus polystachyus
Fagaceae
11 beta-HSD1
Discovery and structure-activity relationships of ent-Kaurene diterpenoids as potent and selective 11 beta-HSD1 inhibitors: Potential impact in diabetes
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 65, 页码: 403-414
作者:
Deng, Xu
;
Shen, Yu
;
Yang, Jing
;
He, Juan
;
Zhao, Yu
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2013/10/16
Ent-kaurene Diterpenoids
Structure-activity Relationship Studies
Selective 11 Beta-hsd1 Inhibitors
Urea Derivatives
Diabetes
Discovery and structure-activity relationships of ent-Kaurene diterpenoids as potent and selective 11 beta-HSD1 inhibitors: Potential impact in diabetes
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 65, 页码: 403-414
作者:
Deng, Xu
;
Shen, Yu
;
Yang, Jing
;
He, Juan
;
Zhao, Yu
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2019/01/08
ent-Kaurene diterpenoids
Structure-activity relationship studies
Selective 11 beta-HSD1 inhibitors
Urea derivatives
Diabetes
Design, synthesis and SAR of piperidyl-oxadiazoles as 11 beta-hydroxysteroid dehydrogenase 1 inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 62, 页码: 1-10
作者:
Xia, Guangxin
;
You, Xiaodi
;
Liu, Lin
;
Liu, Haiyan
;
Wang, Jianfa
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
11 beta-HSD1 inhibitor
Oxadiazole
Bioisostere
SAR
Docking
Inhibition of 11 beta-HSD1 by Tetracyclic Triterpenoids from Euphorbia kansui
期刊论文
OAI收割
MOLECULES, 2012, 卷号: 17, 期号: 10, 页码: 11826-11838
作者:
Guo, Jie
;
Zhou, Li-Yan
;
He, Hong-Ping
;
Leng, Ying
;
Yang, Zhen
收藏
  |  
浏览/下载:63/0
  |  
提交时间:2013/01/22
tetracyclic triterpenoids
Euphorbia kansui
inhibition of 11 beta-HSD1
docking