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Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共8条,第1-8条 帮助

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Discovery of a 1,6-naphthyridin-4-one-based AXL inhibitor with improved pharmacokinetics and enhanced in vivo antitumor efficacy 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 17
作者:  
Lan, Yaohan;  Peng, Xia;  Ji, Yinchun;  Su, Yi;  Duan, Wenhu
  |  收藏  |  浏览/下载:30/0  |  提交时间:2024/02/27
Discovery of pyrido[4,3-d]pyrimidinone derivatives as novel Wee1 inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 87, 页码: 12
作者:  
Ye, Qingqing;  Ma, Jingkun;  Wang, Peipei;  Wang, Chang;  Sun, Mei
  |  收藏  |  浏览/下载:20/0  |  提交时间:2023/10/17
Design, synthesis and biological evaluation of novel dihydrobenzodioxine derivatives as HBV capsid protein inhibitors 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 128, 页码: 12
作者:  
Liu, Linyue;  Li, Chuanju;  Xie, Yong;  Zhang, Lei;  Chen, Yunfu
  |  收藏  |  浏览/下载:19/0  |  提交时间:2023/10/17
Design, synthesis and pharmacological evaluation of bicyclic and tetracyclic pyridopyrimidinone analogues as new KRAS(G12C) inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 213, 页码: 17
作者:  
Xiao, Xuanzheng;  Lai, Mengzhen;  Song, Zilan;  Geng, Meiyu;  Ding, Jian
  |  收藏  |  浏览/下载:57/0  |  提交时间:2021/05/24
Discovery and synthesis of 6,7,8,9-tetrahydro-5H-pyrido[4,3-c]azepin-5-one-based novel chemotype CCR2 antagonists via scaffold hopping strategy 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 12, 页码: 3559-3572
作者:  
Qin, Li-Huai;  Wang, Zhi-Long;  Xie, Xin;  Long, Ya-Qiu
  |  收藏  |  浏览/下载:43/0  |  提交时间:2019/01/08
Discovery of alkyl bis(oxy)dibenzimidamide derivatives as novel protein arginine methyltransferase 1 (PRMT1) inhibitors 期刊论文  OAI收割
CHEMICAL BIOLOGY & DRUG DESIGN, 2017, 卷号: 90, 期号: 6, 页码: 1260-1270
作者:  
Zhang, Wei-yao;  Lu, Wen-chao;  Jiang, Hao;  Lv, Zheng-bing;  Xie, Yi-qian
  |  收藏  |  浏览/下载:37/0  |  提交时间:2019/01/08
Design, synthesis, biological evaluation, and comparative docking study of 1,2,4-triazolones as CB1 receptor selective antagonists 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 74, 页码: 73-84
作者:  
Han, Shuang;  Zhang, Fei-Fei;  Xie, Xin;  Chen, Jian-Zhong
  |  收藏  |  浏览/下载:29/0  |  提交时间:2019/01/08
ScafBank: a public comprehensive Scaffold database to support molecular hopping 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2009, 卷号: 30, 期号: 2, 页码: 251-258
作者:  
Yan, Bi-bo;  Xue, Meng-zhu;  Xiong, Bing;  Liu, Ke;  Hu, Ding-yu
  |  收藏  |  浏览/下载:21/0  |  提交时间:2019/01/08
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