中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [4]
采集方式
OAI收割 [4]
内容类型
期刊论文 [4]
发表日期
2021 [1]
2014 [2]
2012 [1]
学科主题
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Discovery of a series of 1H-pyrrolo[2,3-b]pyridine compounds as potent TNIK inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2021, 卷号: 33, 页码: 127749
作者:
Yang, Bowen
;
Wu, Qian
;
Huan, Xiajuan
;
Wang, Yingqing
;
Sun, Yin
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2024/03/21
TNIK inhibitor
1H-pyrrolo[2,3-b]pyridine
IL-2 secretion inhibitory
Benzimidazole derivative, BM601, a novel inhibitor of hepatitis B virus and HBsAg secretion
期刊论文
OAI收割
ANTIVIRAL RESEARCH, 2014, 卷号: 107, 页码: 6-15
作者:
Xu, Yi-Bin
;
Yang, Li
;
Wang, Gui-Feng
;
Tong, Xian-Kun
;
Wang, Ya-Juan
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2019/01/08
Anti-hepatitis B virus compound
Benzimidazole derivative
Secretion inhibitor
shr3824anovelselectiveinhibitorofrenalsodiumglucosecotransporter2exhibitsantidiabeticefficacyinrodentmodels
期刊论文
OAI收割
actapharmacologicasinica, 2014, 卷号: 35, 期号: 5, 页码: 613
作者:
Yan Pangke
;
Zhang Lina
;
Feng Ying
;
Qu Hui
;
Qin Li
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2020/07/01
BETA-CELL DIFFERENTIATION
IMPROVES GLYCEMIC CONTROL
TYPE-2 DIABETES-MELLITUS
CHRONIC HYPERGLYCEMIA
INSULIN-SECRETION
SGLT-2 INHIBITOR
SKELETAL-MUSCLE
RATS
DAPAGLIFLOZIN
EMPAGLIFLOZIN
sodium glucose cotransporter 2 (SGLT2)
SHR3824
dapagliflozin
type 2 diabetes mellitus
blood glucose
insulin sensitivity
beta-cell function
acuteandchronicadministrationofshr117887anovelandspecificdipeptidylpeptidase4inhibitorimprovesmetaboliccontrolindiabeticrodentmodels
期刊论文
OAI收割
actapharmacologicasinica, 2012, 卷号: 33, 期号: 8, 页码: 1013
作者:
Liu Xiao
;
Zhang Lina
;
Ying Feng
;
Zhang Lei
;
Qu Hui
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2020/07/01
GLUCAGON-LIKE PEPTIDE-1
IMPROVED GLUCOSE-TOLERANCE
DRUG-NAIVE PATIENTS
BETA-CELL FUNCTION
GLYCEMIC CONTROL
IV INHIBITOR
INSULIN-SECRETION
DOUBLE-BLIND
ZUCKER RATS
EFFICACY
SHR117887
vildagliptin (LAF237)
dipeptidyl peptidase-4 (DPP-4)
type 2 diabetes mellitus
glucagon-like peptide-1 (GLP-1)
insulin
beta-cells