中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [18]
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OAI收割 [35]
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期刊论文 [34]
会议论文 [1]
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Bioassay-guided isolation of α-Glucosidase inhibitory constituents from Hypericum sampsonii
期刊论文
OAI收割
CHINESE JOURNAL OF NATURAL MEDICINES, 2023, 卷号: 21, 期号: 6, 页码: 443-453
作者:
Tao,Linlan
;
Xu,Shuangyu
;
Zhang,Zizhen
;
Li,Yanan
;
Yang,Jue
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2024/07/22
Hypericum sampsonii
Chemical constituents
Structure elucidation
alpha-Glucosidase
Molecular docking
POLYCYCLIC POLYPRENYLATED ACYLPHLOROGLUCINOLS
POTENT INHIBITORS
SPECTROSCOPY
DERIVATIVES
CHEMISTRY
AMYLASE
ROOTS
Meroterpenoids and alkaloids from Ganoderma australe
期刊论文
OAI收割
NATURAL PRODUCT RESEARCH, 2021, 卷号: 35, 期号: 19, 页码: 3226-3232
作者:
Zhang,Jiao-Jiao
;
Dong,Yun
;
Qin,Fu-Ying
;
Yan,Yong-Ming
;
Cheng,Yong-Xian
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2022/04/02
Ganoderma australe
meroterpenoids
alkaloids
neuroprotection
LUCIDUM
INHIBITORS
EXTRACT
POTENT
Discovery and Biological evaluation of pyrimido[4,5-d] pyrimidine-2,4(1H, 3H)-dione derivatives as potent Bruton's tyrosine kinase inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 15, 页码: 3390-3395
作者:
Diao, Yanyan
;
Fang, Xiaoyu
;
Song, Peiran
;
Lai, Mengzhen
;
Tong, Linjiang
  |  
收藏
  |  
浏览/下载:58/0
  |  
提交时间:2020/07/01
Bruton's tyrosine kinase
B-cell malignancies
Potent inhibitors
Structure-activity relationship
Cellular activities
A novel non-enzymatic hydrolytic probe for dipeptidyl peptidase IV specific recognition and imaging
期刊论文
OAI收割
CHEMICAL COMMUNICATIONS, 2018, 卷号: 54, 期号: 63, 页码: 8773-8776
作者:
Sun, Shan
;
Wu, Aiguo
;
Xing, Jie
;
Gong, Qiuyu
;
Zhang, Renshuai
  |  
收藏
  |  
浏览/下载:223/0
  |  
提交时间:2018/12/04
Fibroblast Activation Protein
Fluorescence Probes
Inhibitors
Cells
Mechanisms
Enzyme
Potent
Vitro
Dpp4
Vivo
The development of a complementary pathway for the synthesis of aliskiren
期刊论文
OAI收割
organic & biomolecular chemistry, 2015, 卷号: 13, 期号: 4, 页码: 1133-1140
作者:
Li,Le-Le
;
Ding,Jin-Ying
;
Gao,Lian-Xun
;
Han,Fu-She
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2016/05/20
RENIN INHIBITOR ALISKIREN
ORALLY-ACTIVE INHIBITORS
OLEFIN CROSS-METATHESIS
CONVERGENT SYNTHESIS
RUTHENIUM CATALYSTS
OXIDATIVE CLEAVAGE
POTENT
CONVERSION
ALCOHOLS
KETONES
5氨基吡唑及5氨基三唑类成纤维细胞生长因子受体激酶抑制剂的设计合成
期刊论文
OAI收割
有机化学, 2015, 卷号: 35, 期号: 9, 页码: 1939
作者:
董潜
;
彭霞
;
王雯
;
戴阳
;
赵伟利
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2020/07/01
SELECTIVE INHIBITOR
ACTIVATING MUTATIONS
TYROSINE KINASE
CANCER
POTENT
CARCINOMA
FAMILY
FGFR2
5-aminopyrazole
5-amino-1,2,3-triazole
FGFR inhibitors
anti-tumor agent
Design, Synthesis and Biological Evaluation of Novel Benzothiazole Derivatives Bearing Semicarbazone Moiety as Antitumor Agents
期刊论文
OAI收割
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 6, 页码: 958-963
作者:
Ma Junjie
;
Hu Gang
;
Xie Lijun
;
Chen Lei
;
Xu Boxuan
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2021/02/02
POTENT
INHIBITORS
ONCRASIN-1
DISCOVERY
Benzothiazole
Semicarbazone
Antitumor activity
Design, Synthesis and Biological Evaluation of Novel Benzothiazole Derivatives Bearing Semicarbazone Moiety as Antitumor Agents
期刊论文
OAI收割
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 6, 页码: 958-963
作者:
Ma Junjie
;
Hu Gang
;
Xie Lijun
;
Chen Lei
;
Xu Boxuan
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2021/02/02
POTENT
INHIBITORS
ONCRASIN-1
DISCOVERY
Benzothiazole
Semicarbazone
Antitumor activity
Synthesis and antiproliferative activity of novel 4-substituted-phenoxy-benzamide derivatives
期刊论文
OAI收割
CHINESE CHEMICAL LETTERS, 2015, 卷号: 26, 期号: 10, 页码: 1307-1310
作者:
Sun ChiYu
;
Li YangSheng
;
Shi AiLong
;
Li YaFei
;
Cao RuiFang
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2021/02/02
HEDGEHOG SIGNALING PATHWAY
BASAL-CELL CARCINOMA
INHIBITORS
DISCOVERY
DESIGN
ANTAGONISTS
IDENTIFICATION
VISMODEGIB
CANCER
POTENT
Aryl cycloaliphatic amine
Antiproliferative activity
Hedgehog signaling
Synthesis and antiproliferative activity of novel 4-substituted-phenoxy-benzamide derivatives
期刊论文
OAI收割
CHINESE CHEMICAL LETTERS, 2015, 卷号: 26, 期号: 10, 页码: 1307-1310
作者:
Sun ChiYu
;
Li YangSheng
;
Shi AiLong
;
Li YaFei
;
Cao RuiFang
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2021/02/02
HEDGEHOG SIGNALING PATHWAY
BASAL-CELL CARCINOMA
INHIBITORS
DISCOVERY
DESIGN
ANTAGONISTS
IDENTIFICATION
VISMODEGIB
CANCER
POTENT
Aryl cycloaliphatic amine
Antiproliferative activity
Hedgehog signaling