中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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期刊论文 [250]
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Pharmacological characterizationof tachykinin tetrabranched derivatives
期刊论文
OAI收割
出版物, 3111, 期号: 0, 页码: 1-36
作者:
Chiara Ruzza
;
Anna Rizzi
;
Davide Malfacini
;
Maria Camilla Cerlesi
;
Federica Ferrari
  |  
收藏
  |  
浏览/下载:249/0
  |  
提交时间:2017/07/24
Tachykinins
Substance p
Pwt2-sp
Nk1 Receptor
Calcium Mobilization
Bioluminescence Resonance Energy Transfer
Guinea Pig Ileum
Rat Urinary Bladder
Nociceptive Behaviour Induced By Spinal Substance p
Mice
The Tyrosine Kinase Inhibitor Bafetinib Inhibits PAR2-induced Activation of TRPV4 In Vitro and Pain In Vivo1
期刊论文
OAI收割
出版物, 2111, 页码: 1-44
作者:
1M S Grace
;
T Lieu
;
B Darby
;
F C Abogadie
;
N Veldhuis N W Bunnett
;
P McIntyre
  |  
收藏
  |  
浏览/下载:295/0
  |  
提交时间:2017/07/24
Transient Receptor Potential Ion Channel
Trpv4
Protease Activated Receptor
Par2
Pain
Tyrosine Kinase
Bafetinib
Adapter protein 2-modulated μ-opioid receptor trafficking in paraventricular thalamus contributes to fentanyl contextual addiction memory in mice
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 9
作者:
Li, Yu-jie
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2026/01/28
fentanyl
contextual addiction memory
paraventricular thalamus
mu-opioid receptor trafficking
Ap2a1
Discovery and characterization of a novel HIF-2α agonist for the treatment of CKD-related renal anemia
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 14
作者:
Chu, Shu-qing
;
Chen, Yi-jie
;
Yang, Rui-rui
;
Teng, Dan
;
Zhou, Gui-zhen
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/12/04
anemia
HIF-2 alpha
aryl hydrocarbon receptor nuclear translocator
erythropoietin
amide thiazole AT-1
Molidustat
M1002
Discovery of novel TLR2 antagonists as anti-inflammatory agents
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2025, 卷号: 164, 页码: 15
作者:
Tang, Xuehang
;
Qi, Luyao
;
Li, Yingxia
;
Tang, Wei
;
Zhang, Wei
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/12/04
Toll-like receptor 2
TLR2 antagonists
Structure-activity relationship
Anti-inflammatory
Molecular basis for ligand recognition and receptor activation of the prostaglandin D2 receptor DP1
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2025, 卷号: 122, 期号: 22, 页码: 11
作者:
Xu, Jiuyin
;
Wu, Yanli
;
Xu, Youwei
;
Li, Yang
;
He, Xinheng
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2025/08/20
prostaglandin D2 receptor 1
receptor activation
drug design
Structural insights into the activation of the human prostaglandin E
2
receptor EP1 subtype by prostaglandin E
2
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2025, 卷号: 122, 期号: 20, 页码: 12
作者:
Meng, Xue
;
Li, Yang
;
Xu, Jiuyin
;
Wu, Kai
;
Hu, Wen
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2025/07/25
prostaglandin E2
EP1
receptor activation
PGE2 selectivity
Structural basis of the cysteinyl leukotriene receptor type 2 activation by LTD4
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2025, 卷号: 122, 期号: 15, 页码: 9
作者:
Jiang, Mengting
;
Xu, Youwei
;
Luan, Xiaodong
;
Wu, Kai
;
Li, Zhen
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2025/06/23
G protein-coupled receptor
cryo-electron microscopy
cysteinyl leukotriene receptor2
activation mechanism
G alpha q protein coupling
Molecular basis of lipid and ligand regulation of prostaglandin receptor DP2
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2024, 卷号: 121, 期号: 51, 页码: 12
作者:
  |  
收藏
  |  
浏览/下载:86/0
  |  
提交时间:2025/02/28
prostaglandin receptor
DP2
lipid regulation
receptor activation
signal bias
Pyrotinib plus capecitabine for patients with HER2-positive metastatic breast cancer and brain metastases (PERMEATE trial): overall survival results from a multicenter, single-arm, two-cohort, phase 2 trial
期刊论文
OAI收割
ECLINICALMEDICINE, 2024, 卷号: 76
作者:
Yan, Min
;
Ouyang, Quchang
;
Sun, Tao
;
Niu, Limin
;
Yang, Jin
  |  
收藏
  |  
浏览/下载:62/0
  |  
提交时间:2024/11/20
Pyrotinib
Human epidermal growth factor receptor 2
Breast cancer
Brain metastases
Overall survival