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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [5]
成都生物研究所 [1]
海洋研究所 [1]
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OAI收割 [7]
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期刊论文 [7]
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2021 [1]
2018 [2]
2014 [1]
2009 [1]
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Chemistry,... [1]
Oncology [1]
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Two New Cytotoxic Maytansinoids Targeting Tubulin from Trewia nudiflora
期刊论文
OAI收割
PLANTA MEDICA, 2021, 页码: 7
作者:
Lei, Chun
;
Li, Ya-Nan
;
Li, Jia-Nan
;
Zhou, Yu-Bo
;
Cui, Ming-Jun
  |  
收藏
  |  
浏览/下载:58/0
  |  
提交时间:2021/12/16
Trewia nudiflora
Euphorbiaceae
maytansinoids
cytotoxicity
tubulin polymerization
The secretome engages STAT3 to favor a cytokine-rich microenvironment in mediating acquired resistance to FGFR inhibitors
期刊论文
OAI收割
Molecular cancer therapeutics, 2018, 卷号: 145, 页码: 817-842
作者:
Wang, Xinyi
;
Ai, Jing
;
Liu, Hongyan
;
Peng, Xia
;
Chen, Hui
  |  
收藏
  |  
浏览/下载:155/0
  |  
提交时间:2019/01/08
1,4-Diaryl-2-azetidinone
Combretastatin A-4
Tubulin polymerization
Antitumor
Design, synthesis, biological evaluation and cocrystal structures with tubulin of chiral beta-lactam bridged combretastatin A-4 analogues as potent antitumor agents
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 144, 页码: 817-842
作者:
Zhou, Pengfei
;
Liang, Yuru
;
Zhang, Hao
;
Jiang, Hao
;
Feng, Kechang
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2019/01/08
1,4-Diaryl-2-azetidinone
Combretastatin A-4
Tubulin polymerization
Antitumor
Synthesis and biological evaluation of 6H-pyrido[2 ',1 ':2,3] imidazo[4,5-c] isoquinolin-5(6H)-ones as antimitotic agents and inhibitors of tubulin polymerization
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2014, 卷号: 22, 期号: 2, 页码: 848-855
作者:
Meng, Tao
;
Wang, Wei
;
Zhang, Zhixiang
;
Ma, Lanping
;
Zhang, Yongliang
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
6H-Pyrido[2 ',1 ':2,3]imidazo[4,5-c]
isoquinolin-5(6H)-ones
Antitumor agents
Inhibitors of tubulin polymerization
Colchicine binding site
A novel anti-tumor protein extracted from Meretrix meretrix Linnaeus induces cell death by increasing cell permeability and inhibiting tubulin polymerization
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF ONCOLOGY, 2009, 卷号: 35, 期号: 4, 页码: 805-812
作者:
Ning, Xuanxuan
;
Zhao, Jianmin
;
Zhang, Yuyan
;
Cao, Subing
;
Liu, Ming
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2010/12/22
Meretrix Meretrix Linnaeus
Anti-tumor Protein
Cytotoxicity
Cell Membrane Permeability
Cell Cycle
Tubulin Polymerization
Apoptosis
4 '-Alkoxyl substitution enhancing the anti-mitotic effect of 5-(3 ',4 ',5 '-substituted)anilino-4-hydroxy-8-nitroquinazolines as a novel class of anti-microtubule agents
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2006, 卷号: 16, 期号: 22, 页码: 5864-5869
作者:
Jin, Yi
;
Zhou, Zu-Yu
;
Tian, Wei
;
Yu, Qiang
;
Long, Ya-Qiu
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
quinazoline
mitosis inhibitor
tubulin polymerization
anti-microtubule agent
alkoxyl substitution
aniline
antiproliferative effect
cell cycle
tumor cells
Antiproliferative activity of Goldfussia psilostachys ethanolic extract on K562 leukemia cells
期刊论文
OAI收割
FITOTERAPIA, 2004, 卷号: 75, 期号: 7_8, 页码: 639_644
Gao, XP
;
Zhang, GL
;
Zhou, M
;
Luo, DX
;
Li, BG
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2011/07/08
Goldfussia psilostachys
cell growth inhibition
cell cycle
antimitosis
tubulin polymerization
K562 cell line