中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [97]
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期刊论文 [201]
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DRAK2 suppresses autophagy by phosphorylating ULK1 at Ser
56
to diminish pancreatic β cell function upon overnutrition
期刊论文
OAI收割
SCIENCE TRANSLATIONAL MEDICINE, 2024, 卷号: 16, 期号: 733, 页码: 16
作者:
Lu, Yuting
;
Xu, Junyu
;
Li, Yufeng
;
Wang, Ruoran
;
Dai, Chengqiu
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2024/03/13
Discovery and exploration of novel somatostatin receptor subtype 5 (SSTR5) antagonists for the treatment of cholesterol gallstones
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 264, 页码: 16
作者:
Han, Fanghui
;
Zhao, Tingting
;
Zhang, Yanglong
;
Yun, Ying
;
Xu, Yuanyuan
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2024/02/19
SSTR5 antagonist
Gallbladder emptying
Cholesterol gallstones
Obesity induced disruption on diurnal rhythm of insulin sensitivity via gut microbiome-bile acid metabolism
期刊论文
OAI收割
BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR AND CELL BIOLOGY OF LIPIDS, 2024, 卷号: 1869, 期号: 1, 页码: 13
作者:
Guo, Xiaozhen
;
Wang, Jiawen
;
Xu, Hualing
;
Wang, Yangyang
;
Cao, Yutang
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2024/01/16
Diurnal rhythm
Insulin sensitivity
Obesity
Gut microbiota
Ursodeoxycholic acid
Hepatic glucuronyl C5-epimerase combats obesity by stabilising GDF15
期刊论文
OAI收割
JOURNAL OF HEPATOLOGY, 2023, 卷号: 79, 期号: 3, 页码: 14
作者:
He, Fei
;
Jiang, Haowen
;
Peng, Chang
;
Wang, Tingting
;
Xiao, Rongrong
  |  
收藏
  |  
浏览/下载:61/0
  |  
提交时间:2023/10/17
Glucuronyl C5-epimerase
Growth differentiation factor-15
Obesity
Energy expenditure
Ubiquitination
Discovery of Novel 5,6-Dihydro-1,2,4-triazine Derivatives as Efficacious Glucagon-Like Peptide-1 Receptor Agonists
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 23
作者:
Chen, Lili
;
Yun, Ying
;
Guo, Shimeng
;
Wang, Xiaoyan
;
Xiong, Muya
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/10/17
Discovery of orally effective and safe GPR40 agonists by incorporating a chiral, rigid and polar sulfoxide into 8-position to the carboxylic acid
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 251, 页码: 115267
作者:
Chen, Cheng
;
Guo, Shi-Meng
;
Sun, Yuanjun
;
Li, He
;
Hu, Nan
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/03/27
GPR40
Glucose-stimulated insulin secretion
Type 2 diabetes mellitus
Lipophilicity
Liver safety
Three-in-one pharmacophore
2-(phenylsulfinyl)acetic acid
Novel Regulations of Insulin Secretion and Body Energy Expenditure by Selenoproteins
影音
OAI收割
2023,
作者:
Lei XG(雷新根)
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2023/02/01
创新论坛
所庆50周年系列活动
365期
14-Deoxygarcinol improves insulin sensitivity in high-fat diet-induced obese mice via mitigating NF-κB/Sirtuin 2-NLRP3-mediated adipose tissue remodeling
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 卷号: 44, 期号: 2, 页码: 434
作者:
Chen Jiali
;
Feng Zheling
;
Zhou Fei
;
Lou Ruohan
;
Peng Cheng
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/05/22
14-deoxygarcinol
adipose tissue inflammation
insulin resistance
interleukin-1β
NLRP3 inflammasome
Sirtuin 2
Roles of hydroxyeicosatetraenoic acids in diabetes (HETEs and diabetes)
期刊论文
OAI收割
BIOMEDICINE & PHARMACOTHERAPY, 2022, 卷号: 156, 页码: 13
作者:
Dong, Linyue
;
Wang, Heyao
;
Chen, Kaixian
;
Li, Yiming
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/04/10
5-HETE
12-HETE
15-HETE
20-HETE
Lipoxygenases
Diabetes
Obesity
Hepatic thyroid hormone signalling modulates glucose homeostasis through the regulation of GLP-1 production via bile acid-mediated FXR antagonism
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2022, 卷号: 13, 期号: 1, 页码: 16
作者:
Yan, Ying
;
Niu, Zhoumin
;
Sun, Chao
;
Li, Peng
;
Shen, Siyi
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2022/12/13