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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [40]
金属研究所 [8]
长春光学精密机械与物... [1]
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合肥物质科学研究院 [1]
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OAI收割 [51]
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期刊论文 [46]
会议论文 [5]
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2023 [1]
2022 [1]
2020 [1]
2019 [3]
2018 [2]
2017 [1]
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Biochemist... [1]
Chemistry [1]
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共51条,第1-10条
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Cytostatic Activity of Sanguinarine and a Cyanide Derivative in Human Erythroleukemia Cells Is Mediated by Suppression of c-MET/MAPK Signaling
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2023, 卷号: 24, 期号: 9, 页码: 8113
作者:
Xu,Xinglian
;
Deng,Lulu
;
Tang,Yaling
;
Li,Jiang
;
Zhong,Ting
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2024/05/09
leukemia
sanguinarine
c-MET
MAPK
PI3K/mTOR
STAT3
MET
The HDAC inhibitor GCJ-490A suppresses c-Met expression through IKK? and overcomes gefitinib resistance in non-small cell lung cancer
期刊论文
OAI收割
CANCER BIOLOGY & MEDICINE, 2022, 卷号: 19, 期号: 8, 页码: 1172-1192
作者:
He, Ting
;
Gao, Yinglei
;
Fang, Yanfen
;
Zhang, Yangming
;
Zhang, Shuwei
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2024/03/21
HDAC inhibitor
c-Met
IKK?
NSCLC
gefitinib
Synthesis of triazolotriazine derivatives as c-Met inhibitors
期刊论文
OAI收割
MOLECULAR DIVERSITY, 2020, 页码: 8
作者:
Guo, Yuting
;
Peng, Xia
;
Ji, Yinchun
;
Zhang, Yitong
;
Ding, Jian
  |  
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2020/12/24
Receptor tyrosine kinase
c-Met
Triazolotriazine
SAR
Cellular potency
SHR-A1403, a novel c-mesenchymal-epithelial transition factor (c-Met) antibody-drug conjugate, overcomes AZD9291 resistance in non-small cell lung cancer cells overexpressing c-Met
期刊论文
OAI收割
CANCER SCIENCE, 2019, 页码: 11
作者:
Tong, Mengya
;
Gao, Mingzhao
;
Xu, Yongping
;
Fu, Li
;
Li, Yun
  |  
收藏
  |  
浏览/下载:63/0
  |  
提交时间:2020/07/01
AZD9291
c-Met ADC
c-Met overexpression
resistance
SHR-A1403
SHR-A1403, a novel c-Met antibody-drug conjugate, exerts encouraging anti-tumor activity in c-Met-overexpressing models
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 7, 页码: 971-979
作者:
Yang, Chang-yong
;
Wang, Lei
;
Sun, Xing
;
Tang, Mi
;
Quan, Hai-tian
  |  
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2020/07/01
SHR-A1403
c-Met ADC
anti-tumor
patient-derived xenograft (PDX)
molecular mechanisms
Targeting slug-mediated non-canonical activation of c-Met to overcome chemo-resistance in metastatic ovarian cancer cells
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2019, 卷号: 9
-
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2020/10/26
EPITHELIAL-MESENCHYMAL TRANSITION
TUMOR-GROWTH
HETEROGENEITY
AMPLIFICATION
CONTRIBUTES
PROGRESSION
CARCINOMA
REVEALS
PATHWAY
SNAIL
Slug
c-Met
Drug resistance
Ovarian cancer
XL184
Discovery, optimization and biological evaluation for novel c-Met kinase inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 143, 页码: 491-502
作者:
Yuan, Haoliang
;
Liu, Qiufeng
;
Zhang, Li
;
Hu, Shihe
;
Chen, Tiantian
  |  
收藏
  |  
浏览/下载:65/0
  |  
提交时间:2019/01/08
c-Met
Virtual screening
Pharmacophore
X-ray crystallography
Structural optimization
Pharmacologic characterization of CT-711, a novel dual inhibitor of ALK and c-Met
期刊论文
OAI收割
AMERICAN JOURNAL OF CANCER RESEARCH, 2018, 卷号: 8, 期号: 8, 页码: 1541-1550
作者:
Wang, Lei
;
Gao, Mingzhao
;
Tong, Mengya
;
Xie, Chengying
;
He, Ye
  |  
收藏
  |  
浏览/下载:154/0
  |  
提交时间:2019/01/08
CT-711
ALK
c-Met
crizotinib
antitumor activity
pharmacokinetics
Design, Synthesis, and Biological Evaluation of the First c-Met/HDAC Inhibitors Based on Pyridazinone Derivatives
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 8, 期号: 8, 页码: 830-834
作者:
Lu, Dong
;
Yan, Juan
;
Wang, Lang
;
Liu, Hongchun
;
Zeng, Limin
  |  
收藏
  |  
浏览/下载:58/0
  |  
提交时间:2019/01/08
Dual c-Met/HDAC inhibitor
hybrid
designed multiple ligand (DML)
Design, synthesis and biological evaluation of c-Met kinase inhibitors bearing 2-oxo-1,2-dihydroquinoline scaffold
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 18, 页码: 4483-4486
作者:
Cui, Hong
;
Peng, Xia
;
Liu, Jian
;
Ma, Chunhua
;
Ji, Yinchun
  |  
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2019/01/08
c-Met
Synthesis
Antiproliferative activity