中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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A patent review of BRD4 inhibitors (2020-present)
期刊论文
OAI收割
EXPERT OPINION ON THERAPEUTIC PATENTS, 2025, 页码: 16
作者:
Chen, Yanfang
;
Zhou, Huanmin
;
Yu, Jiamin
;
Gao, Jing
;
Xue, Shengyu
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/04/01
BET
BRD4
inhibitor
cancer treatment
selectivity
Molecular simulation on Cs, Rb retention in Na/K-montmorillonite interlayer coupling clay swelling/collapse
期刊论文
OAI收割
APPLIED GEOCHEMISTRY, 2025, 卷号: 178, 页码: 15
作者:
Zhou, Mengzi
;
Lu, Xiancai
;
Chen, Meng
;
Li, Qin
;
Wang, Kai
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2025/04/01
Cs
Rb
Retention
Cation selectivity
Montmorillonite
Molecular simulation
Design, synthesis and pharmacological evaluation of 1,2,3,4-tetrahydrobenzofuro[2,3-c] pyridine derivatives as p21-activated kinase 4 inhibitors for treatment of pancreatic cancer
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 1, 页码: 438-466
作者:
Li, Yang
;
Fang, Yan
;
Chen, Xiaoyu
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2025/04/01
P21-activated kinase 4
Tetrahydrobenzofuro[2
3-c]pyridine
Structure-activity relationship
Allosteric inhibitor
Pharmacokinetics properties
Kinase selectivity
Pancreatic cancer
Immune infiltration
Design and synthesis of pyridazin-4-one derivatives as necroptosis inhibitors
期刊论文
OAI收割
ARCHIV DER PHARMAZIE, 2024, 页码: 16
作者:
An, Yuxiang
;
Peng, Xia
;
Wang, Tianchen
;
Liu, Kaiyuan
;
Feng, Dazhi
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/12/25
inhibitor
pharmacokinetic study
pyridazin-4-one
receptor-interacting protein kinase 1
selectivity
Selective ligand recognition and activation of somatostatin receptors SSTR1 and SSTR3
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2024, 卷号: 121, 期号: 41, 页码: 11
作者:
Wang, Yujue
;
Xu, Youwei
;
Wang, Yue
;
Zhang, Jie
;
Chen, Lan
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/12/11
GPCR
somatostatin receptors
ligand selectivity
neuroendocrine tumor
|cryo-EM
Effects of rill morphology characteristics on particle size selectivity using indoor simulation experiments with two types of soil from the Loess Plateau
期刊论文
OAI收割
JOURNAL OF SOILS AND SEDIMENTS, 2024, 卷号: N/A
作者:
Sun, Liying
;
Dai, Qingyuan
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/10/21
Rill erosion
Rill morphology
Particle selectivity
Indoor rainfall experiment
Particle size distribution
Functional characterization, structural basis, and protein engineering of a rare flavonoid 2'-O-glycosyltransferase from Scutellaria baicalensis
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2024, 卷号: 14, 期号: 8, 页码: 3746-3759
作者:
Wang, Zilong
;
Du, Xueqing
;
Ye, Guo
;
Wang, Haotian
;
Liu, Yizhan
  |  
收藏
  |  
浏览/下载:92/0
  |  
提交时间:2024/09/26
Glycosyltransferase
Regio-selectivity
Crystal structure
De-glycosylation
Catalytic mechanisms
Lithium extraction from salt lake brine by four-stage ion-distillation of flow electrode capacitive deionization
期刊论文
OAI收割
CHEMICAL ENGINEERING JOURNAL, 2024, 卷号: 493
作者:
Ma, Guangqiang
;
Zhang, Xinyuan
;
Cai, Anjiang
;
Liu, Fei
;
Wang, Lei
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/11/20
Flow-electrode capacitive deionization
Lithium extraction
Monovalent selectivity membranes
Ion-distillation
Salt lake
Design, Synthesis, and Biological Evaluation of 2,4-Diaminopyrimidine Derivatives as Potent CDK7 Inhibitors
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2024, 页码: 8
作者:
Zhang, Hualin
;
Tu, Yutong
;
Tao, Zhaofan
;
Gao, Lixin
;
Huang, Shengjie
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/08/22
CDK7 inhibitor
2,4-diaminopyrimidine
selectivity
anticancer
Structural basis for activation of somatostatin receptor 5 by cyclic neuropeptide agonists
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2024, 卷号: 121, 期号: 26, 页码: 10
作者:
Li, Jingru
;
You, Chongzhao
;
Li, Yang
;
Li, Changyao
;
Fan, Wenjia
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/08/22
SSTR5
peptide agonists
agonist selectivity
receptor activation