中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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Design, Synthesis, and Biological Evaluation of Orally Bioavailable CHK1 Inhibitors Active against Acute Myeloid Leukemia 期刊论文  OAI收割
CHEMMEDCHEM, 2021, 页码: 12
作者:  
Jin, Tingting;  Wang, Peipei;  Long, Xiubing;  Jiang, Kailong;  Song, Pinrao
  |  收藏  |  浏览/下载:137/0  |  提交时间:2021/05/24
Discovery of (R)-5-((5-(1-methyl-1H-pyrazol-4-yl)-4-(methylamino) pyrimidin-2-yl)amino)-3-(piperidin-3-yloxy)picolinonitrile, a novel CHK1 inhibitor for hematologic malignancies 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 173, 页码: 44-62
作者:  
Tong, Lexian;  Song, Pinrao;  Jiang, Kailong;  Xu, Lei;  Jin, Tingting
  |  收藏  |  浏览/下载:31/0  |  提交时间:2020/07/01
Design, synthesis and biological evaluation of thienopyridinones as Chk1 inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2014, 卷号: 22, 期号: 17, 页码: 4882-4892
作者:  
Song, Pinrao;  Peng, Peng;  Han, Mengmeng;  Cao, Xianchao;  Ma, Xiaodong
  |  收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
Proteasome-dependent degradation of Chk1 kinase induced by the topoisomerase II inhibitor R16 contributes to its anticancer activity 期刊论文  OAI收割
CANCER BIOLOGY & THERAPY, 2008, 卷号: 7, 期号: 11, 页码: 1726-1731
作者:  
Feng, Jian-Ming;  Zhu, Hong;  Zhang, Xiao-Wei;  Ding, Jian;  Miao, Ze-Hong
  |  收藏  |  浏览/下载:27/0  |  提交时间:2019/01/08