中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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大连化学物理研究所 [76]
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Structural insights into the activation of the human prostaglandin E
2
receptor EP1 subtype by prostaglandin E
2
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2025, 卷号: 122, 期号: 20, 页码: 12
作者:
Meng, Xue
;
Li, Yang
;
Xu, Jiuyin
;
Wu, Kai
;
Hu, Wen
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2025/07/25
prostaglandin E2
EP1
receptor activation
PGE2 selectivity
Discovery of a potential hematologic malignancies therapy: Selective and potent HDAC7 PROTAC degrader targeting non-enzymatic function
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 3, 页码: 1659-1679
作者:
Jin, Yuheng
;
Qi, Xuxin
;
Yu, Xiaoli
;
Cheng, Xirui
;
Chen, Boya
  |  
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2025/06/23
HDAC7
PROTAC
Selectivity
Hematologic malignancies
Non-enzymatic function
Metal incorporated into magnetic hybrid covalent organic framework for high selective uptake of scandium ion
期刊论文
OAI收割
SEPARATION AND PURIFICATION TECHNOLOGY, 2025, 卷号: 355, 页码: 15
作者:
Pittman, Aaron S.
;
Cao, Yan
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/11/20
Covalent organic framework
Red mud
Rare-earth elements
Scandium
Selectivity
Metal-incorporation
A patent review of BRD4 inhibitors (2020-present)
期刊论文
OAI收割
EXPERT OPINION ON THERAPEUTIC PATENTS, 2025, 页码: 16
作者:
Chen, Yanfang
;
Zhou, Huanmin
;
Yu, Jiamin
;
Gao, Jing
;
Xue, Shengyu
  |  
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2025/04/01
BET
BRD4
inhibitor
cancer treatment
selectivity
Molecular simulation on Cs, Rb retention in Na/K-montmorillonite interlayer coupling clay swelling/collapse
期刊论文
OAI收割
APPLIED GEOCHEMISTRY, 2025, 卷号: 178, 页码: 15
作者:
Zhou, Mengzi
;
Lu, Xiancai
;
Chen, Meng
;
Li, Qin
;
Wang, Kai
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2025/04/01
Cs
Rb
Retention
Cation selectivity
Montmorillonite
Molecular simulation
Design, synthesis and pharmacological evaluation of 1,2,3,4-tetrahydrobenzofuro[2,3-c] pyridine derivatives as p21-activated kinase 4 inhibitors for treatment of pancreatic cancer
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 1, 页码: 438-466
作者:
Li, Yang
;
Fang, Yan
;
Chen, Xiaoyu
;
Tong, Linjiang
;
Feng, Fang
  |  
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2025/04/01
P21-activated kinase 4
Tetrahydrobenzofuro[2
3-c]pyridine
Structure-activity relationship
Allosteric inhibitor
Pharmacokinetics properties
Kinase selectivity
Pancreatic cancer
Immune infiltration
Visible Light-Switchable Lattice Oxygen Sites for Selective C-H and C(O)-C Bond Electrooxidation
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2024, 卷号: 63, 期号: 49, 页码: 11
作者:
Wang, Keping
;
Huang, Jinshu
;
Hu, Jinguang
;
Wu, Mei
;
Liao, Yuhe
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/11/20
Biomass conversion
C(O)-C bond cleavage
electrocatalytic oxidation
lattice-oxygen
selectivity control
Enhancement of ethylene selectivity in chemical looping oxidative dehydrogenation of ethane using manganese-based redox catalysts supported on HY zeolite
期刊论文
OAI收割
APPLIED CATALYSIS A-GENERAL, 2024, 卷号: 687, 页码: 11
作者:
Mao, Min
;
Wang, Xuemei
;
Zhou, Yuchao
;
Chen, Haitao
;
Yu, Xiang
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/11/20
Mn-based catalyst
Zeolite
Ethane oxidative dehydrogenation
Ethylene selectivity
Lewis acid
Design and synthesis of pyridazin-4-one derivatives as necroptosis inhibitors
期刊论文
OAI收割
ARCHIV DER PHARMAZIE, 2024, 页码: 16
作者:
An, Yuxiang
;
Peng, Xia
;
Wang, Tianchen
;
Liu, Kaiyuan
;
Feng, Dazhi
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2024/12/25
inhibitor
pharmacokinetic study
pyridazin-4-one
receptor-interacting protein kinase 1
selectivity
Selective ligand recognition and activation of somatostatin receptors SSTR1 and SSTR3
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2024, 卷号: 121, 期号: 41, 页码: 11
作者:
Wang, Yujue
;
Xu, Youwei
;
Wang, Yue
;
Zhang, Jie
;
Chen, Lan
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2024/12/11
GPCR
somatostatin receptors
ligand selectivity
neuroendocrine tumor
|cryo-EM